CA1118412A - Procede d'obtention d'amidinopenicillanoyloxyalkylcephalosporanates - Google Patents

Procede d'obtention d'amidinopenicillanoyloxyalkylcephalosporanates

Info

Publication number
CA1118412A
CA1118412A CA000272706A CA272706A CA1118412A CA 1118412 A CA1118412 A CA 1118412A CA 000272706 A CA000272706 A CA 000272706A CA 272706 A CA272706 A CA 272706A CA 1118412 A CA1118412 A CA 1118412A
Authority
CA
Canada
Prior art keywords
acid
alpha
formula
methyl
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA000272706A
Other languages
English (en)
Inventor
Wagn O. Godtfredsen
Ernst T. Binderup
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Leo Pharma AS
Original Assignee
Leo Pharmaceutical Products Ltd AS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Leo Pharmaceutical Products Ltd AS filed Critical Leo Pharmaceutical Products Ltd AS
Application granted granted Critical
Publication of CA1118412A publication Critical patent/CA1118412A/fr
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Cephalosporin Compounds (AREA)
CA000272706A 1976-02-25 1977-02-25 Procede d'obtention d'amidinopenicillanoyloxyalkylcephalosporanates Expired CA1118412A (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB7472/76 1976-02-25
GB7472/76A GB1573614A (en) 1976-02-25 1976-02-25 Amidinopenicillanoyloxyalkyl cephalosporanates

Publications (1)

Publication Number Publication Date
CA1118412A true CA1118412A (fr) 1982-02-16

Family

ID=9833766

Family Applications (1)

Application Number Title Priority Date Filing Date
CA000272706A Expired CA1118412A (fr) 1976-02-25 1977-02-25 Procede d'obtention d'amidinopenicillanoyloxyalkylcephalosporanates

Country Status (6)

Country Link
JP (1) JPS52102295A (fr)
CA (1) CA1118412A (fr)
DE (1) DE2707577A1 (fr)
DK (1) DK77577A (fr)
FR (1) FR2342294A1 (fr)
GB (1) GB1573614A (fr)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4322347A (en) * 1978-04-03 1982-03-30 Bristol-Myers Company 2-Carbamoyloxymethyl-penicillin derivatives
IE49881B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd B-lactam intermediates
DE3051044C2 (fr) * 1979-06-19 1989-03-30 Leo Pharmaceutical Products Ltd. A/S (Loevens Kemiske Fabrik Produktionsaktieselskab), Ballerup, Dk
FR2520362B1 (fr) * 1982-01-26 1986-04-11 Leo Pharm Prod Ltd Nouveaux composes de type b-lactame, y compris leurs sels formes avec des acides ou des bases acceptables en pharmacie, procedes pour produire ces composes, medicaments les contenant et leur utilisation pour combattre les maladies infectieuses
CN100384857C (zh) * 2003-11-28 2008-04-30 浙江永宁制药厂 耐β-内酰胺酶的头孢菌素酯化合物及其盐

Also Published As

Publication number Publication date
JPS52102295A (en) 1977-08-27
DE2707577A1 (de) 1977-09-01
FR2342294A1 (fr) 1977-09-23
DK77577A (da) 1977-08-26
FR2342294B1 (fr) 1980-07-18
GB1573614A (en) 1980-08-28

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Legal Events

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