BR112022022527A2 - Compostos de metiltionínio para uso no tratamento de covid-19 - Google Patents

Compostos de metiltionínio para uso no tratamento de covid-19

Info

Publication number
BR112022022527A2
BR112022022527A2 BR112022022527A BR112022022527A BR112022022527A2 BR 112022022527 A2 BR112022022527 A2 BR 112022022527A2 BR 112022022527 A BR112022022527 A BR 112022022527A BR 112022022527 A BR112022022527 A BR 112022022527A BR 112022022527 A2 BR112022022527 A2 BR 112022022527A2
Authority
BR
Brazil
Prior art keywords
compounds
covid
methylthionium
treatment
methylthioninium
Prior art date
Application number
BR112022022527A
Other languages
English (en)
Inventor
Arastoo Mohammad
Philip Mazanetz Michel
Michel Wischik Claude
Original Assignee
Wista Lab Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wista Lab Ltd filed Critical Wista Lab Ltd
Publication of BR112022022527A2 publication Critical patent/BR112022022527A2/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/5415Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with carbocyclic ring systems, e.g. phenothiazine, chlorpromazine, piroxicam
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/47064-Aminoquinolines; 8-Aminoquinolines, e.g. chloroquine, primaquine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Virology (AREA)
  • Molecular Biology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)

Abstract

COMPOSTOS DE METILTIONÍNIO PARA USO NO TRATAMENTO DE COVID-19. A presente invenção se refere a métodos de tratamento de COVID-19 em um indivíduo usando compostos de metiltionínio.
BR112022022527A 2020-05-05 2021-04-30 Compostos de metiltionínio para uso no tratamento de covid-19 BR112022022527A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB2006659.3A GB202006659D0 (en) 2020-05-05 2020-05-05 Therapeutic treatments
PCT/EP2021/061481 WO2021224145A1 (en) 2020-05-05 2021-04-30 Methylthioninium compounds for use in the treatment of covid-19

Publications (1)

Publication Number Publication Date
BR112022022527A2 true BR112022022527A2 (pt) 2022-12-13

Family

ID=71080353

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112022022527A BR112022022527A2 (pt) 2020-05-05 2021-04-30 Compostos de metiltionínio para uso no tratamento de covid-19

Country Status (12)

Country Link
US (1) US20230165876A1 (pt)
EP (1) EP4146224A1 (pt)
JP (1) JP2023524127A (pt)
KR (1) KR20230014709A (pt)
CN (1) CN116194107A (pt)
AU (1) AU2021269001A1 (pt)
BR (1) BR112022022527A2 (pt)
CA (1) CA3181391A1 (pt)
GB (1) GB202006659D0 (pt)
MX (1) MX2022013885A (pt)
TW (1) TW202200151A (pt)
WO (1) WO2021224145A1 (pt)

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20060264423A1 (en) 2005-05-20 2006-11-23 Bioenvision, Inc. Methylene Blue Therapy of Viral Disease
PT2013191E (pt) 2006-03-29 2010-10-29 Wista Lab Ltd Sais de 3,7-diamino-10h-fenotiazina e a sua utilização
US9283230B2 (en) * 2011-02-11 2016-03-15 Wista Laboratories Ltd. Phenothiazine diaminium salts and their use
KR102475825B1 (ko) 2016-07-25 2022-12-08 위스타 레보레이토리스 리미티드 디아미노페노티아진 (diaminophenothiazines)의 투여 및 투여량 (dosage)
EP4364801A2 (en) * 2018-07-26 2024-05-08 WisTa Laboratories Ltd. Optimised dosage of diaminophenothiazines in populations

Also Published As

Publication number Publication date
AU2021269001A1 (en) 2022-12-08
US20230165876A1 (en) 2023-06-01
EP4146224A1 (en) 2023-03-15
CN116194107A (zh) 2023-05-30
CA3181391A1 (en) 2021-11-11
KR20230014709A (ko) 2023-01-30
TW202200151A (zh) 2022-01-01
GB202006659D0 (en) 2020-06-17
JP2023524127A (ja) 2023-06-08
WO2021224145A1 (en) 2021-11-11
MX2022013885A (es) 2022-11-30

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Legal Events

Date Code Title Description
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]