BRPI0908627A2 - processo para se produzir moléculas escolhidas entre as das fórmulas (iia), (iib), (iic) e (iii), molécula de fórmula (iia), (iib), (iic), (iii), (iv) e (v), processo para produzir uma molécula que corresponde à formula (v), (vi), ou (vii), moléculas, composição farmacêutica e uso de uma composição - Google Patents

processo para se produzir moléculas escolhidas entre as das fórmulas (iia), (iib), (iic) e (iii), molécula de fórmula (iia), (iib), (iic), (iii), (iv) e (v), processo para produzir uma molécula que corresponde à formula (v), (vi), ou (vii), moléculas, composição farmacêutica e uso de uma composição

Info

Publication number
BRPI0908627A2
BRPI0908627A2 BRPI0908627A BRPI0908627A BRPI0908627A2 BR PI0908627 A2 BRPI0908627 A2 BR PI0908627A2 BR PI0908627 A BRPI0908627 A BR PI0908627A BR PI0908627 A BRPI0908627 A BR PI0908627A BR PI0908627 A2 BRPI0908627 A2 BR PI0908627A2
Authority
BR
Brazil
Prior art keywords
iic
iib
iia
iii
formula
Prior art date
Application number
BRPI0908627A
Other languages
English (en)
Inventor
Alain Fournet
Anh Tuan Lormier
Bernardin Akagah
Bruno Figadere
Original Assignee
Alpha Chimica
Inst Rech Developpement Ird
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Alpha Chimica, Inst Rech Developpement Ird filed Critical Alpha Chimica
Publication of BRPI0908627A2 publication Critical patent/BRPI0908627A2/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20Oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/12Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/12Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D215/14Radicals substituted by oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Virology (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BRPI0908627A 2008-05-20 2009-05-15 processo para se produzir moléculas escolhidas entre as das fórmulas (iia), (iib), (iic) e (iii), molécula de fórmula (iia), (iib), (iic), (iii), (iv) e (v), processo para produzir uma molécula que corresponde à formula (v), (vi), ou (vii), moléculas, composição farmacêutica e uso de uma composição BRPI0908627A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0802745A FR2931479B1 (fr) 2008-05-20 2008-05-20 Nouveaux derives de quinoleines 2-substituees et un procede pour leur preparation
PCT/FR2009/000573 WO2009150318A1 (fr) 2008-05-20 2009-05-15 Nouveaux derives de quinoleines 2-substituees et un procede pour leur preparation

Publications (1)

Publication Number Publication Date
BRPI0908627A2 true BRPI0908627A2 (pt) 2015-09-15

Family

ID=40149587

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0908627A BRPI0908627A2 (pt) 2008-05-20 2009-05-15 processo para se produzir moléculas escolhidas entre as das fórmulas (iia), (iib), (iic) e (iii), molécula de fórmula (iia), (iib), (iic), (iii), (iv) e (v), processo para produzir uma molécula que corresponde à formula (v), (vi), ou (vii), moléculas, composição farmacêutica e uso de uma composição

Country Status (5)

Country Link
US (1) US20120225903A1 (pt)
EP (1) EP2291381A1 (pt)
BR (1) BRPI0908627A2 (pt)
FR (1) FR2931479B1 (pt)
WO (1) WO2009150318A1 (pt)

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE282457C (pt) *
US4440771A (en) * 1982-02-12 1984-04-03 The United States Of America As Represented By The Secretary Of The Army 2-Acetyl quinoline thiosemicarbazones useful in treatment of gonorrhea, malaria or bacterial infections
FR2682107B1 (fr) * 1991-10-03 1995-04-21 Orstom Inst Fs Rech Scient Quinoleines 2-substituees pour le traitement des leishmanioses.
FR2819507B1 (fr) * 2001-01-17 2007-09-28 Inst Rech Developpement Ird Quinoleines substituees pour le traitement de co-infections a protozoaires et a retrovirus
EP1734939A4 (en) * 2004-03-05 2010-06-30 Univ California PEST CONTROL COMPOUNDS AND METHODS OF USE

Also Published As

Publication number Publication date
US20120225903A1 (en) 2012-09-06
FR2931479B1 (fr) 2012-12-07
WO2009150318A1 (fr) 2009-12-17
FR2931479A1 (fr) 2009-11-27
EP2291381A1 (fr) 2011-03-09

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE AS 5A E 6A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2344 DE 08-12-2015 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.