BRPI0805841A2 - agente para tratamento de esclerose múltipla - Google Patents

agente para tratamento de esclerose múltipla Download PDF

Info

Publication number
BRPI0805841A2
BRPI0805841A2 BRPI0805841-5A BRPI0805841A BRPI0805841A2 BR PI0805841 A2 BRPI0805841 A2 BR PI0805841A2 BR PI0805841 A BRPI0805841 A BR PI0805841A BR PI0805841 A2 BRPI0805841 A2 BR PI0805841A2
Authority
BR
Brazil
Prior art keywords
multiple sclerosis
treatment agent
agent
treatment
sclerosis treatment
Prior art date
Application number
BRPI0805841-5A
Other languages
English (en)
Inventor
Masaki Yamabi
Yuchiro Tabunoki
Toshiyuki Edano
Original Assignee
Kowa Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kowa Co filed Critical Kowa Co
Publication of BRPI0805841A2 publication Critical patent/BRPI0805841A2/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50Pyridazines; Hydrogenated pyridazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D237/00Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/02Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
    • C07D237/06Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D237/10Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D237/14Oxygen atoms

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

AGENTE PARA TRATAMENTO DE ESCLEROSE MúLTIPLA. é descrito um agente oralmente administrável para prevenção e/ou tratamento de esclerose múltipla, que é altamente eficaz para esclerose múltipla e excelente na segurança. Especificamente descrito é um agente para prevenção e/ou tratamento de esclerose múltipla, que contém 2-benzil-5-(4-clorofenil)-6-[4-(metiltio)fenil]-2H-piridazin-3-ona ou um solvato do mesmo como um ativo ingrediente.
BRPI0805841-5A 2007-01-29 2008-01-28 agente para tratamento de esclerose múltipla BRPI0805841A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2007017328 2007-01-29
PCT/JP2008/000099 WO2008093495A1 (ja) 2007-01-29 2008-01-28 多発性硬化症治療剤

Publications (1)

Publication Number Publication Date
BRPI0805841A2 true BRPI0805841A2 (pt) 2011-08-30

Family

ID=39673809

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0805841-5A BRPI0805841A2 (pt) 2007-01-29 2008-01-28 agente para tratamento de esclerose múltipla

Country Status (12)

Country Link
US (1) US20100075972A1 (pt)
EP (1) EP2127653A1 (pt)
JP (1) JPWO2008093495A1 (pt)
KR (1) KR20090114371A (pt)
CN (1) CN101600435A (pt)
AU (1) AU2008211480A1 (pt)
BR (1) BRPI0805841A2 (pt)
CA (1) CA2669563A1 (pt)
EA (1) EA200970720A1 (pt)
MX (1) MX2009008059A (pt)
TW (1) TW200838535A (pt)
WO (1) WO2008093495A1 (pt)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100626605B1 (ko) 1997-11-19 2006-09-22 코와 가부시키가이샤 신규 피리다진 유도체 및 이를 유효성분으로 하는 의약
CA2742411A1 (en) * 2000-09-18 2002-03-21 Eisai R&D Management Co., Ltd. Pyridazinone and triazinone compounds and use thereof as pharmaceutical preparations

Also Published As

Publication number Publication date
JPWO2008093495A1 (ja) 2010-05-20
AU2008211480A1 (en) 2008-08-07
EA200970720A1 (ru) 2009-12-30
MX2009008059A (es) 2009-08-12
TW200838535A (en) 2008-10-01
CN101600435A (zh) 2009-12-09
US20100075972A1 (en) 2010-03-25
CA2669563A1 (en) 2008-08-07
EP2127653A1 (en) 2009-12-02
WO2008093495A1 (ja) 2008-08-07
KR20090114371A (ko) 2009-11-03

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 4A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: NAO APRESENTADA A GUIA DE CUMPRIMENTO DE EXIGENCIA. REFERENTE A 4A ANUIDADE.