BRPI0408464A - processos de hidrogenação e para minimizar a sobre-hidrogenação de uma piridina substituìda com arila - Google Patents

processos de hidrogenação e para minimizar a sobre-hidrogenação de uma piridina substituìda com arila

Info

Publication number
BRPI0408464A
BRPI0408464A BRPI0408464-0A BRPI0408464A BRPI0408464A BR PI0408464 A BRPI0408464 A BR PI0408464A BR PI0408464 A BRPI0408464 A BR PI0408464A BR PI0408464 A BRPI0408464 A BR PI0408464A
Authority
BR
Brazil
Prior art keywords
minimize
aryl substituted
overhydrogenation
substituted pyridine
hydrogenation processes
Prior art date
Application number
BRPI0408464-0A
Other languages
English (en)
Inventor
Timothy James Norman Watson
Michael Girard Vetelino
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of BRPI0408464A publication Critical patent/BRPI0408464A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56Nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Pulmonology (AREA)
  • Psychiatry (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pyridine Compounds (AREA)
  • Catalysts (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

"PROCESSOS DE HIDROGENAçãO E PARA MINIMIZAR A SOBRE-HIDROGENAçãO DE UMA PIRIDINA SUBSTITUìDA COM ARILA". A presente invenção refere-se a processo para hidrogenar uma piridina substituída com arila, tal como 2-fenil-3-aminopiridina, sem sobreredução do anel arila utilizando um catalisador Pt/C específico.
BRPI0408464-0A 2003-03-17 2004-03-04 processos de hidrogenação e para minimizar a sobre-hidrogenação de uma piridina substituìda com arila BRPI0408464A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US45560403P 2003-03-17 2003-03-17
PCT/IB2004/000667 WO2004083181A1 (en) 2003-03-17 2004-03-04 Synthesis of aryl-substituted piperidines by hydrogenation of aryl-substituted pyridines

Publications (1)

Publication Number Publication Date
BRPI0408464A true BRPI0408464A (pt) 2006-04-04

Family

ID=33030028

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0408464-0A BRPI0408464A (pt) 2003-03-17 2004-03-04 processos de hidrogenação e para minimizar a sobre-hidrogenação de uma piridina substituìda com arila

Country Status (10)

Country Link
US (1) US6995270B2 (pt)
EP (1) EP1606257A1 (pt)
JP (1) JP2006523205A (pt)
AR (1) AR043625A1 (pt)
BR (1) BRPI0408464A (pt)
CA (1) CA2518447A1 (pt)
CL (1) CL2004000430A1 (pt)
MX (1) MXPA05008147A (pt)
TW (1) TW200420539A (pt)
WO (1) WO2004083181A1 (pt)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR102544704B1 (ko) * 2021-01-12 2023-06-20 한국화학연구원 수소화 및 탈수소화 반응 속도가 향상된 피리딘계 수소 저장 물질 및 이를 이용한 수소 저장 및 방출 방법

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4680283A (en) 1984-09-26 1987-07-14 Merck & Co., Inc. Analogs of substance P and eledoisin
FI955708L (fi) * 1993-05-28 1995-11-27 Pfizer Menetelmä 2-fenyyli-3-aminopiperidiinin valmistamiseksi ja erottamiseksi

Also Published As

Publication number Publication date
CA2518447A1 (en) 2004-09-30
MXPA05008147A (es) 2007-08-02
TW200420539A (en) 2004-10-16
WO2004083181A1 (en) 2004-09-30
US20040249160A1 (en) 2004-12-09
US6995270B2 (en) 2006-02-07
CL2004000430A1 (es) 2005-02-04
EP1606257A1 (en) 2005-12-21
JP2006523205A (ja) 2006-10-12
AR043625A1 (es) 2005-08-03

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 6A, 7A E 8A ANUIDADE(S).

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: NAO APRESENTADA A GUIA DE CUMPRIMENTO DE EXIGENCIA. REFERENTE AS 6A, 7A E 8A ANUIDADES.