BR6683864D0 - Processo para a preparacao de um composto de citosina - Google Patents

Processo para a preparacao de um composto de citosina

Info

Publication number
BR6683864D0
BR6683864D0 BR183864/66A BR18386466A BR6683864D0 BR 6683864 D0 BR6683864 D0 BR 6683864D0 BR 183864/66 A BR183864/66 A BR 183864/66A BR 18386466 A BR18386466 A BR 18386466A BR 6683864 D0 BR6683864 D0 BR 6683864D0
Authority
BR
Brazil
Prior art keywords
cytosine
compound
preparation
Prior art date
Application number
BR183864/66A
Other languages
English (en)
Portuguese (pt)
Inventor
R Duschinsky
M Hoffer
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of BR6683864D0 publication Critical patent/BR6683864D0/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06—Pyrimidine radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BR183864/66A 1965-10-22 1966-10-21 Processo para a preparacao de um composto de citosina BR6683864D0 (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US502586A US3309359A (en) 1965-10-22 1965-10-22 N-mono-acyl-5-fluorocytosine derivatives and process

Publications (1)

Publication Number Publication Date
BR6683864D0 true BR6683864D0 (pt) 1973-12-26

Family

ID=23998481

Family Applications (1)

Application Number Title Priority Date Filing Date
BR183864/66A BR6683864D0 (pt) 1965-10-22 1966-10-21 Processo para a preparacao de um composto de citosina

Country Status (11)

Country Link
US (1) US3309359A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
BE (1) BE688539A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
BR (1) BR6683864D0 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CH (1) CH475258A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DE (1) DE1695160A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DK (1) DK115474B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FR (1) FR5908M (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
GB (1) GB1110357A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IL (1) IL26726A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NL (1) NL6614240A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
SE (1) SE330176B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)

Families Citing this family (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3894000A (en) * 1971-01-27 1975-07-08 Upjohn Co Ara-cytidine derivatives and process of preparation
US3975367A (en) * 1971-06-08 1976-08-17 The Upjohn Company Arabinofuranosyl N4 -aminoacyl cytosine containing compounds
US4022963A (en) * 1972-06-08 1977-05-10 Deutsch Daniel Harold Acetylation process for nucleoside compounds
US3991045A (en) * 1973-05-30 1976-11-09 Asahi Kasei Kogyo Kabushiki Kaisha N4 -acylarabinonucleosides
JPS5159880A (en) * 1974-11-22 1976-05-25 Asahi Chemical Ind N44 ashirunukureoshidojikarubonsanesuteruno seiho
JPS5924999B2 (ja) * 1978-06-10 1984-06-13 富山化学工業株式会社 新規な５−フルオロ−２′−デオキシ−β−ウリジン誘導体の製造法
JPS5535057A (en) * 1978-09-05 1980-03-11 Funai Corp 2'-deoxy-5-fluorouridine derivative, its preparation, and antitumor agent comprising it
JPS59167600A (ja) * 1983-03-14 1984-09-21 Microbial Chem Res Found ２′−デオキシオキザノシンおよびその製造法
JP2005519916A (ja) 2001-12-14 2005-07-07 フアーマセツト・リミテツド ウィルス感染治療用ｎ４−アシルシトシンヌクレオシド類
UA107445C2 (uk) * 2008-01-22 2015-01-12 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі 5-фторпіримідинові похідні як фунгіциди
KR20110042204A (ko) 2008-08-01 2011-04-25 다우 아그로사이언시즈 엘엘씨 살진균제로서의 5-플루오로시토신의 용도
UA112284C2 (uk) * 2009-08-07 2016-08-25 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Похідні 5-фторпіримідинону
UA107671C2 (en) * 2009-08-07 2015-02-10 Dow Agrosciences Llc N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
PT2462134E (pt) 2009-08-07 2014-07-28 Dow Agrosciences Llc Derivados de n1-sulfonil-5-fluoropirimidinona
UA106889C2 (uk) * 2009-08-07 2014-10-27 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Похідні n1-ацил-5-фторпіримідинону
US8921382B2 (en) * 2010-01-07 2014-12-30 Dow Agrosciences, Llc. Thiazolo[5,4-d] pyrimidines and their use as agrochemicals
KR102012992B1 (ko) 2011-08-17 2019-08-21 아다마 마켓심 리미티드 5-플루오로-4-이미노-3-(치환된)-3,4-디히드로피리미딘-2-(1ｈ)-온 유도체
RU2656101C2 (ru) 2012-12-28 2018-05-31 Адама Мактешим Лтд. Производные 1-(замещенный бензоил)-5-фтор-4-имино-3-метил-3,4-дигидропиримидин-2(1h)-она
UA117743C2 (uk) 2012-12-28 2018-09-25 Адама Махтешім Лтд. N-(заміщені)-5-фтор-4-іміно-3-метил-2-оксо-3,4-дигідропіримідин-1(2h)-карбоксамідні похідні
DK2938194T3 (da) 2012-12-28 2020-01-02 Adama Makhteshim Ltd N-(substituerede)-5-fluor-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidin-1 (2h)-carboxylatderivater
NZ708981A (en) 2012-12-31 2020-01-31 Adama Makhteshim Ltd 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides
JP6608366B2 (ja) 2013-12-31 2019-11-20 アダマ・マクテシム・リミテッド 真菌防除のための相乗的殺真菌性混合物および組成物
CN106068268A (zh) 2013-12-31 2016-11-02 阿达玛马克西姆股份有限公司 5‑氟‑4‑亚氨基‑3‑（烷基/取代烷基）‑1‑（芳基磺酰基）‑3,4‑二氢嘧啶‑2（1h）‑酮及其制备方法
CN118515619A (zh) 2017-07-17 2024-08-20 阿达玛克西姆股份有限公司 5-氟-4-亚氨基-3-甲基-1-甲苯磺酰基-3,4-二氢嘧啶-2-酮的多晶型物
CN109651467A (zh) * 2019-01-15 2019-04-19 齐鲁天和惠世制药有限公司 一种卡培他滨杂质及其制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2949451A (en) * 1959-04-21 1960-08-16 Hoffmann La Roche Preparation of thymidine and deoxyfluorouridine, and intermediates therefor
NL299755A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) * 1959-06-03
GB1070413A (en) * 1962-11-15 1967-06-01 Sankyo Co A process for preparing purine and pyrimidine nucleosides

Also Published As

Publication number Publication date
DK115474B (da) 1969-10-13
SE330176B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1970-11-09
NL6614240A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1967-04-24
IL26726A (en) 1970-06-17
FR5908M (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1968-03-25
CH475258A (de) 1969-07-15
US3309359A (en) 1967-03-14
BE688539A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1967-04-20
GB1110357A (en) 1968-04-18
DE1695160A1 (de) 1970-12-17

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