BRPI0806265A2 - ciclosporina não-imunossupressora para tratamento de distrofia muscular congênita de ullrich - Google Patents

ciclosporina não-imunossupressora para tratamento de distrofia muscular congênita de ullrich Download PDF

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Publication number
BRPI0806265A2
BRPI0806265A2 BRPI0806265-0A BRPI0806265A BRPI0806265A2 BR PI0806265 A2 BRPI0806265 A2 BR PI0806265A2 BR PI0806265 A BRPI0806265 A BR PI0806265A BR PI0806265 A2 BRPI0806265 A2 BR PI0806265A2
Authority
BR
Brazil
Prior art keywords
derivative
cyclosporin
formula
immunosuppressive
csa
Prior art date
Application number
BRPI0806265-0A
Other languages
English (en)
Portuguese (pt)
Inventor
Paolo Bernardi
Gregoire Vuagniaux
Rafael Crabbe
Original Assignee
Debiopharm Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Debiopharm Sa filed Critical Debiopharm Sa
Publication of BRPI0806265A2 publication Critical patent/BRPI0806265A2/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/12Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
    • A61K38/13Cyclosporins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Neurology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Epidemiology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
BRPI0806265-0A 2007-01-04 2008-01-03 ciclosporina não-imunossupressora para tratamento de distrofia muscular congênita de ullrich BRPI0806265A2 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US87841407P 2007-01-04 2007-01-04
US60/878,414 2007-01-04
PCT/IB2008/000003 WO2008084368A2 (en) 2007-01-04 2008-01-03 Non-immunosuppressive cyclosporin for treatment of ullrich congenital muscular dystrophy

Publications (1)

Publication Number Publication Date
BRPI0806265A2 true BRPI0806265A2 (pt) 2011-09-06

Family

ID=39514754

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0806265-0A BRPI0806265A2 (pt) 2007-01-04 2008-01-03 ciclosporina não-imunossupressora para tratamento de distrofia muscular congênita de ullrich

Country Status (12)

Country Link
US (1) US8450281B2 (OSRAM)
EP (1) EP2124992A2 (OSRAM)
JP (1) JP5801534B2 (OSRAM)
CN (2) CN105056207A (OSRAM)
AU (1) AU2008204344B2 (OSRAM)
BR (1) BRPI0806265A2 (OSRAM)
CA (1) CA2674296C (OSRAM)
HK (1) HK1210951A1 (OSRAM)
IL (1) IL199674A (OSRAM)
MX (1) MX2009007045A (OSRAM)
RU (1) RU2462262C2 (OSRAM)
WO (1) WO2008084368A2 (OSRAM)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2009098533A1 (en) * 2008-02-08 2009-08-13 Debiopharm Sa Non -immunosuppressive cyclosporin for the treatment of muscular dystrophy
WO2011098808A1 (en) 2010-02-09 2011-08-18 Biotica Technology Limited Sanglifehrin based compounds
MX2012008873A (es) 2010-02-09 2012-11-22 Biotica Tech Ltd Compuestos a base de sangliferina.
WO2011098805A1 (en) 2010-02-09 2011-08-18 Biotica Technology Limited Sanglifehrin based compounds
GB201008123D0 (en) 2010-05-17 2010-06-30 Biotica Tech Ltd Novel compounds
WO2012085553A1 (en) 2010-12-20 2012-06-28 Biotica Technology Limited Sanglifehrin derivatives and methods for their production
JO3063B1 (ar) 2011-03-29 2017-03-15 Neurovive Pharmaceutical Ab مركب مبتكر وطرق لانتاجه
WO2013169616A1 (en) 2012-05-07 2013-11-14 Novartis Ag Pharmacokinetic modulation with alisporivir
AR090964A1 (es) 2012-05-09 2014-12-17 Novartis Ag Proceso para la elaboracion de undecapeptidos ciclicos

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3884470T2 (de) * 1987-06-17 1994-03-10 Sandoz Ag Cyclosporine und deren Benutzung als Arzneimittel.
GB2222770B (en) 1988-09-16 1992-07-29 Sandoz Ltd Pharmaceutical compositions containing cyclosporins
AU3965699A (en) * 1998-04-24 1999-11-16 Mitokor Compounds and methods for treating mitochondria-associated diseases
EP1091975B1 (fr) * 1998-07-01 2005-12-14 Debiopharm S.A. Nouvelle cyclosporine ayant un profil d'activite ameliore
US6323039B1 (en) * 1999-06-22 2001-11-27 Mitokor Compositions and methods for assaying subcellular conditions and processes using energy transfer
US7368423B1 (en) 2001-12-05 2008-05-06 The Scripps Research Institute Composition and method for treating chronic allograft rejection
GB0320638D0 (en) * 2003-09-03 2003-10-01 Novartis Ag Organic compounds
WO2009098533A1 (en) * 2008-02-08 2009-08-13 Debiopharm Sa Non -immunosuppressive cyclosporin for the treatment of muscular dystrophy

Also Published As

Publication number Publication date
IL199674A0 (en) 2010-04-15
JP2010514834A (ja) 2010-05-06
AU2008204344A9 (en) 2012-06-28
AU2008204344B2 (en) 2013-01-31
EP2124992A2 (en) 2009-12-02
HK1210951A1 (en) 2016-05-13
WO2008084368A9 (en) 2009-02-26
RU2462262C2 (ru) 2012-09-27
IL199674A (en) 2016-10-31
CA2674296A1 (en) 2008-07-17
US20100041593A1 (en) 2010-02-18
WO2008084368A8 (en) 2009-09-17
RU2009129212A (ru) 2011-02-10
CA2674296C (en) 2015-11-24
MX2009007045A (es) 2009-10-07
JP5801534B2 (ja) 2015-10-28
CN101616683A (zh) 2009-12-30
US8450281B2 (en) 2013-05-28
CN105056207A (zh) 2015-11-18
WO2008084368A2 (en) 2008-07-17
AU2008204344A1 (en) 2008-07-17

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Legal Events

Date Code Title Description
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B06I Publication of requirement cancelled [chapter 6.9 patent gazette]
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]

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