BR9916919A - Compósito de sulfonamida e seu uso - Google Patents
Compósito de sulfonamida e seu usoInfo
- Publication number
- BR9916919A BR9916919A BR9916919-3A BR9916919A BR9916919A BR 9916919 A BR9916919 A BR 9916919A BR 9916919 A BR9916919 A BR 9916919A BR 9916919 A BR9916919 A BR 9916919A
- Authority
- BR
- Brazil
- Prior art keywords
- action
- compound
- sulfonamide
- diseases based
- composite
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Diabetes (AREA)
- Pulmonology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Immunology (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
"COMPOSTO DE SULFONAMIDA E SEU USO". A presente invenção refere-se a um composto de sulfonamida da fórmula (I): onde cada símbolo é conforme definido na especificação, um sal do mesmo, e uma composição farmacêutica contendo o mesmo. Este composto pode ser um agente eficaz na profilaxia e tratamento das doenças curáveis com base numa ação hipoglicêmica, e das doenças curáveis com base numa ação inibidora de cGMP-PDE, ação relaxante sobre a musculatura lisa, ação broncodilatadora, ação vasodilatadora, ação inibidora de células da musculatura lisa e ação supressora de alergia.
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP34617598 | 1998-12-04 | ||
JP36754098 | 1998-12-24 | ||
JP25928399 | 1999-08-09 | ||
PCT/JP1999/006748 WO2000034277A1 (fr) | 1998-12-04 | 1999-12-01 | Composes de sulfamide et utilisations de ces derniers en tant que medicaments |
Publications (1)
Publication Number | Publication Date |
---|---|
BR9916919A true BR9916919A (pt) | 2002-01-15 |
Family
ID=27334802
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR9916919-3A BR9916919A (pt) | 1998-12-04 | 1999-12-01 | Compósito de sulfonamida e seu uso |
Country Status (15)
Country | Link |
---|---|
US (2) | US6573274B1 (pt) |
EP (1) | EP1136492A4 (pt) |
KR (1) | KR20010086593A (pt) |
CN (1) | CN1335847A (pt) |
AR (1) | AR021542A1 (pt) |
AU (1) | AU769890B2 (pt) |
BR (1) | BR9916919A (pt) |
CA (1) | CA2352871A1 (pt) |
CZ (1) | CZ20011981A3 (pt) |
HK (1) | HK1044154A1 (pt) |
HU (1) | HUP0104549A3 (pt) |
IL (1) | IL143439A0 (pt) |
TR (1) | TR200101568T2 (pt) |
TW (1) | TW577889B (pt) |
WO (1) | WO2000034277A1 (pt) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6348474B1 (en) * | 1997-06-27 | 2002-02-19 | Fujisawa Pharmaceutical Co., Ltd. | Sulfonamide compounds and medicinal use thereof |
AU2001276607A1 (en) * | 2000-08-11 | 2002-02-25 | Pfizer Inc. | Treatment of the insulin resistance syndrome with selective CGMP PDE5 inhibitors |
US7098231B2 (en) | 2003-01-22 | 2006-08-29 | Boehringer Ingelheim International Gmbh | Viral polymerase inhibitors |
US7223785B2 (en) | 2003-01-22 | 2007-05-29 | Boehringer Ingelheim International Gmbh | Viral polymerase inhibitors |
US20050197376A1 (en) * | 2004-03-02 | 2005-09-08 | Fujisawa Pharmaceutical Co. Ltd. | Concomitant drugs |
EP2114856A1 (en) * | 2007-02-06 | 2009-11-11 | Cipla Limited | Process for the preparation of ethyl-n-(2, 3-dichloro-6-nitrobenzyl) glycine hydrochloride |
WO2014123203A1 (ja) * | 2013-02-06 | 2014-08-14 | 京都薬品工業株式会社 | 糖尿病治療薬 |
