BR9608473A - Complexo organometálico do ferro, composição para o tratamento do paludismo, e, utilização de um composto - Google Patents
Complexo organometálico do ferro, composição para o tratamento do paludismo, e, utilização de um compostoInfo
- Publication number
- BR9608473A BR9608473A BR9608473-1A BR9608473A BR9608473A BR 9608473 A BR9608473 A BR 9608473A BR 9608473 A BR9608473 A BR 9608473A BR 9608473 A BR9608473 A BR 9608473A
- Authority
- BR
- Brazil
- Prior art keywords
- malaria
- compound
- treatment
- composition
- iron complex
- Prior art date
Links
- -1 Organometallic iron complex Chemical class 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 title abstract 2
- 201000004792 malaria Diseases 0.000 title abstract 2
- XEEYBQQBJWHFJM-UHFFFAOYSA-N Iron Chemical compound [Fe] XEEYBQQBJWHFJM-UHFFFAOYSA-N 0.000 abstract 3
- LOUPRKONTZGTKE-WZBLMQSHSA-N Quinine Chemical compound C([C@H]([C@H](C1)C=C)C2)C[N@@]1[C@@H]2[C@H](O)C1=CC=NC2=CC=C(OC)C=C21 LOUPRKONTZGTKE-WZBLMQSHSA-N 0.000 abstract 2
- WHTVZRBIWZFKQO-AWEZNQCLSA-N (S)-chloroquine Chemical compound ClC1=CC=C2C(N[C@@H](C)CCCN(CC)CC)=CC=NC2=C1 WHTVZRBIWZFKQO-AWEZNQCLSA-N 0.000 abstract 1
- 235000001258 Cinchona calisaya Nutrition 0.000 abstract 1
- 230000000078 anti-malarial effect Effects 0.000 abstract 1
- 229960003677 chloroquine Drugs 0.000 abstract 1
- WHTVZRBIWZFKQO-UHFFFAOYSA-N chloroquine Natural products ClC1=CC=C2C(NC(C)CCCN(CC)CC)=CC=NC2=C1 WHTVZRBIWZFKQO-UHFFFAOYSA-N 0.000 abstract 1
- LOUPRKONTZGTKE-UHFFFAOYSA-N cinchonine Natural products C1C(C(C2)C=C)CCN2C1C(O)C1=CC=NC2=CC=C(OC)C=C21 LOUPRKONTZGTKE-UHFFFAOYSA-N 0.000 abstract 1
- KTWOOEGAPBSYNW-UHFFFAOYSA-N ferrocene Chemical group [Fe+2].C=1C=C[CH-]C=1.C=1C=C[CH-]C=1 KTWOOEGAPBSYNW-UHFFFAOYSA-N 0.000 abstract 1
- 229910052742 iron Inorganic materials 0.000 abstract 1
- 229960000948 quinine Drugs 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F15/00—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table
- C07F15/02—Iron compounds
- C07F15/025—Iron compounds without a metal-carbon linkage
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A61P33/06—Antimalarials
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F15/00—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table
- C07F15/02—Iron compounds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F17/00—Metallocenes
- C07F17/02—Metallocenes of metals of Groups 8, 9 or 10 of the Periodic System
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Tropical Medicine & Parasitology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9505532A FR2733985B1 (fr) | 1995-05-10 | 1995-05-10 | Complexes organometalliques du fer antipaludiques |
PCT/FR1996/000721 WO1996035698A1 (fr) | 1995-05-10 | 1996-05-10 | Complexes organometalliques du fer antipaludiques |
Publications (1)
Publication Number | Publication Date |
---|---|
BR9608473A true BR9608473A (pt) | 1999-11-30 |
Family
ID=9478836
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR9608473-1A BR9608473A (pt) | 1995-05-10 | 1996-05-10 | Complexo organometálico do ferro, composição para o tratamento do paludismo, e, utilização de um composto |
Country Status (14)
Country | Link |
---|---|
US (1) | US6127543A (pt) |
EP (1) | EP0824536B1 (pt) |
JP (1) | JP4394163B2 (pt) |
AP (1) | AP953A (pt) |
AT (1) | ATE204581T1 (pt) |
AU (1) | AU718946B2 (pt) |
BR (1) | BR9608473A (pt) |
DE (1) | DE69614679T2 (pt) |
DK (1) | DK0824536T3 (pt) |
ES (1) | ES2163022T3 (pt) |
FR (1) | FR2733985B1 (pt) |
OA (1) | OA10535A (pt) |
PT (1) | PT824536E (pt) |
WO (1) | WO1996035698A1 (pt) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0205455D0 (en) | 2002-03-07 | 2002-04-24 | Molecular Sensing Plc | Nucleic acid probes, their synthesis and use |
FR2952823B1 (fr) | 2009-10-30 | 2012-04-20 | Sanofi Aventis | Utilisation de la ferroquine dans le traitement ou la prevention du paludisme |
FR2951945B1 (fr) | 2009-11-05 | 2013-08-09 | Sanofi Aventis | Composition pharmaceutique |
FR2961209B1 (fr) * | 2010-06-11 | 2013-03-01 | Sanofi Aventis | Procede de synthese de la ferroquine par amination reductrice convergente. |
