BR112022026233A2 - Processo para sintetizar lipídios catiônicos - Google Patents
Processo para sintetizar lipídios catiônicosInfo
- Publication number
- BR112022026233A2 BR112022026233A2 BR112022026233A BR112022026233A BR112022026233A2 BR 112022026233 A2 BR112022026233 A2 BR 112022026233A2 BR 112022026233 A BR112022026233 A BR 112022026233A BR 112022026233 A BR112022026233 A BR 112022026233A BR 112022026233 A2 BR112022026233 A2 BR 112022026233A2
- Authority
- BR
- Brazil
- Prior art keywords
- synthesizing
- cation lipids
- lipids
- cation
- targeting
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
- C07C237/02—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton
- C07C237/22—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton having nitrogen atoms of amino groups bound to the carbon skeleton of the acid part, further acylated
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C231/00—Preparation of carboxylic acid amides
- C07C231/02—Preparation of carboxylic acid amides from carboxylic acids or from esters, anhydrides, or halides thereof by reaction with ammonia or amines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
- C07C237/50—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the nitrogen atom of at least one of the carboxamide groups quaternised
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Abstract
PROCESSO PARA SINTETIZAR LIPÍDIOS CATIÔNICOS. A presente invenção refere-se a processos para sintetizar lipídios catiônicos de Fórmula I úteis na síntese de composições solúveis em gordura para direcionamento e aumento da atividade de moléculas terapêuticas, incluindo siRNA.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US202063043518P | 2020-06-24 | 2020-06-24 | |
PCT/US2021/038524 WO2021262745A1 (en) | 2020-06-24 | 2021-06-22 | Process for synthesizing cationic lipids |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112022026233A2 true BR112022026233A2 (pt) | 2023-01-17 |
Family
ID=79281775
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112022026233A BR112022026233A2 (pt) | 2020-06-24 | 2021-06-22 | Processo para sintetizar lipídios catiônicos |
Country Status (11)
Country | Link |
---|---|
US (1) | US20230265050A1 (pt) |
EP (1) | EP4171578A1 (pt) |
JP (1) | JP2023532014A (pt) |
KR (1) | KR20230042022A (pt) |
CN (1) | CN115996730A (pt) |
AU (1) | AU2021297806A1 (pt) |
BR (1) | BR112022026233A2 (pt) |
CA (1) | CA3183536A1 (pt) |
IL (1) | IL299271A (pt) |
MX (1) | MX2022016523A (pt) |
WO (1) | WO2021262745A1 (pt) |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US9011903B2 (en) * | 2011-06-08 | 2015-04-21 | Nitto Denko Corporation | Cationic lipids for therapeutic agent delivery formulations |
AU2013270685B2 (en) * | 2012-06-08 | 2017-11-30 | Nitto Denko Corporation | Lipids for therapeutic agent delivery formulations |
CN106164089B (zh) * | 2014-04-02 | 2020-11-03 | 日东电工株式会社 | 靶向分子及其用途 |
US20180235995A1 (en) * | 2015-02-19 | 2018-08-23 | Nitto Denko Corporation | Rna interference therapeutics against ebola virus |
-
2021
- 2021-06-22 JP JP2022580027A patent/JP2023532014A/ja active Pending
- 2021-06-22 KR KR1020237002608A patent/KR20230042022A/ko unknown
- 2021-06-22 CN CN202180045292.9A patent/CN115996730A/zh active Pending
- 2021-06-22 MX MX2022016523A patent/MX2022016523A/es unknown
- 2021-06-22 US US18/003,232 patent/US20230265050A1/en active Pending
- 2021-06-22 AU AU2021297806A patent/AU2021297806A1/en active Pending
- 2021-06-22 BR BR112022026233A patent/BR112022026233A2/pt unknown
- 2021-06-22 CA CA3183536A patent/CA3183536A1/en active Pending
- 2021-06-22 EP EP21829641.6A patent/EP4171578A1/en active Pending
- 2021-06-22 IL IL299271A patent/IL299271A/en unknown
- 2021-06-22 WO PCT/US2021/038524 patent/WO2021262745A1/en unknown
Also Published As
Publication number | Publication date |
---|---|
EP4171578A1 (en) | 2023-05-03 |
CA3183536A1 (en) | 2021-12-30 |
US20230265050A1 (en) | 2023-08-24 |
CN115996730A (zh) | 2023-04-21 |
IL299271A (en) | 2023-02-01 |
WO2021262745A1 (en) | 2021-12-30 |
JP2023532014A (ja) | 2023-07-26 |
AU2021297806A1 (en) | 2023-02-23 |
KR20230042022A (ko) | 2023-03-27 |
MX2022016523A (es) | 2023-01-30 |
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