GB201321741D0 (en) * | 2013-12-09 | 2014-01-22 | Ucb Pharma Sa | Therapeutic agents |
TWI731317B (zh) * | 2013-12-10 | 2021-06-21 | 美商健臻公司 | 原肌球蛋白相關之激酶(trk)抑制劑 |
LT3762368T (lt) | 2018-03-08 | 2022-06-10 | Incyte Corporation | Aminopirazindiolio junginiai, kaip pi3k-γ inhibitoriai |
WO2020010003A1 (en) | 2018-07-02 | 2020-01-09 | Incyte Corporation | AMINOPYRAZINE DERIVATIVES AS PI3K-γ INHIBITORS |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5215994A (en) | 1990-09-25 | 1993-06-01 | Fujisawa Pharmaceutical Co., Ltd. | Angiotenin II antagonizing heterocyclic derivatives |
EP0503838A3 (en) * | 1991-03-08 | 1992-10-07 | Merck & Co. Inc. | Heterocyclic compounds bearing acidic functional groups as angiotensin ii antagonists |
US5128327A (en) * | 1991-03-25 | 1992-07-07 | Merck & Co., Inc. | Angiotensin II antagonists incorporating a nitrogen containing six membered ring heterocycle |
WO1993019067A1 (en) | 1991-09-12 | 1993-09-30 | Fujisawa Pharmaceutical Co., Ltd. | Imidazopyridine derivatives as angiotensin ii antagonists |
IL124969A (en) | 1995-12-28 | 2002-09-12 | Fujisawa Pharmaceutical Co | History of benzimidazole, processes for their preparation and pharmaceutical preparations containing them |
EP1000932B9 (en) | 1997-06-27 | 2005-12-28 | Fujisawa Pharmaceutical Co., Ltd. | Aromatic ring derivatives |
US6348474B1 (en) * | 1997-06-27 | 2002-02-19 | Fujisawa Pharmaceutical Co., Ltd. | Sulfonamide compounds and medicinal use thereof |
-
1999
- 1999-12-01 IL IL14343999A patent/IL143439A0/xx unknown
- 1999-12-01 TR TR2001/01568T patent/TR200101568T2/xx unknown
- 1999-12-01 BR BR9916919-3A patent/BR9916919A/pt not_active IP Right Cessation
- 1999-12-01 HU HU0104549A patent/HUP0104549A3/hu unknown
- 1999-12-01 KR KR1020017006948A patent/KR20010086593A/ko not_active Application Discontinuation
- 1999-12-01 AU AU14141/00A patent/AU769890B2/en not_active Ceased
- 1999-12-01 US US09/856,172 patent/US6573274B1/en not_active Expired - Fee Related
- 1999-12-01 WO PCT/JP1999/006748 patent/WO2000034277A1/ja not_active Application Discontinuation
- 1999-12-01 CZ CZ20011981A patent/CZ20011981A3/cs unknown
- 1999-12-01 CA CA002352871A patent/CA2352871A1/en not_active Abandoned
- 1999-12-01 CN CN99816022A patent/CN1335847A/zh active Pending
- 1999-12-01 EP EP99973290A patent/EP1136492A4/en not_active Withdrawn
- 1999-12-02 TW TW088121089A patent/TW577889B/zh not_active IP Right Cessation
- 1999-12-03 AR ARP990106177A patent/AR021542A1/es not_active Application Discontinuation
-
2002
- 2002-08-06 HK HK02105752.5A patent/HK1044154A1/zh unknown
-
2003
- 2003-02-10 US US10/360,806 patent/US6890934B2/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
HK1044154A1 (zh) | 2002-10-11 |
WO2000034277A1 (fr) | 2000-06-15 |
AU769890B2 (en) | 2004-02-05 |
TR200101568T2 (tr) | 2001-10-22 |
EP1136492A4 (en) | 2002-03-27 |
HUP0104549A2 (hu) | 2002-04-29 |
EP1136492A1 (en) | 2001-09-26 |
AR021542A1 (es) | 2002-07-24 |
CA2352871A1 (en) | 2000-06-15 |
AU1414100A (en) | 2000-06-26 |
US6573274B1 (en) | 2003-06-03 |
IL143439A0 (en) | 2002-04-21 |
TW577889B (en) | 2004-03-01 |
CN1335847A (zh) | 2002-02-13 |
US20030171396A1 (en) | 2003-09-11 |