WO2012104204A1 (en) | 2011-01-31 | 2012-08-09 | Vifor (International) Ag | Iron-carbohydrate complex compounds for the intravenous therapy of malaria |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1470210A (en) * | 1974-10-30 | 1977-04-14 | Edwards E | Organometallic derivatives of penicillin |
DE2815930A1 (de) * | 1978-04-13 | 1979-10-18 | Bayer Ag | Duengemittel zur versorgung von pflanzen mit eisen |
EP0214933A3 (de) * | 1985-09-03 | 1989-05-24 | Ciba-Geigy Ag | Kombinationspräparate zur Behandlung von Malaria |
-
1995
- 1995-05-10 FR FR9505532A patent/FR2733985B1/fr not_active Expired - Lifetime
-
1996
- 1996-05-10 WO PCT/FR1996/000721 patent/WO1996035698A1/fr active IP Right Grant
- 1996-05-10 PT PT96916196T patent/PT824536E/pt unknown
- 1996-05-10 ES ES96916196T patent/ES2163022T3/es not_active Expired - Lifetime
- 1996-05-10 BR BR9608473-1A patent/BR9608473A/pt not_active IP Right Cessation
- 1996-05-10 DE DE69614679T patent/DE69614679T2/de not_active Expired - Lifetime
- 1996-05-10 AU AU59037/96A patent/AU718946B2/en not_active Expired
- 1996-05-10 DK DK96916196T patent/DK0824536T3/da active
- 1996-05-10 EP EP96916196A patent/EP0824536B1/fr not_active Expired - Lifetime
- 1996-05-10 AT AT96916196T patent/ATE204581T1/de active
- 1996-05-10 AP APAP/P/1997/001141A patent/AP953A/en active
- 1996-05-10 US US08/952,093 patent/US6127543A/en not_active Expired - Lifetime
- 1996-05-10 JP JP53384296A patent/JP4394163B2/ja not_active Expired - Lifetime
-
1997
- 1997-11-10 OA OA70125A patent/OA10535A/fr unknown
Also Published As
Publication number | Publication date |
---|---|
AU5903796A (en) | 1996-11-29 |
PT824536E (pt) | 2002-02-28 |
JP4394163B2 (ja) | 2010-01-06 |
DE69614679T2 (de) | 2002-06-27 |
DK0824536T3 (da) | 2001-12-17 |
EP0824536A1 (fr) | 1998-02-25 |
US6127543A (en) | 2000-10-03 |
ES2163022T3 (es) | 2002-01-16 |
DE69614679D1 (de) | 2001-09-27 |
FR2733985B1 (fr) | 1997-07-18 |
OA10535A (fr) | 2002-04-26 |
ATE204581T1 (de) | 2001-09-15 |
AP953A (en) | 2001-04-02 |
JPH11511738A (ja) | 1999-10-12 |
AU718946B2 (en) | 2000-05-04 |
WO1996035698A1 (fr) | 1996-11-14 |
EP0824536B1 (fr) | 2001-08-22 |
FR2733985A1 (fr) | 1996-11-15 |
AP9701141A0 (en) | 1998-01-31 |
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Legal Events
Date | Code | Title | Description |
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FB36 | Technical and formal requirements: requirement - article 36 of industrial property law | ||
FB36 | Technical and formal requirements: requirement - article 36 of industrial property law | ||
B06A | Patent application procedure suspended [chapter 6.1 patent gazette] | ||
B09A | Decision: intention to grant [chapter 9.1 patent gazette] | ||
B16A | Patent or certificate of addition of invention granted [chapter 16.1 patent gazette] |
Free format text: PRAZO DE VALIDADE: 10 (DEZ) ANOS CONTADOS A PARTIR DE 01/08/2006, OBSERVADAS AS CONDICOES LEGAIS. |
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B22O | Other matters related to patents and certificates of addition of invention: legal action concerning patent |
Free format text: INPI-52400.061556/2013 ORIGEM: JUIZO DA 013A VARA FEDERAL DO RIO DE JANEIRO PROCESSO NO 0132361-55.2013.4.02.5101 ACAO DE NULIDADE DAS PATENTES SUBMETIDAS AO MAILBOX (ART. 229, PARAGRAFO UNICO DA LPI); ALTERNATIVAMENTE, A DECRETACAO DA NULIDADE PARCIAL PARA CORRECAO DO PRAZO DE VIGENCIA; SUBSIDIARIAMENTE, CASO SE ENTENDA NAO SER O CASO DE NULIDADE, A CORRECAO DO ATO ADMINISTRATIVO PARA ADEQUACAO DA VIGENCIA DAS PATENTES. AUTOR: INSTITUTO NACIONAL DA PROPRIEDADE INDUSTRIAL - INPI REU:UNIVERSITE DES SCIENCES ET TECHNOLOGIES DE LILLE, WYETH HOLDINGS CORPORATION, YEDA RESEARCH AND DEVELOPMENT CO LTD. |
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B21B | Extinction acc. art. 78, item ii - on waiver by the patentee, without prejudice to the rights of third parties |
Free format text: HOMOLOGADA A RENUNCIA DA PATENTE, SOLICITADA ATRAVES DA PETICAO DEINPI/RJ NO 020140004672 DE 03/02/2014. |