BR112022008892A2 - Processo e intermediário para a preparação de oxetan-2-ilmetanamina - Google Patents
Processo e intermediário para a preparação de oxetan-2-ilmetanaminaInfo
- Publication number
- BR112022008892A2 BR112022008892A2 BR112022008892A BR112022008892A BR112022008892A2 BR 112022008892 A2 BR112022008892 A2 BR 112022008892A2 BR 112022008892 A BR112022008892 A BR 112022008892A BR 112022008892 A BR112022008892 A BR 112022008892A BR 112022008892 A2 BR112022008892 A2 BR 112022008892A2
- Authority
- BR
- Brazil
- Prior art keywords
- preparation
- ilmethanamine
- oxetan
- salt
- compound
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
- C07D305/02—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms not condensed with other rings
- C07D305/04—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C07D305/06—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Epoxy Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
A presente invenção refere-se a um processo e intermediário para a preparação de um composto de fórmula (I), ou seu sal. (I)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201962946146P | 2019-12-10 | 2019-12-10 | |
PCT/US2020/063546 WO2021118906A1 (en) | 2019-12-10 | 2020-12-07 | Process and intermediate for the preparation of oxetan-2-ylmethanamine |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112022008892A2 true BR112022008892A2 (pt) | 2022-08-23 |
Family
ID=74003942
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112022008892A BR112022008892A2 (pt) | 2019-12-10 | 2020-12-07 | Processo e intermediário para a preparação de oxetan-2-ilmetanamina |
Country Status (25)
Country | Link |
---|---|
US (1) | US20230013840A1 (pt) |
EP (1) | EP4073051B1 (pt) |
JP (1) | JP7292517B2 (pt) |
KR (1) | KR102635237B1 (pt) |
CN (1) | CN114728923A (pt) |
AU (1) | AU2020401539B2 (pt) |
BR (1) | BR112022008892A2 (pt) |
CA (1) | CA3160419A1 (pt) |
CL (1) | CL2022001511A1 (pt) |
CO (1) | CO2022008127A2 (pt) |
DK (1) | DK4073051T3 (pt) |
EC (1) | ECSP22046595A (pt) |
FI (1) | FI4073051T3 (pt) |
HR (1) | HRP20240343T1 (pt) |
IL (1) | IL292707A (pt) |
LT (1) | LT4073051T (pt) |
MA (1) | MA58104B1 (pt) |
MX (1) | MX2022006984A (pt) |
PE (1) | PE20230183A1 (pt) |
PL (1) | PL4073051T3 (pt) |
PT (1) | PT4073051T (pt) |
RS (1) | RS65238B1 (pt) |
SI (1) | SI4073051T1 (pt) |
UA (1) | UA127884C2 (pt) |
WO (1) | WO2021118906A1 (pt) |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7208140B2 (en) | 2003-02-19 | 2007-04-24 | Schering Aktiengesellschaft | Trimeric macrocyclic substituted benzene derivatives |
UA114601C2 (uk) | 2011-05-06 | 2017-07-10 | Егіш Дьйодьсердьяр Нільваношан Мюкеде Ресвеньтаршашаг | Спосіб одержання ривароксабану та проміжних сполук, які одержано в даному способі |
WO2013169531A1 (en) * | 2012-05-09 | 2013-11-14 | Boehringer Ingelheim International Gmbh | Methods for making oxetan-3-ylmethanamines |
PE20191501A1 (es) * | 2016-12-16 | 2019-10-22 | Pfizer | Agonistas receptores de glp-1 y sus usos de los mismos |
CN109265389B (zh) * | 2018-08-31 | 2020-08-18 | 南京富润凯德生物医药有限公司 | 2-(氨基甲基)-1-氧杂-7-氮杂螺[3.5]壬烷衍生物、中间体及其制备方法 |
-
2020
- 2020-12-07 MX MX2022006984A patent/MX2022006984A/es unknown
- 2020-12-07 FI FIEP20829133.6T patent/FI4073051T3/fi active
- 2020-12-07 WO PCT/US2020/063546 patent/WO2021118906A1/en active Application Filing
- 2020-12-07 PT PT208291336T patent/PT4073051T/pt unknown
- 2020-12-07 LT LTEPPCT/US2020/063546T patent/LT4073051T/lt unknown
- 2020-12-07 CN CN202080082957.9A patent/CN114728923A/zh active Pending
- 2020-12-07 CA CA3160419A patent/CA3160419A1/en active Pending
- 2020-12-07 RS RS20240243A patent/RS65238B1/sr unknown
- 2020-12-07 HR HRP20240343TT patent/HRP20240343T1/hr unknown
- 2020-12-07 BR BR112022008892A patent/BR112022008892A2/pt unknown
- 2020-12-07 UA UAA202201389A patent/UA127884C2/uk unknown
- 2020-12-07 PL PL20829133.6T patent/PL4073051T3/pl unknown
- 2020-12-07 SI SI202030381T patent/SI4073051T1/sl unknown
- 2020-12-07 IL IL292707A patent/IL292707A/en unknown
