BR9508482A - Novos derivados do imidazol seu processo de preparo os novos intermedíarios obtidos sua aplicação a título de medicamentos e as composições farmacéuticas que os comtém - Google Patents

Novos derivados do imidazol seu processo de preparo os novos intermedíarios obtidos sua aplicação a título de medicamentos e as composições farmacéuticas que os comtém

Info

Publication number
BR9508482A
BR9508482A BR9508482A BR9508482A BR9508482A BR 9508482 A BR9508482 A BR 9508482A BR 9508482 A BR9508482 A BR 9508482A BR 9508482 A BR9508482 A BR 9508482A BR 9508482 A BR9508482 A BR 9508482A
Authority
BR
Brazil
Prior art keywords
pct
new
medicines
imidazole
contain
Prior art date
Application number
BR9508482A
Other languages
English (en)
Inventor
Bertrand Heckmann
Jean-Paul Vevert
Jidong Zhang
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of BR9508482A publication Critical patent/BR9508482A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/02Nutrients, e.g. vitamins, minerals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Nutrition Science (AREA)
  • Diabetes (AREA)
  • Vascular Medicine (AREA)
  • Obesity (AREA)
  • Pulmonology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BR9508482A 1994-08-02 1995-08-01 Novos derivados do imidazol seu processo de preparo os novos intermedíarios obtidos sua aplicação a título de medicamentos e as composições farmacéuticas que os comtém BR9508482A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9409565A FR2723369B1 (fr) 1994-08-02 1994-08-02 Nouveaux derives de l'imidazole, leur procede de preparation, les nouveaux intermediaires obtenus, leur application a titre de medicaments et les compositions pharmaceutiques les renfermant.
PCT/FR1995/001033 WO1996004275A1 (fr) 1994-08-02 1995-08-01 Nouveaux derives de l'imidazole, leur procede de preparation, les nouveaux intermediaires obtenus, leur application a titre de medicaments et les compositions pharmaceutiques les renfermant

Publications (1)

Publication Number Publication Date
BR9508482A true BR9508482A (pt) 1999-06-01

Family

ID=9465985

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9508482A BR9508482A (pt) 1994-08-02 1995-08-01 Novos derivados do imidazol seu processo de preparo os novos intermedíarios obtidos sua aplicação a título de medicamentos e as composições farmacéuticas que os comtém

Country Status (18)

Country Link
US (1) US5856509A (pt)
EP (1) EP0804435B1 (pt)
JP (1) JP3950475B2 (pt)
CN (1) CN1083838C (pt)
AT (1) ATE261442T1 (pt)
AU (1) AU703078B2 (pt)
BR (1) BR9508482A (pt)
CA (1) CA2196219A1 (pt)
DE (1) DE69532684T2 (pt)
ES (1) ES2214504T3 (pt)
FI (1) FI970423A (pt)
FR (1) FR2723369B1 (pt)
HU (1) HU221463B (pt)
IL (1) IL114663A0 (pt)
MX (1) MX9700820A (pt)
RU (1) RU2171257C2 (pt)
WO (1) WO1996004275A1 (pt)
ZA (1) ZA956450B (pt)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2740774B1 (fr) * 1995-11-08 1997-12-19 Roussel Uclaf Nouveaux derives d'imidazole n-benzyldioxole, leur procede de preparation, leur application a titre de medicaments, compositions pharmaceutiques et nouvelle utilisation
WO1998052551A1 (fr) * 1997-05-22 1998-11-26 Kyowa Hakko Kogyo Co., Ltd. Composes bisaryle et remedes contre le cancer contenant ces composes
EP2095819A1 (en) * 2008-02-28 2009-09-02 Maastricht University N-benzyl imidazole derivatives and their use as aldosterone synthase inhibitors

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2862340D1 (en) * 1978-02-01 1983-11-24 Wellcome Found Imidazole derivatives and salts thereof, their synthesis, and pharmaceutical formulations thereof
JPH07509465A (ja) * 1992-07-17 1995-10-19 スミスクライン・ビーチャム・コーポレイション エンドセリン受容体アンタゴニスト

Also Published As

Publication number Publication date
DE69532684D1 (de) 2004-04-22
AU3117895A (en) 1996-03-04
ES2214504T3 (es) 2004-09-16
US5856509A (en) 1999-01-05
HUT76838A (en) 1997-11-28
JPH10503512A (ja) 1998-03-31
EP0804435A1 (fr) 1997-11-05
ZA956450B (en) 1996-08-05
MX9700820A (es) 1997-05-31
FI970423A0 (fi) 1997-01-31
RU2171257C2 (ru) 2001-07-27
AU703078B2 (en) 1999-03-11
JP3950475B2 (ja) 2007-08-01
CA2196219A1 (fr) 1996-02-15
EP0804435B1 (fr) 2004-03-10
CN1083838C (zh) 2002-05-01
WO1996004275A1 (fr) 1996-02-15
FI970423A (fi) 1997-04-01
FR2723369B1 (fr) 1996-09-13
HU221463B (en) 2002-10-28
IL114663A0 (en) 1995-11-27
DE69532684T2 (de) 2004-07-29
CN1159805A (zh) 1997-09-17
FR2723369A1 (fr) 1996-02-09
ATE261442T1 (de) 2004-03-15

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Legal Events

Date Code Title Description
PC Transfer

Owner name: HOECHST MARION ROUSSEL (FR)

B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]