BRPI0919807A2 - compostos nitrogenosos heterocíclicos , sua preparação e seu uso como medicamentos antibacterianos - Google Patents
compostos nitrogenosos heterocíclicos , sua preparação e seu uso como medicamentos antibacterianosInfo
- Publication number
- BRPI0919807A2 BRPI0919807A2 BRPI0919807A BRPI0919807A BRPI0919807A2 BR PI0919807 A2 BRPI0919807 A2 BR PI0919807A2 BR PI0919807 A BRPI0919807 A BR PI0919807A BR PI0919807 A BRPI0919807 A BR PI0919807A BR PI0919807 A2 BRPI0919807 A2 BR PI0919807A2
- Authority
- BR
- Brazil
- Prior art keywords
- preparation
- nitrogenous compounds
- heterocyclic nitrogenous
- antibacterial medicines
- medicines
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/08—Bridged systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
- C07D487/18—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/18—Bridged systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0805602A FR2937034B1 (fr) | 2008-10-10 | 2008-10-10 | Nouveaux composes heterocycliques azotes, leur preparation et leur utilisation comme medicaments antibacteriens |
PCT/IB2009/006403 WO2010041108A1 (fr) | 2008-10-10 | 2009-07-29 | Composes heterocycliques azotes, leur preparation et leur utilisation comme medicaments antibacteriens |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0919807A2 true BRPI0919807A2 (pt) | 2015-12-22 |
Family
ID=40530144
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0919807A BRPI0919807A2 (pt) | 2008-10-10 | 2009-07-29 | compostos nitrogenosos heterocíclicos , sua preparação e seu uso como medicamentos antibacterianos |
Country Status (19)
Country | Link |
---|---|
US (1) | US8148366B2 (pt) |
EP (2) | EP2358722A1 (pt) |
JP (1) | JP2012505195A (pt) |
KR (1) | KR20110067140A (pt) |
CN (1) | CN102216307B (pt) |
AU (1) | AU2009302149A1 (pt) |
BR (1) | BRPI0919807A2 (pt) |
CA (1) | CA2739776A1 (pt) |
CL (1) | CL2011000784A1 (pt) |
CO (1) | CO6382121A2 (pt) |
EA (1) | EA201170546A1 (pt) |
EC (1) | ECSP11010962A (pt) |
FR (1) | FR2937034B1 (pt) |
IL (1) | IL212179A0 (pt) |
MX (1) | MX2011003811A (pt) |
NZ (1) | NZ592168A (pt) |
PE (1) | PE20120054A1 (pt) |
WO (1) | WO2010041108A1 (pt) |
ZA (1) | ZA201102497B (pt) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2936798B1 (fr) * | 2008-10-03 | 2012-09-28 | Novexel | Nouveaux composes heterocycliques azotes, leur preparation et leur utilisation comme medicaments antibacteriens. |
JP5666743B2 (ja) | 2011-08-27 | 2015-02-12 | ウォックハート リミテッド | 1,6−ジアザビシクロ[3,2,1]オクタン−7−オン誘導体および細菌感染の処置におけるそれらの使用 |
AR090539A1 (es) | 2012-04-02 | 2014-11-19 | Astrazeneca Ab | COMPUESTOS INHIBIDORES DE b LACTAMASA |
WO2015052682A1 (en) * | 2013-10-11 | 2015-04-16 | Wockhardt Limited | Nitrogen containing compounds and their use |
RS58429B1 (sr) | 2014-11-17 | 2019-04-30 | Entasis Therapeutics Ltd | Kombinovana terapija za lečenje rezistentnih bakterijskih infekcija |
JP2018510198A (ja) * | 2015-04-03 | 2018-04-12 | ミュタビリスMutabilis | 複素環式化合物及びそれらの細菌感染症の予防または治療のための使用 |
CN114591223A (zh) | 2016-09-16 | 2022-06-07 | 恩塔西斯治疗有限公司 | β-内酰胺酶抑制剂化合物 |
EP3301094A1 (en) | 2016-09-30 | 2018-04-04 | Mutabilis | Heterocyclic compounds and their use in preventing or treating bacterial infections |
TWI791018B (zh) | 2017-05-08 | 2023-02-01 | 美商安特西醫療公司 | 治療細菌感染之化合物及方法 |
WO2019093450A1 (ja) * | 2017-11-10 | 2019-05-16 | 塩野義製薬株式会社 | ジアザビシクロオクタン誘導体 |
Family Cites Families (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6387928B1 (en) | 1997-09-15 | 2002-05-14 | The Procter & Gamble Co. | Antimicrobial quinolones, their compositions and uses |
SK286420B6 (sk) | 1997-09-15 | 2008-09-05 | The Procter & Gamble Company | Zlúčenina so štruktúrou chinolónu, farmaceutický prostriedok s jej obsahom a jej použitie |
FR2812635B1 (fr) | 2000-08-01 | 2002-10-11 | Aventis Pharma Sa | Nouveaux composes heterocycliques, preparation et utilisation comme medicaments notamment comme anti- bacteriens |
AU3089302A (en) | 2000-12-14 | 2002-06-24 | Procter & Gamble | Antimicrobial 2-pyridones, their compositions and uses |
JP2004515548A (ja) | 2000-12-14 | 2004-05-27 | ザ プロクター アンド ギャンブル カンパニー | 抗微生物キノロン |
FR2825705B1 (fr) * | 2001-06-08 | 2005-05-20 | Aventis Pharma Sa | Nouveaux composes heterocycliques, leur preparation et leur utilisation comme medicaments, notamment comme anti-bacteriens |
FR2833596B1 (fr) | 2001-12-14 | 2005-02-18 | Aventis Pharma Sa | Procede de preparation de derives d'echinocandine |
