BR9813982A - Anticoncepcionais orais contendo antiestrogênio mais progestina - Google Patents

Anticoncepcionais orais contendo antiestrogênio mais progestina

Info

Publication number
BR9813982A
BR9813982A BR9813982-7A BR9813982A BR9813982A BR 9813982 A BR9813982 A BR 9813982A BR 9813982 A BR9813982 A BR 9813982A BR 9813982 A BR9813982 A BR 9813982A
Authority
BR
Brazil
Prior art keywords
antiestrogen
oral contraceptives
contraceptives containing
plus progestin
progestin
Prior art date
Application number
BR9813982-7A
Other languages
English (en)
Inventor
Michael Jay Gast
Christopher Paul Miller
Original Assignee
Americam Home Products Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Americam Home Products Corp filed Critical Americam Home Products Corp
Publication of BR9813982A publication Critical patent/BR9813982A/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Reproductive Health (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Endocrinology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Patente de Invenção: <B>"ANTICONCEPCIONAIS ORAIS CONTENDO ANTIESTROGêNIO MAIS PROGESTINA"<D>. Esta invenção refere-se a um método para proporcionar anticoncepção que compreende a administração a uma mulher em idade procriativa de uma combinação de antiestrogênio não-uterotrófico e uma progestina por 28 dias por ciclo menstrual de 28 dias.
BR9813982-7A 1997-11-06 1998-11-04 Anticoncepcionais orais contendo antiestrogênio mais progestina BR9813982A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US96508397A 1997-11-06 1997-11-06
PCT/US1998/023427 WO1999024027A2 (en) 1997-11-06 1998-11-04 Anti-estrogen plus progestin containing oral contraceptives

Publications (1)

Publication Number Publication Date
BR9813982A true BR9813982A (pt) 2000-09-26

Family

ID=25509417

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9813982-7A BR9813982A (pt) 1997-11-06 1998-11-04 Anticoncepcionais orais contendo antiestrogênio mais progestina

Country Status (28)

Country Link
EP (1) EP1051179B1 (pt)
JP (1) JP2001522798A (pt)
CN (1) CN1278732A (pt)
AR (1) AR016667A1 (pt)
AT (1) ATE304359T1 (pt)
AU (2) AU760540B2 (pt)
BG (1) BG104451A (pt)
BR (1) BR9813982A (pt)
CA (1) CA2307210A1 (pt)
CZ (1) CZ294155B6 (pt)
DE (1) DE69831605T2 (pt)
DK (1) DK1051179T3 (pt)
EA (1) EA200000492A1 (pt)
EE (1) EE04092B1 (pt)
ES (1) ES2246541T3 (pt)
GE (1) GEP20043290B (pt)
HR (1) HRP20000269A2 (pt)
HU (1) HUP0100293A3 (pt)
ID (1) ID24568A (pt)
IL (1) IL135621A0 (pt)
NO (1) NO20002167L (pt)
NZ (1) NZ503890A (pt)
PL (1) PL340623A1 (pt)
SK (1) SK6482000A3 (pt)
TR (1) TR200001268T2 (pt)
UA (1) UA68365C2 (pt)
WO (1) WO1999024027A2 (pt)
ZA (1) ZA9810136B (pt)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL120263A0 (en) * 1996-02-28 1997-06-10 Pfizer Combination therapy to prevent bone loss-progesterone and estrogen agonists
US6479535B1 (en) 1998-05-15 2002-11-12 Wyeth 2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indole and estrogen formulations
UA66861C2 (uk) * 1998-05-15 2004-06-15 Уайт 2-феніл-1-[4-(2-аміноетокси)бензил]індол в комбінації з естрогенами, способи лікування та продукт для лікування
US6380166B1 (en) 1999-09-13 2002-04-30 American Home Products Corporation Glucopyranosides conjugates of 2-(4-hydroxy-phenyl)-3-methyl-1-[4-(2-amin-1-yl-ethoxy)-benzyl]-1H-indol-5-ols
WO2001019839A1 (en) * 1999-09-13 2001-03-22 American Home Products Corporation Glucopyranosides conjugates of 2-(4-hydroxy-phenyl)-1-[4-(2-amin-1-yl-ethoxy)-benzyl]-1h-indol-5-ols
US6376486B1 (en) * 2000-07-06 2002-04-23 American Home Products Corporation Methods of inhibiting sphincter incontinence
WO2003011282A1 (en) 2001-07-31 2003-02-13 Pfizer Products Inc. Pharmaceutical compositions, kits and methods comprising combinations of estrogen agonists/antagonists, estrogens and progestins
EP1809602B1 (en) 2004-10-27 2008-10-29 Janssen Pharmaceutica N.V. Indole derivatives useful as progesterone receptor modulators
FR2880625B1 (fr) * 2005-01-07 2007-03-09 Sanofi Aventis Sa Derives de n-(heteroaryl)-1h-indole-2-carboxamides, leur preparation et leur application en therapeutique
UY29527A1 (es) * 2005-05-13 2006-12-29 Schering Ag Composicinn farmaccutica que contienen gestrgenos y/o estrngenos y 5-metil - (6s) - tetrhidrofolato.
DE102008057230A1 (de) * 2008-11-11 2010-05-12 Bayer Schering Pharma Aktiengesellschaft Synergistische pharmazeutische Kombination mit einem Estrogenrezeptorantagonisten und einem Progestin
EP2580210B1 (en) 2010-06-10 2017-03-01 Seragon Pharmaceuticals, Inc. Estrogen receptor modulators and uses thereof
US9187460B2 (en) 2011-12-14 2015-11-17 Seragon Pharmaceuticals, Inc. Estrogen receptor modulators and uses thereof
AU2016331065B2 (en) 2015-10-01 2021-04-29 Olema Pharmaceuticals, Inc. Tetrahydro-1H-pyrido(3,4-b)indole anti-estrogenic drugs
EP3386968A4 (en) 2015-12-09 2019-09-25 The Board of Trustees of the University of Illinois BENZOTHIOPHEN-BASED SELECTIVE ESTROGEN RECEPTOR-DOWN-REGULATING PREPARATIONS
EP3455218A4 (en) 2016-05-10 2019-12-18 C4 Therapeutics, Inc. C3 CARBON-BASED GLUTARIMIDE DEGRONIMERS FOR TARGET PROTEIN REDUCTION
EP3454856A4 (en) 2016-05-10 2019-12-25 C4 Therapeutics, Inc. HETEROCYCLIC DEGRONIMERS FOR TARGET PROTEIN REDUCTION
WO2017197036A1 (en) 2016-05-10 2017-11-16 C4 Therapeutics, Inc. Spirocyclic degronimers for target protein degradation
CN109789143A (zh) 2016-07-01 2019-05-21 G1治疗公司 基于嘧啶的抗增殖剂
WO2018081168A2 (en) 2016-10-24 2018-05-03 The Board Of Trustees Of The University Of Illinois Benzothiophene-based selective mixed estrogen receptor downregulators
BR112019013814A2 (pt) 2017-01-06 2020-01-21 G1 Therapeutics Inc método para tratamento de câncer ou de um tumor em um indivíduo, composição farmacêutica, combinação, e, kit.
AU2018217809A1 (en) 2017-02-10 2019-08-22 G1 Therapeutics, Inc. Benzothiophene estrogen receptor modulators
WO2019006393A1 (en) 2017-06-29 2019-01-03 G1 Therapeutics, Inc. MORPHIC FORMS OF GIT38 AND METHODS OF MAKING SAME
CN113453679A (zh) 2018-12-20 2021-09-28 C4医药公司 靶向蛋白降解
WO2024030968A1 (en) 2022-08-03 2024-02-08 Brystol-Myers Squibb Company Compounds for modulating ret protein
WO2024097989A1 (en) 2022-11-04 2024-05-10 Bristol-Myers Squibb Company Ret-ldd protein degraders
WO2024097980A1 (en) 2022-11-04 2024-05-10 Bristol-Myers Squibb Company Ret-ldd protein inhibitors