- 2020-12-07 AU AU2020401539A patent/AU2020401539B2/en active Active
- 2020-12-07 JP JP2022534655A patent/JP7292517B2/ja active Active
- 2020-12-07 MA MA58104A patent/MA58104B1/fr unknown
- 2020-12-07 DK DK20829133.6T patent/DK4073051T3/da active
- 2020-12-07 PE PE2022001046A patent/PE20230183A1/es unknown
- 2020-12-07 US US17/779,447 patent/US20230013840A1/en active Pending
- 2020-12-07 EP EP20829133.6A patent/EP4073051B1/en active Active
- 2020-12-07 KR KR1020227018626A patent/KR102635237B1/ko active IP Right Grant
-
2022
- 2022-06-08 CL CL2022001511A patent/CL2022001511A1/es unknown
- 2022-06-08 CO CONC2022/0008127A patent/CO2022008127A2/es unknown
- 2022-06-10 EC ECSENADI202246595A patent/ECSP22046595A/es unknown
Also Published As
Publication number | Publication date |
---|---|
UA127884C2 (uk) | 2024-01-31 |
CL2022001511A1 (es) | 2023-01-20 |
PT4073051T (pt) | 2024-02-21 |
AU2020401539A1 (en) | 2022-06-16 |
AU2020401539B2 (en) | 2023-06-01 |
HRP20240343T1 (hr) | 2024-05-24 |
EP4073051A1 (en) | 2022-10-19 |
KR20220097941A (ko) | 2022-07-08 |
PL4073051T3 (pl) | 2024-05-20 |
KR102635237B1 (ko) | 2024-02-13 |
PE20230183A1 (es) | 2023-02-01 |
ECSP22046595A (es) | 2022-07-29 |
CO2022008127A2 (es) | 2022-06-10 |
MA58104B1 (fr) | 2024-05-31 |
JP2023504581A (ja) | 2023-02-03 |
IL292707A (en) | 2022-07-01 |
MX2022006984A (es) | 2022-07-13 |
CA3160419A1 (en) | 2021-06-17 |
CN114728923A (zh) | 2022-07-08 |
WO2021118906A1 (en) | 2021-06-17 |
SI4073051T1 (sl) | 2024-04-30 |
RS65238B1 (sr) | 2024-03-29 |
JP7292517B2 (ja) | 2023-06-16 |
US20230013840A1 (en) | 2023-01-19 |
EP4073051B1 (en) | 2024-02-07 |
FI4073051T3 (fi) | 2024-03-28 |
LT4073051T (lt) | 2024-03-12 |
DK4073051T3 (da) | 2024-02-26 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
BR112022012585A2 (pt) | Inibidores de formas mutantes de egfr | |
BR112018002499A2 (pt) | método de preparação de um composto da fórmula (a) ou um seu sal, solvato ou conjugado de aminoácido farmaceuticamente aceitável, composto produzido pelo método e composição farmacêutica | |
BR112018007381A2 (pt) | compostos úteis como imunomoduladores | |
BR112017006253A2 (pt) | novos compostos | |
EA201890308A1 (ru) | Замещенные азасоединения как ингибиторы irak-4 | |
EA201890899A1 (ru) | Модуляторы фарнезоидного x-рецептора | |
BR112017006116A2 (pt) | processos de preparação de compostos e compostos | |
BR112017002403A2 (pt) | formas de cristais de inibidores de glutaminase | |
EA201891666A1 (ru) | Арилзамещенные пиримидины для применения при инфекции, вызванной вирусом гриппа | |
BR112018014712A2 (pt) | processo melhorado para a preparação de osimertinib (azd9291) ou um sal do mesmo e | |
BR112023002939A2 (pt) | Processo e intermediários para preparar um inibidor de jak1 | |
BR112017019850A2 (pt) | ?processo melhorado para a preparação de apremilast? | |
BR112022008183A2 (pt) | Formas de sal de um receptor de c5a de componente do complemento | |
BR112018012325A2 (pt) | métodos para a preparação de 5,6-di-hidro-6-fenilbenzo[f]isoquinolin-2-amina substituída | |
BR112018070345A2 (pt) | processo para a preparação de derivados de 4-aminoindano e amidas de aminoindano relacionadas | |
CO2021009309A2 (es) | Formas de sal y cristalinas de un compuesto orgánico y composiciones farmacéuticas del mismo | |
MX2020004842A (es) | Compuestos heterociclicos antiinfecciosos y sus usos. | |
BR112021026618A2 (pt) | Composto de pirazolpirimidina, método de preparação do mesmo e aplicações do mesmo | |
BR112019000988A2 (pt) | derivado de triazolopirazinona útil como inibidor de pde1 humana | |
BR112022009493A2 (pt) | Fabricação de do3a protegido | |
BR112018009754A2 (pt) | bloqueador de canal de sódio | |
BR112023023729A2 (pt) | Novo intermediário para preparação de piroxasulfona | |
BR112022008892A2 (pt) | Processo e intermediário para a preparação de oxetan-2-ilmetanamina | |
BR112017017209A2 (pt) | processo para inibir incrustação. | |
BR112015031945A2 (pt) | processos para a preparação de compostos |