FR2835186B1 (fr) * | 2002-01-28 | 2006-10-20 | Aventis Pharma Sa | Nouveaux composes heterocycliques, actifs comme inhibiteurs de beta-lactamases |
US6900224B2 (en) | 2002-07-31 | 2005-05-31 | The Procter & Gamble Company | Antimicrobial quinolones, their compositions and uses |
FR2844273B1 (fr) | 2002-09-05 | 2008-04-04 | Aventis Pharma Sa | Nouveaux composes heterocycliques, procede et intermediaires de preparation et utilisation comme medicament, notamment comme inhibiteurs de beta-lactamases et anti-bacteriens. |
FR2844270B1 (fr) | 2002-09-11 | 2006-05-19 | Aventis Pharma Sa | Derives de la quinolyl propyl piperidine, leur procede et intermediaires de preparation et les compositions qui les contiennent |
FR2844268B1 (fr) | 2002-09-11 | 2004-10-22 | Aventis Pharma Sa | Derives de la quinolyl propyl piperidine, leurs procedes et intermediaires de preparation et les compositions qui les contiennent |
US7439253B2 (en) | 2002-12-06 | 2008-10-21 | Novexel | Heterocyclic compounds, their preparation and their use as medicaments, in particular as antibacterials and beta-lactamase inhibitors |
FR2848210B1 (fr) * | 2002-12-06 | 2007-10-19 | Aventis Pharma Sa | Nouveaux composes heterocycliques, leur preparation et leur utilisation comme medicaments, notamment comme anti-bacteriens et inhibiteurs de beta-lactamases |
US7232833B2 (en) | 2003-03-28 | 2007-06-19 | Novexel | 4-substituted quinoline derivatives, method and intermediates for their preparation and pharmaceutical compositions containing them |
US7449481B2 (en) | 2004-04-13 | 2008-11-11 | Cephalon, Inc. | Thio-substituted biaryl-methanesulfinyl derivatives |
FR2914923B1 (fr) * | 2007-04-12 | 2013-06-14 | Novexel | Nouveaux composes heterocycliques azotes,leur preparation et leur utilisation comme medicaments antibacteriens. |
-
2008
- 2008-10-10 FR FR0805602A patent/FR2937034B1/fr not_active Expired - Fee Related
-
2009
- 2009-07-29 CA CA2739776A patent/CA2739776A1/fr not_active Abandoned
- 2009-07-29 EP EP09786084A patent/EP2358722A1/fr not_active Withdrawn
- 2009-07-29 NZ NZ592168A patent/NZ592168A/xx not_active IP Right Cessation
- 2009-07-29 KR KR1020117009785A patent/KR20110067140A/ko not_active Application Discontinuation
- 2009-07-29 MX MX2011003811A patent/MX2011003811A/es unknown
- 2009-07-29 PE PE2011000846A patent/PE20120054A1/es not_active Application Discontinuation
- 2009-07-29 JP JP2011530583A patent/JP2012505195A/ja not_active Ceased
- 2009-07-29 EP EP14192364.9A patent/EP2853534A1/fr not_active Withdrawn
- 2009-07-29 BR BRPI0919807A patent/BRPI0919807A2/pt not_active IP Right Cessation
- 2009-07-29 AU AU2009302149A patent/AU2009302149A1/en not_active Abandoned
- 2009-07-29 WO PCT/IB2009/006403 patent/WO2010041108A1/fr active Application Filing
- 2009-07-29 EA EA201170546A patent/EA201170546A1/ru unknown
- 2009-07-29 CN CN200980146341.7A patent/CN102216307B/zh not_active Expired - Fee Related
- 2009-08-05 US US12/536,034 patent/US8148366B2/en not_active Expired - Fee Related
-
2011
- 2011-04-05 ZA ZA2011/02497A patent/ZA201102497B/en unknown
- 2011-04-06 IL IL212179A patent/IL212179A0/en unknown
- 2011-04-07 EC EC2011010962A patent/ECSP11010962A/es unknown
- 2011-04-08 CL CL2011000784A patent/CL2011000784A1/es unknown
- 2011-04-08 CO CO11043787A patent/CO6382121A2/es not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
EP2853534A1 (fr) | 2015-04-01 |
EP2358722A1 (fr) | 2011-08-24 |
IL212179A0 (en) | 2011-06-30 |
MX2011003811A (es) | 2011-07-29 |
US8148366B2 (en) | 2012-04-03 |
WO2010041108A1 (fr) | 2010-04-15 |
ECSP11010962A (es) | 2011-05-31 |
AU2009302149A1 (en) | 2010-04-15 |
NZ592168A (en) | 2013-03-28 |
PE20120054A1 (es) | 2012-01-26 |
CA2739776A1 (fr) | 2010-04-15 |
CL2011000784A1 (es) | 2011-10-07 |
CN102216307B (zh) | 2015-02-25 |
JP2012505195A (ja) | 2012-03-01 |
CO6382121A2 (es) | 2012-02-15 |
US20100093784A1 (en) | 2010-04-15 |
FR2937034A1 (fr) | 2010-04-16 |
CN102216307A (zh) | 2011-10-12 |
FR2937034B1 (fr) | 2012-11-23 |
ZA201102497B (en) | 2011-12-28 |
EA201170546A1 (ru) | 2011-12-30 |
KR20110067140A (ko) | 2011-06-21 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 7A ANUIDADE. |
|
B25A | Requested transfer of rights approved |
Owner name: ASTRA ZENECA HOLDING FRANCE S.A.S. (FR) |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2384 DE 13-09-2016 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |