CA1129412A - Process for the preparation of imidazo-and pyrimido-pyridoindoles - Google Patents

Process for the preparation of imidazo-and pyrimido-pyridoindoles

Info

Publication number
CA1129412A
CA1129412A CA343,699A CA343699A CA1129412A CA 1129412 A CA1129412 A CA 1129412A CA 343699 A CA343699 A CA 343699A CA 1129412 A CA1129412 A CA 1129412A
Authority
CA
Canada
Prior art keywords
radical
formula
alkyl
compound
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA343,699A
Other languages
English (en)
French (fr)
Inventor
Gabor I. Koletar
Patrick Lardenois
Regis Dupont
Jonathan R. Frost
Henry Najer
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Synthelabo SA
Original Assignee
Synthelabo SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo SA filed Critical Synthelabo SA
Application granted granted Critical
Publication of CA1129412A publication Critical patent/CA1129412A/en
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CA343,699A 1979-02-05 1980-01-15 Process for the preparation of imidazo-and pyrimido-pyridoindoles Expired CA1129412A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR7902839A FR2447921A1 (fr) 1979-02-05 1979-02-05 Imidazo et pyrimido-pyrido-indoles et leur application en therapeutique
FR7902839 1979-02-05

Publications (1)

Publication Number Publication Date
CA1129412A true CA1129412A (en) 1982-08-10

Family

ID=9221588

Family Applications (1)

Application Number Title Priority Date Filing Date
CA343,699A Expired CA1129412A (en) 1979-02-05 1980-01-15 Process for the preparation of imidazo-and pyrimido-pyridoindoles

Country Status (15)

Country Link
EP (1) EP0015786B1 (no)
JP (1) JPS55104282A (no)
AT (1) ATE878T1 (no)
AU (1) AU528425B2 (no)
CA (1) CA1129412A (no)
DE (1) DE3060292D1 (no)
DK (1) DK17080A (no)
ES (1) ES487712A1 (no)
FR (1) FR2447921A1 (no)
GR (1) GR74450B (no)
IE (1) IE49629B1 (no)
IL (1) IL59127A (no)
NO (1) NO151289C (no)
PT (1) PT70697A (no)
ZA (1) ZA80241B (no)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2485538B1 (fr) * 1980-06-24 1985-01-11 Chinoin Gyogyszer Es Vegyeszet Nouveau procede de preparation d'indolo(2',3';3,4)-pyrido(1,2-b)quinazoline-5-ones
JPH0425576Y2 (no) * 1987-02-02 1992-06-18
DE3827727A1 (de) * 1988-08-16 1990-02-22 Boehringer Ingelheim Kg Anellierte tetrahydropyridinessigsaeurederivate, verfahren zu deren herstellung und verwendung solcher verbindungen zur kardioprotektion

Also Published As

Publication number Publication date
EP0015786A1 (fr) 1980-09-17
DK17080A (da) 1980-08-06
NO151289C (no) 1985-03-13
AU5462980A (en) 1980-08-14
IL59127A (en) 1983-12-30
DE3060292D1 (en) 1982-06-03
JPS616073B2 (no) 1986-02-24
ES487712A1 (es) 1980-06-16
FR2447921B1 (no) 1982-01-29
ZA80241B (en) 1980-12-31
PT70697A (fr) 1980-02-01
JPS55104282A (en) 1980-08-09
EP0015786B1 (fr) 1982-04-21
IL59127A0 (en) 1980-05-30
IE800077L (en) 1980-08-05
NO151289B (no) 1984-12-03
ATE878T1 (de) 1982-05-15
FR2447921A1 (fr) 1980-08-29
IE49629B1 (en) 1985-11-13
GR74450B (no) 1984-06-28
NO794270L (no) 1980-08-06
AU528425B2 (en) 1983-04-28

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