BR112022010702A2 - Macrociclos para uso no tratamento de doenças - Google Patents
Macrociclos para uso no tratamento de doençasInfo
- Publication number
- BR112022010702A2 BR112022010702A2 BR112022010702A BR112022010702A BR112022010702A2 BR 112022010702 A2 BR112022010702 A2 BR 112022010702A2 BR 112022010702 A BR112022010702 A BR 112022010702A BR 112022010702 A BR112022010702 A BR 112022010702A BR 112022010702 A2 BR112022010702 A2 BR 112022010702A2
- Authority
- BR
- Brazil
- Prior art keywords
- macrocycles
- diseases
- treatment
- present disclosure
- methods
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/22—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains four or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5383—1,4-Oxazines, e.g. morpholine ortho- or peri-condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Abstract
MACROCICLOS PARA USO NO TRATAMENTO DE DOENÇAS. A presente divulgação refere-se a certos derivados macrocíclicos de diaril quirais, composições farmacêuticas que os contêm e métodos para usá-los para tratar câncer.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201962943098P | 2019-12-03 | 2019-12-03 | |
US202063015937P | 2020-04-27 | 2020-04-27 | |
PCT/US2020/062859 WO2021113339A1 (en) | 2019-12-03 | 2020-12-02 | Macrocycles for use in treating disease |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112022010702A2 true BR112022010702A2 (pt) | 2022-10-04 |
Family
ID=76091584
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112022010702A BR112022010702A2 (pt) | 2019-12-03 | 2020-12-02 | Macrociclos para uso no tratamento de doenças |
Country Status (14)
Country | Link |
---|---|
US (3) | US11634433B2 (pt) |
EP (1) | EP4069700A4 (pt) |
JP (1) | JP2023504523A (pt) |
KR (1) | KR20220133869A (pt) |
CN (1) | CN114929710B (pt) |
AU (1) | AU2020395136A1 (pt) |
BR (1) | BR112022010702A2 (pt) |
CA (1) | CA3163735A1 (pt) |
CO (1) | CO2022008817A2 (pt) |
IL (1) | IL293458A (pt) |
MX (1) | MX2022006853A (pt) |
PE (1) | PE20221485A1 (pt) |
TW (1) | TW202134249A (pt) |
WO (1) | WO2021113339A1 (pt) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN114929710B (zh) | 2019-12-03 | 2024-03-29 | 特普医药公司 | 用于治疗疾病的巨环 |
CN113336774B (zh) * | 2021-06-25 | 2023-05-23 | 江南大学 | 作为trk抑制剂的取代的手性二芳基大环化合物 |
WO2024017380A1 (zh) * | 2022-07-22 | 2024-01-25 | 南京明德新药研发有限公司 | 含三并环的大环类化合物及其应用 |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ATE526330T1 (de) * | 2000-12-28 | 2011-10-15 | Ono Pharmaceutical Co | Heterotrizyklische verbindungen als antagonisten des crf-rezeptors |
US8211891B2 (en) * | 2008-04-30 | 2012-07-03 | Enanta Pharmaceuticals, Inc. | Difluoromethyl-containing macrocyclic compounds as hepatitis C virus inhibitors |
CA2849999A1 (en) | 2011-09-30 | 2013-04-04 | Oncodesign S.A. | Macrocyclic flt3 kinase inhibitors |
CN104513253A (zh) * | 2013-10-01 | 2015-04-15 | 南京波尔泰药业科技有限公司 | 用于治疗增殖性疾病的大环化合物 |
US9714258B2 (en) * | 2014-01-24 | 2017-07-25 | Tp Therapeutics, Inc. | Diaryl macrocycles as modulators of protein kinases |
JP6871903B2 (ja) * | 2015-07-02 | 2021-05-19 | ターニング・ポイント・セラピューティクス・インコーポレイテッドTurning Point Therapeutics,Inc. | プロテインキナーゼのモジュレーターとしてのキラルジアリール大環状分子 |
PL3728271T3 (pl) * | 2017-12-19 | 2023-01-23 | Turning Point Therapeutics, Inc. | Związki makrocykliczne do leczenia chorób |
US20210087206A1 (en) * | 2017-12-19 | 2021-03-25 | Turning Point Therapeutics, Inc. | Macrocyclic kinase inhibitors and their use |
TW201932472A (zh) * | 2018-01-30 | 2019-08-16 | 大陸商上海吉倍生物技術有限公司 | 具有大環分子結構的化合物及其用途 |
CN114929710B (zh) | 2019-12-03 | 2024-03-29 | 特普医药公司 | 用于治疗疾病的巨环 |
-
2020
- 2020-12-02 CN CN202080092056.8A patent/CN114929710B/zh active Active
- 2020-12-02 TW TW109142431A patent/TW202134249A/zh unknown
- 2020-12-02 US US17/110,051 patent/US11634433B2/en active Active
- 2020-12-02 PE PE2022001016A patent/PE20221485A1/es unknown
- 2020-12-02 EP EP20897539.1A patent/EP4069700A4/en active Pending
- 2020-12-02 IL IL293458A patent/IL293458A/en unknown
- 2020-12-02 CA CA3163735A patent/CA3163735A1/en active Pending
- 2020-12-02 MX MX2022006853A patent/MX2022006853A/es unknown
- 2020-12-02 BR BR112022010702A patent/BR112022010702A2/pt unknown
- 2020-12-02 AU AU2020395136A patent/AU2020395136A1/en active Pending
- 2020-12-02 JP JP2022533150A patent/JP2023504523A/ja active Pending
- 2020-12-02 KR KR1020227022836A patent/KR20220133869A/ko unknown
- 2020-12-02 WO PCT/US2020/062859 patent/WO2021113339A1/en active Application Filing
-
2021
- 2021-03-26 US US17/214,096 patent/US11142533B2/en active Active
-
2022
- 2022-06-24 CO CONC2022/0008817A patent/CO2022008817A2/es unknown
-
2023
- 2023-03-17 US US18/123,080 patent/US20230322806A1/en active Pending
Also Published As
Publication number | Publication date |
---|---|
PE20221485A1 (es) | 2022-09-26 |
US11142533B2 (en) | 2021-10-12 |
AU2020395136A1 (en) | 2022-07-07 |
US20230322806A1 (en) | 2023-10-12 |
US11634433B2 (en) | 2023-04-25 |
CO2022008817A2 (es) | 2022-09-20 |
TW202134249A (zh) | 2021-09-16 |
CA3163735A1 (en) | 2021-06-10 |
MX2022006853A (es) | 2022-09-19 |
IL293458A (en) | 2022-07-01 |
WO2021113339A1 (en) | 2021-06-10 |
JP2023504523A (ja) | 2023-02-03 |
CN114929710B (zh) | 2024-03-29 |
CN114929710A (zh) | 2022-08-19 |
KR20220133869A (ko) | 2022-10-05 |
US20210163499A1 (en) | 2021-06-03 |
EP4069700A4 (en) | 2023-05-17 |
US20210246145A1 (en) | 2021-08-12 |
EP4069700A1 (en) | 2022-10-12 |
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