BRPI0608978A2 - terapia ocular usando agonistas de receptor alfa-2 adrenérgico possuindo taxas de depuração anterior realçadas - Google Patents

terapia ocular usando agonistas de receptor alfa-2 adrenérgico possuindo taxas de depuração anterior realçadas Download PDF

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Publication number
BRPI0608978A2
BRPI0608978A2 BRPI0608978-0A BRPI0608978A BRPI0608978A2 BR PI0608978 A2 BRPI0608978 A2 BR PI0608978A2 BR PI0608978 A BRPI0608978 A BR PI0608978A BR PI0608978 A2 BRPI0608978 A2 BR PI0608978A2
Authority
BR
Brazil
Prior art keywords
alpha
eye
adrenergic receptor
receptor agonist
administration
Prior art date
Application number
BRPI0608978-0A
Other languages
English (en)
Portuguese (pt)
Inventor
Patrick M Hugues
James A Burke
Joan-En Chang-Lin
Original Assignee
Allergan Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Allergan Inc filed Critical Allergan Inc
Publication of BRPI0608978A2 publication Critical patent/BRPI0608978A2/pt

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0048Eye, e.g. artificial tears
    • A61K9/0051Ocular inserts, ocular implants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0048Eye, e.g. artificial tears
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/06Antiglaucoma agents or miotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/10Ophthalmic agents for accommodation disorders, e.g. myopia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1641Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
    • A61K9/1647Polyesters, e.g. poly(lactide-co-glycolide)

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Ophthalmology & Optometry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Materials For Medical Uses (AREA)
BRPI0608978-0A 2005-05-10 2006-05-09 terapia ocular usando agonistas de receptor alfa-2 adrenérgico possuindo taxas de depuração anterior realçadas BRPI0608978A2 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US67977105P 2005-05-10 2005-05-10
US60/679,771 2005-05-10
PCT/US2006/018019 WO2006122165A2 (en) 2005-05-10 2006-05-09 Ocular therapy using alpha-2 adrenergic receptor agonists having enhanced anterior clearance rates

Publications (1)

Publication Number Publication Date
BRPI0608978A2 true BRPI0608978A2 (pt) 2010-02-17

Family

ID=37397258

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0608978-0A BRPI0608978A2 (pt) 2005-05-10 2006-05-09 terapia ocular usando agonistas de receptor alfa-2 adrenérgico possuindo taxas de depuração anterior realçadas

Country Status (8)

Country Link
US (3) US7931909B2 (OSRAM)
EP (2) EP3656374A1 (OSRAM)
JP (3) JP2008540552A (OSRAM)
AU (1) AU2006244083A1 (OSRAM)
BR (1) BRPI0608978A2 (OSRAM)
CA (1) CA2603069C (OSRAM)
ES (1) ES2798259T3 (OSRAM)
WO (1) WO2006122165A2 (OSRAM)

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Also Published As

Publication number Publication date
EP1879553A2 (en) 2008-01-23
US20060257452A1 (en) 2006-11-16
EP3656374A1 (en) 2020-05-27
JP2012046530A (ja) 2012-03-08
WO2006122165A2 (en) 2006-11-16
EP1879553B1 (en) 2020-02-12
AU2006244083A1 (en) 2006-11-16
JP2008540552A (ja) 2008-11-20
US20080112922A1 (en) 2008-05-15
WO2006122165A3 (en) 2007-05-31
CA2603069C (en) 2014-01-28
US7931909B2 (en) 2011-04-26
CA2603069A1 (en) 2006-11-16
US20080112923A1 (en) 2008-05-15
ES2798259T3 (es) 2020-12-10
JP2015013863A (ja) 2015-01-22

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Legal Events

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B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 10A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2385 DE 20-09-2016 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.