CA1062654A - Process for preparing 3-methylene cephalosporins - Google Patents

Process for preparing 3-methylene cephalosporins

Info

Publication number
CA1062654A
CA1062654A CA271,660A CA271660A CA1062654A CA 1062654 A CA1062654 A CA 1062654A CA 271660 A CA271660 A CA 271660A CA 1062654 A CA1062654 A CA 1062654A
Authority
CA
Canada
Prior art keywords
formula
azetidin
hydrogen
methylene
cephalosporins
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA271,660A
Other languages
English (en)
French (fr)
Inventor
Eric M. Gordon
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
ER Squibb and Sons LLC
Original Assignee
ER Squibb and Sons LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ER Squibb and Sons LLC filed Critical ER Squibb and Sons LLC
Application granted granted Critical
Publication of CA1062654A publication Critical patent/CA1062654A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/02—Preparation
    • C07D501/08—Preparation by forming the ring or condensed ring systems
    • C07D501/10—Preparation by forming the ring or condensed ring systems from compounds containing the penicillin ring system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • Molecular Biology (AREA)
  • Cephalosporin Compounds (AREA)
CA271,660A 1976-03-15 1977-02-14 Process for preparing 3-methylene cephalosporins Expired CA1062654A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/666,989 US4375397A (en) 1976-03-15 1976-03-15 Process for preparing 3-methylene cephalosporins

Publications (1)

Publication Number Publication Date
CA1062654A true CA1062654A (en) 1979-09-18

Family

ID=24676364

Family Applications (1)

Application Number Title Priority Date Filing Date
CA271,660A Expired CA1062654A (en) 1976-03-15 1977-02-14 Process for preparing 3-methylene cephalosporins

Country Status (12)

Country Link
US (1) US4375397A (OSRAM)
JP (1) JPS52111592A (OSRAM)
BE (1) BE852469A (OSRAM)
CA (1) CA1062654A (OSRAM)
CH (1) CH597239A5 (OSRAM)
DE (1) DE2709529C2 (OSRAM)
DK (1) DK155008C (OSRAM)
FR (1) FR2344561A1 (OSRAM)
GB (1) GB1579296A (OSRAM)
HU (1) HU172544B (OSRAM)
IE (1) IE45116B1 (OSRAM)
NL (1) NL7702342A (OSRAM)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4190724A (en) * 1978-11-13 1980-02-26 Eli Lilly And Company Process for 3-exomethylenecepham sulfoxides
US4966443A (en) * 1988-02-22 1990-10-30 Fuji Photo Film Co., Ltd. Light beam scanner
JPH023451U (OSRAM) * 1988-06-16 1990-01-10

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2265798C2 (de) * 1971-06-24 1985-09-26 Fujisawa Pharmaceutical Co., Ltd., Osaka Verfahren zur Herstellung von Oxoazetidin-Derivaten
US3898142A (en) * 1972-03-24 1975-08-05 Schering Corp Photolytic cyclization of an amino-keto acylate

Also Published As

Publication number Publication date
BE852469A (fr) 1977-09-15
DE2709529C2 (de) 1986-01-02
NL7702342A (nl) 1977-09-19
DE2709529A1 (de) 1977-09-22
IE45116B1 (en) 1982-06-30
CH597239A5 (OSRAM) 1978-03-31
IE45116L (en) 1977-09-15
DK155008C (da) 1989-06-12
US4375397A (en) 1983-03-01
GB1579296A (en) 1980-11-19
JPS52111592A (en) 1977-09-19
FR2344561A1 (fr) 1977-10-14
JPS6120554B2 (OSRAM) 1986-05-22
DK106677A (da) 1977-09-16
HU172544B (hu) 1978-09-28
DK155008B (da) 1989-01-23

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