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA716118B (en) * 1970-10-05 1972-05-31 Richardson Merrell Inc Contraception
ZA9510926B (en) * 1994-12-23 1996-07-03 Schering Ag Compounds with progesterone-antagonistic and antiestrogenic action to be used together for female contraception
IL120266A (en) * 1996-02-28 2005-05-17 Pfizer Use of estrogen antagonists and estrogen agonists in the preparation of medicaments for inhibiting pathological conditions
IL120263A0 (en) * 1996-02-28 1997-06-10 Pfizer Combination therapy to prevent bone loss-progesterone and estrogen agonists
DK0802183T3 (da) * 1996-04-19 2002-02-04 American Home Prod Østrogenforbindelser
US5747480A (en) * 1996-05-08 1998-05-05 American Home Products Corporation Oral contraceptive

Also Published As

Publication number Publication date
SK6482000A3 (en) 2000-11-07
ATE304359T1 (de) 2005-09-15
EE200000211A (et) 2001-04-16
AU760540B2 (en) 2003-05-15
WO1999024027A3 (en) 1999-07-15
UA68365C2 (en) 2004-08-16
CN1278732A (zh) 2001-01-03
NO20002167L (no) 2000-06-28
ZA9810136B (en) 2000-05-05
GEP20043290B (en) 2004-07-26
EP1051179B1 (en) 2005-09-14
BG104451A (en) 2000-12-29
EE04092B1 (et) 2003-08-15
CZ20001661A3 (cs) 2000-12-13
WO1999024027A2 (en) 1999-05-20
ID24568A (id) 2000-07-27
HUP0100293A3 (en) 2002-12-28
DK1051179T3 (da) 2005-10-31
NO20002167D0 (no) 2000-04-27
TR200001268T2 (tr) 2001-01-22
EA200000492A1 (ru) 2000-10-30
JP2001522798A (ja) 2001-11-20
CZ294155B6 (cs) 2004-10-13
HRP20000269A2 (en) 2000-12-31
AR016667A1 (es) 2001-07-25
DE69831605T2 (de) 2006-06-14
AU2003204896B2 (en) 2006-06-15
EP1051179A2 (en) 2000-11-15
PL340623A1 (en) 2001-02-12
CA2307210A1 (en) 1999-05-20
IL135621A0 (en) 2001-05-20
DE69831605D1 (de) 2005-10-20
NZ503890A (en) 2002-08-28
ES2246541T3 (es) 2006-02-16
AU1303199A (en) 1999-05-31
HUP0100293A2 (hu) 2001-10-28

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Legal Events

Date Code Title Description
B25D Requested change of name of applicant approved
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B15K Others concerning applications: alteration of classification

Free format text: ALTERADA DE INT.CL.8: A61K 31/57, A61K 31/495, A61P 15/18

Ipc: A61K 31/57 (2007.01), A61K 31/495 (2007.01), A61P

B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: IDEFERIMENTO DO PRESENTE PEDIDO, UMA VEZ QUE O PRESENTE PEDIDO NAO ATENDE AO DISPOSTO NOS ARTIGOS 8O, 15 E 25 DA LPI

B12B Appeal against refusal [chapter 12.2 patent gazette]