HUP0104549A3 (en) | 2002-12-28 |
CZ20011981A3 (cs) | 2002-01-16 |
US6890934B2 (en) | 2005-05-10 |
KR20010086593A (ko) | 2001-09-13 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
BRPI0405166A (pt) | Composição de cuidados pessoais e processo para preparar a mesma | |
BR0111196A (pt) | Composições e uso das mesmas para tratamento de flavivìrus e pestivìrus | |
IT1252868B (it) | Composizione farmaceutica anticefalalgica per somministrazione endonasale, procedimento per prepararla e suo impiego terapeutico | |
BRPI0113042B8 (pt) | composto da fórmula ou um seu solvato fisiologicamente aceitável, uso do mesmo, composição farmacêutica, formulação farmacêutica, método para o tratamento de um indivíduo humano ou animal com uma condição inflamatória e/ou alérgica, e, processo para preparar um composto ou um seu solvato | |
BR0312286A (pt) | pró-medicamentos de 2' e 3' - nucleosìdeo modificado para tratamento de infecções por flaviviridae | |
BR0108173A (pt) | Composições farmacêuticas de toxina de botulina | |
BR9916919A (pt) | Compósito de sulfonamida e seu uso | |
BR9911076A (pt) | Uso de peg-ifn-alfa e ribavirina para o tratamento de hepatite c crÈnica | |
BRPI0517773A (pt) | composição para cuidados pessoais contendo um derivado de polìmero de galactomanano não-guar | |
BRPI0412489A (pt) | composição de confeito mastigável liberando para as superfìcies dentárias uma dose unitária de uma enzima | |
BR0316082A (pt) | Métodos de tratar ou prevenir e de controlar uma doença mieloproliferative, de reduzir ou evitar um efeito adverso associado com a administração de um segundo agente ativo em um paciente sofrendo de uma doença mieloproliferativa e de aumentar a eficácia terapêutica de um tratamento de doenças mieloproliferativa, composição farmacêutica e kit | |
BR9702362A (pt) | Novas fomrulações lìquidas estáveis à base de paracetamol e seu modo de preparação. | |
BR9917112A (pt) | Compostos de imidazol e seu uso medicinal | |
SE0101387D0 (sv) | Novel compounds | |
BR9914954A (pt) | Implante com cavidades contendo agentes terapêuticos | |
BR0113087A (pt) | Novas composições de minoxidil | |
BR0113643A (pt) | Compostos de guanidinobenzamidas como agonistas de mc4-r e seus usos | |
BRPI0407950A (pt) | processo para a preparação de uma composição de higiene pessoal | |
BR0111358A (pt) | Compostos de tioacetamida e seu uso | |
BR0316310A (pt) | Composições farmacêuticas tendo um veìculo modificado | |
EP0937453A3 (en) | Cosmetic and tissue cleansing and moisturizing composition | |
BRPI0406796A (pt) | Métodos para tratar hipertrofia prostática benigna, para reduzir um sintoma associado com a mesma, para reduzir o tamanho da próstata em um indivìduo humano e para profilaxia de bhp, composição farmacêutica oral de dose unitária, e, uso de lonidamina ou um análogo de lonidamina | |
EP1074245A3 (en) | Composition using mineral salts for therapeutic treatment | |
BR9814214A (pt) | Composição com ácido azeláico | |
BR0012444A (pt) | Composições de pó seco |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 6O, 7O E 8O ANUIDADES. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 1913 DE 04/09/2007. |