BR9916919A - Compósito de sulfonamida e seu uso - Google Patents

Compósito de sulfonamida e seu uso

Info

Publication number
BR9916919A
BR9916919A BR9916919-3A BR9916919A BR9916919A BR 9916919 A BR9916919 A BR 9916919A BR 9916919 A BR9916919 A BR 9916919A BR 9916919 A BR9916919 A BR 9916919A
Authority
BR
Brazil
Prior art keywords
action
compound
sulfonamide
diseases based
composite
Prior art date
Application number
BR9916919-3A
Other languages
English (en)
Inventor
Hiroshi Kayakiri
Yoshito Abe
Hitoshi Hamashima
Hitoshi Sawada
Naoki Ishibashi
Hiroyuki Setol
Teruo Oku
Noritsugu Yamasaki
Takafumi Imoto
Takahiro Hiramura
Original Assignee
Fujisawa Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fujisawa Pharmaceutical Co filed Critical Fujisawa Pharmaceutical Co
Publication of BR9916919A publication Critical patent/BR9916919A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Pulmonology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Immunology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

"COMPOSTO DE SULFONAMIDA E SEU USO". A presente invenção refere-se a um composto de sulfonamida da fórmula (I): onde cada símbolo é conforme definido na especificação, um sal do mesmo, e uma composição farmacêutica contendo o mesmo. Este composto pode ser um agente eficaz na profilaxia e tratamento das doenças curáveis com base numa ação hipoglicêmica, e das doenças curáveis com base numa ação inibidora de cGMP-PDE, ação relaxante sobre a musculatura lisa, ação broncodilatadora, ação vasodilatadora, ação inibidora de células da musculatura lisa e ação supressora de alergia.
BR9916919-3A 1998-12-04 1999-12-01 Compósito de sulfonamida e seu uso BR9916919A (pt)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP34617598 1998-12-04
JP36754098 1998-12-24
JP25928399 1999-08-09
PCT/JP1999/006748 WO2000034277A1 (fr) 1998-12-04 1999-12-01 Composes de sulfamide et utilisations de ces derniers en tant que medicaments

Publications (1)

Publication Number Publication Date
BR9916919A true BR9916919A (pt) 2002-01-15

Family

ID=27334802

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9916919-3A BR9916919A (pt) 1998-12-04 1999-12-01 Compósito de sulfonamida e seu uso

Country Status (15)

Country Link
US (2) US6573274B1 (pt)
EP (1) EP1136492A4 (pt)
KR (1) KR20010086593A (pt)
CN (1) CN1335847A (pt)
AR (1) AR021542A1 (pt)
AU (1) AU769890B2 (pt)
BR (1) BR9916919A (pt)
CA (1) CA2352871A1 (pt)
CZ (1) CZ20011981A3 (pt)
HK (1) HK1044154A1 (pt)
HU (1) HUP0104549A3 (pt)
IL (1) IL143439A0 (pt)
TR (1) TR200101568T2 (pt)
TW (1) TW577889B (pt)
WO (1) WO2000034277A1 (pt)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6348474B1 (en) * 1997-06-27 2002-02-19 Fujisawa Pharmaceutical Co., Ltd. Sulfonamide compounds and medicinal use thereof
AU2001276607A1 (en) * 2000-08-11 2002-02-25 Pfizer Inc. Treatment of the insulin resistance syndrome with selective CGMP PDE5 inhibitors
US7098231B2 (en) 2003-01-22 2006-08-29 Boehringer Ingelheim International Gmbh Viral polymerase inhibitors
US7223785B2 (en) 2003-01-22 2007-05-29 Boehringer Ingelheim International Gmbh Viral polymerase inhibitors
US20050197376A1 (en) * 2004-03-02 2005-09-08 Fujisawa Pharmaceutical Co. Ltd. Concomitant drugs
EP2114856A1 (en) * 2007-02-06 2009-11-11 Cipla Limited Process for the preparation of ethyl-n-(2, 3-dichloro-6-nitrobenzyl) glycine hydrochloride
WO2014123203A1 (ja) * 2013-02-06 2014-08-14 京都薬品工業株式会社 糖尿病治療薬
GB201321741D0 (en) * 2013-12-09 2014-01-22 Ucb Pharma Sa Therapeutic agents
TWI731317B (zh) * 2013-12-10 2021-06-21 美商健臻公司 原肌球蛋白相關之激酶(trk)抑制劑
LT3762368T (lt) 2018-03-08 2022-06-10 Incyte Corporation Aminopirazindiolio junginiai, kaip pi3k-γ inhibitoriai
WO2020010003A1 (en) 2018-07-02 2020-01-09 Incyte Corporation AMINOPYRAZINE DERIVATIVES AS PI3K-γ INHIBITORS

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5215994A (en) 1990-09-25 1993-06-01 Fujisawa Pharmaceutical Co., Ltd. Angiotenin II antagonizing heterocyclic derivatives
EP0503838A3 (en) * 1991-03-08 1992-10-07 Merck & Co. Inc. Heterocyclic compounds bearing acidic functional groups as angiotensin ii antagonists
US5128327A (en) * 1991-03-25 1992-07-07 Merck & Co., Inc. Angiotensin II antagonists incorporating a nitrogen containing six membered ring heterocycle
WO1993019067A1 (en) 1991-09-12 1993-09-30 Fujisawa Pharmaceutical Co., Ltd. Imidazopyridine derivatives as angiotensin ii antagonists
IL124969A (en) 1995-12-28 2002-09-12 Fujisawa Pharmaceutical Co History of benzimidazole, processes for their preparation and pharmaceutical preparations containing them
EP1000932B9 (en) 1997-06-27 2005-12-28 Fujisawa Pharmaceutical Co., Ltd. Aromatic ring derivatives
US6348474B1 (en) * 1997-06-27 2002-02-19 Fujisawa Pharmaceutical Co., Ltd. Sulfonamide compounds and medicinal use thereof

Also Published As

Publication number Publication date
HK1044154A1 (zh) 2002-10-11
WO2000034277A1 (fr) 2000-06-15
AU769890B2 (en) 2004-02-05
TR200101568T2 (tr) 2001-10-22
EP1136492A4 (en) 2002-03-27
HUP0104549A2 (hu) 2002-04-29
EP1136492A1 (en) 2001-09-26
AR021542A1 (es) 2002-07-24
CA2352871A1 (en) 2000-06-15
AU1414100A (en) 2000-06-26
US6573274B1 (en) 2003-06-03
IL143439A0 (en) 2002-04-21
TW577889B (en) 2004-03-01
CN1335847A (zh) 2002-02-13
US20030171396A1 (en) 2003-09-11
HUP0104549A3 (en) 2002-12-28
CZ20011981A3 (cs) 2002-01-16
US6890934B2 (en) 2005-05-10
KR20010086593A (ko) 2001-09-13

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 6O, 7O E 8O ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 1913 DE 04/09/2007.