BRPI0722096A2 - Compostos de 4-hidróxi-2-oxo-2,3-dihidro-1,3-benzotiazol-7-il para modulação de atividade de b2-adrenorreceptor - Google Patents

Compostos de 4-hidróxi-2-oxo-2,3-dihidro-1,3-benzotiazol-7-il para modulação de atividade de b2-adrenorreceptor

Info

Publication number
BRPI0722096A2
BRPI0722096A2 BRPI0722096-0A2A BRPI0722096A BRPI0722096A2 BR PI0722096 A2 BRPI0722096 A2 BR PI0722096A2 BR PI0722096 A BRPI0722096 A BR PI0722096A BR PI0722096 A2 BRPI0722096 A2 BR PI0722096A2
Authority
BR
Brazil
Prior art keywords
adrenorreceptor
benzotiazol
dihydro
oxo
modulating
Prior art date
Application number
BRPI0722096-0A2A
Other languages
English (en)
Inventor
Stephen Connolly
Alexander Humphries
Premji Meghani
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of BRPI0722096A2 publication Critical patent/BRPI0722096A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/08—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D277/12—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/14—Oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/16—Otologicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/14—Thiadiazoles; Hydrogenated thiadiazoles condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Steroid Compounds (AREA)
BRPI0722096-0A2A 2006-12-20 2007-12-19 Compostos de 4-hidróxi-2-oxo-2,3-dihidro-1,3-benzotiazol-7-il para modulação de atividade de b2-adrenorreceptor BRPI0722096A2 (pt)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US87092206P 2006-12-20 2006-12-20
US91004507P 2007-04-04 2007-04-04
US95198007P 2007-07-26 2007-07-26
PCT/GB2007/004861 WO2008075026A1 (en) 2006-12-20 2007-12-19 4-hydr0xy-2-0x0-2, 3 -dihydro- 1, 3-benzothiazol- 7yl compounds for modulation of b2-adrenoreceptor activity

Publications (1)

Publication Number Publication Date
BRPI0722096A2 true BRPI0722096A2 (pt) 2014-04-01

Family

ID=39167020

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0722096-0A2A BRPI0722096A2 (pt) 2006-12-20 2007-12-19 Compostos de 4-hidróxi-2-oxo-2,3-dihidro-1,3-benzotiazol-7-il para modulação de atividade de b2-adrenorreceptor

Country Status (21)

Country Link
US (3) US7700782B2 (pt)
EP (1) EP2121642B1 (pt)
JP (1) JP2010513440A (pt)
KR (1) KR20090091342A (pt)
AR (1) AR064635A1 (pt)
AT (1) ATE517879T1 (pt)
AU (1) AU2007336075B2 (pt)
BR (1) BRPI0722096A2 (pt)
CA (1) CA2672811A1 (pt)
CL (1) CL2007003765A1 (pt)
CO (1) CO6190554A2 (pt)
EC (1) ECSP099426A (pt)
HK (1) HK1136572A1 (pt)
IL (1) IL199014A0 (pt)
MX (1) MX2009006009A (pt)
NO (1) NO20092691L (pt)
PE (1) PE20081544A1 (pt)
SA (1) SA07280728B1 (pt)
TW (1) TW200833670A (pt)
UY (1) UY30808A1 (pt)
WO (1) WO2008075026A1 (pt)

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AU2008356409B2 (en) 2008-05-13 2012-01-19 Astrazeneca Ab Quinuclidine derivatives as muscarinic M3 receptor antagonists
WO2009154557A1 (en) 2008-06-18 2009-12-23 Astrazeneca Ab Benzoxazinone derivatives acting as beta2-adrenoreceptor agonist for the treatment of respiratory disorders
RU2011101664A (ru) * 2008-06-20 2012-07-27 Астразенека Аб (Se) Фармацевтическая композиция, содержащая 4-гидрокси-2-оксо-2, 3-дигидро-1, 3-бензотиазол-7-ильное соединение, для модулирования активности бета2- адренорецепторов
GB0814728D0 (en) * 2008-08-12 2008-09-17 Argenta Discovery Ltd New combination
TW201036957A (en) 2009-02-20 2010-10-16 Astrazeneca Ab Novel salt 628
GB0913342D0 (en) 2009-07-31 2009-09-16 Astrazeneca Ab Compounds - 801
WO2011061527A1 (en) 2009-11-17 2011-05-26 Astrazeneca Ab Combinations comprising a glucocorticoid receptor modulator for the treatment of respiratory diseases
GB201016912D0 (en) 2010-10-07 2010-11-24 Astrazeneca Ab Novel combination
JO3192B1 (ar) * 2011-09-06 2018-03-08 Novartis Ag مركب بنزوثيازولون
WO2015050984A1 (en) * 2013-10-01 2015-04-09 New York University Amino, amido, and heterocyclic compounds as modulators of rage activity and uses thereof

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Also Published As

Publication number Publication date
US20100249200A1 (en) 2010-09-30
US20100022491A1 (en) 2010-01-28
US7700782B2 (en) 2010-04-20
CL2007003765A1 (es) 2008-08-22
ECSP099426A (es) 2009-07-31
TW200833670A (en) 2008-08-16
ATE517879T1 (de) 2011-08-15
CA2672811A1 (en) 2008-06-26
AU2007336075A1 (en) 2008-06-26
HK1136572A1 (en) 2010-07-02
JP2010513440A (ja) 2010-04-30
UY30808A1 (es) 2008-07-31
WO2008075026A1 (en) 2008-06-26
AU2007336075B2 (en) 2011-10-27
NO20092691L (no) 2009-09-16
IL199014A0 (en) 2010-02-17
KR20090091342A (ko) 2009-08-27
AR064635A1 (es) 2009-04-15
SA07280728B1 (ar) 2010-12-01
MX2009006009A (es) 2009-06-16
EP2121642A1 (en) 2009-11-25
US20080207698A1 (en) 2008-08-28
EP2121642B1 (en) 2011-07-27
CO6190554A2 (es) 2010-08-19
PE20081544A1 (es) 2009-01-11

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