BR112023003690A2 - Conjugado ou sal farmaceuticamente aceitável do mesmo, composição, radiofármaco, kit de peças, uso do conjugado ou sal e uso do kit de peças - Google Patents

Conjugado ou sal farmaceuticamente aceitável do mesmo, composição, radiofármaco, kit de peças, uso do conjugado ou sal e uso do kit de peças

Info

Publication number
BR112023003690A2
BR112023003690A2 BR112023003690A BR112023003690A BR112023003690A2 BR 112023003690 A2 BR112023003690 A2 BR 112023003690A2 BR 112023003690 A BR112023003690 A BR 112023003690A BR 112023003690 A BR112023003690 A BR 112023003690A BR 112023003690 A2 BR112023003690 A2 BR 112023003690A2
Authority
BR
Brazil
Prior art keywords
conjugate
kit
parts
salt
pharmaceutically acceptable
Prior art date
Application number
BR112023003690A
Other languages
English (en)
Portuguese (pt)
Inventor
Torgue Julien
Stallons Tania
Wong Amy
Saidi Amal
Original Assignee
Orano Med
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Orano Med filed Critical Orano Med
Publication of BR112023003690A2 publication Critical patent/BR112023003690A2/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K51/00Preparations containing radioactive substances for use in therapy or testing in vivo
    • A61K51/02Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
    • A61K51/04Organic compounds
    • A61K51/08Peptides, e.g. proteins, carriers being peptides, polyamino acids, proteins
    • A61K51/088Peptides, e.g. proteins, carriers being peptides, polyamino acids, proteins conjugates with carriers being peptides, polyamino acids or proteins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/02Linear peptides containing at least one abnormal peptide link
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/06Linear peptides containing only normal peptide links having 5 to 11 amino acids

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Optics & Photonics (AREA)
  • Epidemiology (AREA)
  • Physics & Mathematics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BR112023003690A 2020-09-28 2021-09-22 Conjugado ou sal farmaceuticamente aceitável do mesmo, composição, radiofármaco, kit de peças, uso do conjugado ou sal e uso do kit de peças BR112023003690A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP20306109.8A EP3973999A1 (en) 2020-09-28 2020-09-28 Conjugate or its salt comprising a gastrin-releasing peptide receptor antagonist and uses thereof
PCT/EP2021/076107 WO2022063850A1 (en) 2020-09-28 2021-09-22 Conjugate or its salt comprising a gastrin-releasing peptide receptor antagonist and uses thereof

Publications (1)

Publication Number Publication Date
BR112023003690A2 true BR112023003690A2 (pt) 2023-04-04

Family

ID=74180915

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112023003690A BR112023003690A2 (pt) 2020-09-28 2021-09-22 Conjugado ou sal farmaceuticamente aceitável do mesmo, composição, radiofármaco, kit de peças, uso do conjugado ou sal e uso do kit de peças

Country Status (21)

Country Link
US (1) US20230372552A1 (https=)
EP (2) EP3973999A1 (https=)
JP (1) JP7824281B2 (https=)
KR (1) KR20230078690A (https=)
CN (1) CN116322798A (https=)
AU (1) AU2021348219A1 (https=)
BR (1) BR112023003690A2 (https=)
CA (1) CA3189680A1 (https=)
DK (1) DK4188457T3 (https=)
ES (1) ES2989009T3 (https=)
FI (1) FI4188457T3 (https=)
HR (1) HRP20241285T1 (https=)
HU (1) HUE068360T2 (https=)
IL (1) IL300486A (https=)
LT (1) LT4188457T (https=)
PL (1) PL4188457T3 (https=)
PT (1) PT4188457T (https=)
RS (1) RS65994B1 (https=)
SI (1) SI4188457T1 (https=)
SM (1) SMT202400392T1 (https=)
WO (1) WO2022063850A1 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2025163083A1 (en) 2024-01-31 2025-08-07 Molecular Partners Ag Recobminant dll3 binding proteins and their use

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2100900A1 (en) 2008-03-07 2009-09-16 Universitätsspital Basel Bombesin analog peptide antagonist conjugates
US20150217006A1 (en) * 2014-02-06 2015-08-06 Immunomedics, Inc. Al-f-18-labeled, al-f-19-labeled and ga-68-labeled gastrin-releasing peptide receptor (grpr)-antagonists for imaging of prostate cancer
HRP20231458T1 (hr) * 2017-01-12 2024-05-10 Radiomedix Inc. Liječenje stanica raka koje prekomjerno eksprimiraju receptore za somatostatin primjenom derivata oktreotida keliranih sa radioizotopima

Also Published As

Publication number Publication date
JP7824281B2 (ja) 2026-03-04
AU2021348219A1 (en) 2023-03-09
KR20230078690A (ko) 2023-06-02
SI4188457T1 (sl) 2025-01-31
LT4188457T (lt) 2024-12-27
SMT202400392T1 (it) 2024-11-15
PT4188457T (pt) 2024-09-10
CN116322798A (zh) 2023-06-23
WO2022063850A1 (en) 2022-03-31
DK4188457T3 (da) 2024-08-26
US20230372552A1 (en) 2023-11-23
FI4188457T3 (fi) 2024-09-23
HRP20241285T1 (hr) 2025-01-03
RS65994B1 (sr) 2024-10-31
PL4188457T3 (pl) 2025-01-07
EP3973999A1 (en) 2022-03-30
ES2989009T3 (es) 2024-11-25
IL300486A (en) 2023-04-01
EP4188457A1 (en) 2023-06-07
HUE068360T2 (hu) 2024-12-28
JP2023542218A (ja) 2023-10-05
CA3189680A1 (en) 2022-03-31
EP4188457B1 (en) 2024-07-03

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