BRPI0805841A2 - agente para tratamento de esclerose múltipla - Google Patents
agente para tratamento de esclerose múltipla Download PDFInfo
- Publication number
- BRPI0805841A2 BRPI0805841A2 BRPI0805841-5A BRPI0805841A BRPI0805841A2 BR PI0805841 A2 BRPI0805841 A2 BR PI0805841A2 BR PI0805841 A BRPI0805841 A BR PI0805841A BR PI0805841 A2 BRPI0805841 A2 BR PI0805841A2
- Authority
- BR
- Brazil
- Prior art keywords
- multiple sclerosis
- treatment agent
- agent
- treatment
- sclerosis treatment
- Prior art date
Links
- 239000002749 multiple sclerosis treatment agent Substances 0.000 title abstract 2
- 201000006417 multiple sclerosis Diseases 0.000 abstract 3
- 239000003795 chemical substances by application Substances 0.000 abstract 2
- 230000002265 prevention Effects 0.000 abstract 2
- HEUAVAATAFEENP-UHFFFAOYSA-N 2-benzyl-5-(4-chlorophenyl)-6-(4-methylsulfanylphenyl)pyridazin-3-one Chemical compound C1=CC(SC)=CC=C1C(C(=CC1=O)C=2C=CC(Cl)=CC=2)=NN1CC1=CC=CC=C1 HEUAVAATAFEENP-UHFFFAOYSA-N 0.000 abstract 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/50—Pyridazines; Hydrogenated pyridazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
- C07D237/06—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D237/10—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D237/14—Oxygen atoms
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
AGENTE PARA TRATAMENTO DE ESCLEROSE MúLTIPLA. é descrito um agente oralmente administrável para prevenção e/ou tratamento de esclerose múltipla, que é altamente eficaz para esclerose múltipla e excelente na segurança. Especificamente descrito é um agente para prevenção e/ou tratamento de esclerose múltipla, que contém 2-benzil-5-(4-clorofenil)-6-[4-(metiltio)fenil]-2H-piridazin-3-ona ou um solvato do mesmo como um ativo ingrediente.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2007017328 | 2007-01-29 | ||
| PCT/JP2008/000099 WO2008093495A1 (ja) | 2007-01-29 | 2008-01-28 | 多発性硬化症治療剤 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0805841A2 true BRPI0805841A2 (pt) | 2011-08-30 |
Family
ID=39673809
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0805841-5A BRPI0805841A2 (pt) | 2007-01-29 | 2008-01-28 | agente para tratamento de esclerose múltipla |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US20100075972A1 (pt) |
| EP (1) | EP2127653A1 (pt) |
| JP (1) | JPWO2008093495A1 (pt) |
| KR (1) | KR20090114371A (pt) |
| CN (1) | CN101600435A (pt) |
| AU (1) | AU2008211480A1 (pt) |
| BR (1) | BRPI0805841A2 (pt) |
| CA (1) | CA2669563A1 (pt) |
| EA (1) | EA200970720A1 (pt) |
| MX (1) | MX2009008059A (pt) |
| TW (1) | TW200838535A (pt) |
| WO (1) | WO2008093495A1 (pt) |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR100626605B1 (ko) | 1997-11-19 | 2006-09-22 | 코와 가부시키가이샤 | 신규 피리다진 유도체 및 이를 유효성분으로 하는 의약 |
| CA2742411A1 (en) * | 2000-09-18 | 2002-03-21 | Eisai R&D Management Co., Ltd. | Pyridazinone and triazinone compounds and use thereof as pharmaceutical preparations |
-
2008
- 2008-01-28 AU AU2008211480A patent/AU2008211480A1/en not_active Abandoned
- 2008-01-28 CN CNA2008800032965A patent/CN101600435A/zh active Pending
- 2008-01-28 MX MX2009008059A patent/MX2009008059A/es unknown
- 2008-01-28 EP EP08710303A patent/EP2127653A1/en not_active Withdrawn
- 2008-01-28 WO PCT/JP2008/000099 patent/WO2008093495A1/ja not_active Ceased
- 2008-01-28 CA CA002669563A patent/CA2669563A1/en not_active Abandoned
- 2008-01-28 BR BRPI0805841-5A patent/BRPI0805841A2/pt not_active IP Right Cessation
- 2008-01-28 JP JP2008556026A patent/JPWO2008093495A1/ja active Pending
- 2008-01-28 EA EA200970720A patent/EA200970720A1/ru unknown
- 2008-01-28 US US12/516,595 patent/US20100075972A1/en not_active Abandoned
- 2008-01-28 TW TW097103099A patent/TW200838535A/zh unknown
- 2008-01-28 KR KR1020097015733A patent/KR20090114371A/ko not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| JPWO2008093495A1 (ja) | 2010-05-20 |
| AU2008211480A1 (en) | 2008-08-07 |
| EA200970720A1 (ru) | 2009-12-30 |
| MX2009008059A (es) | 2009-08-12 |
| TW200838535A (en) | 2008-10-01 |
| CN101600435A (zh) | 2009-12-09 |
| US20100075972A1 (en) | 2010-03-25 |
| CA2669563A1 (en) | 2008-08-07 |
| EP2127653A1 (en) | 2009-12-02 |
| WO2008093495A1 (ja) | 2008-08-07 |
| KR20090114371A (ko) | 2009-11-03 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 4A ANUIDADE. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: NAO APRESENTADA A GUIA DE CUMPRIMENTO DE EXIGENCIA. REFERENTE A 4A ANUIDADE. |