BR112022008892A2 - Processo e intermediário para a preparação de oxetan-2-ilmetanamina - Google Patents

Processo e intermediário para a preparação de oxetan-2-ilmetanamina

Info

Publication number
BR112022008892A2
BR112022008892A2 BR112022008892A BR112022008892A BR112022008892A2 BR 112022008892 A2 BR112022008892 A2 BR 112022008892A2 BR 112022008892 A BR112022008892 A BR 112022008892A BR 112022008892 A BR112022008892 A BR 112022008892A BR 112022008892 A2 BR112022008892 A2 BR 112022008892A2
Authority
BR
Brazil
Prior art keywords
preparation
ilmethanamine
oxetan
salt
compound
Prior art date
Application number
BR112022008892A
Other languages
English (en)
Inventor
Paul Cole Kevin
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of BR112022008892A2 publication Critical patent/BR112022008892A2/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D305/00Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/02Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D305/04Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D305/06Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Epoxy Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

A presente invenção refere-se a um processo e intermediário para a preparação de um composto de fórmula (I), ou seu sal. (I)
BR112022008892A 2019-12-10 2020-12-07 Processo e intermediário para a preparação de oxetan-2-ilmetanamina BR112022008892A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201962946146P 2019-12-10 2019-12-10
PCT/US2020/063546 WO2021118906A1 (en) 2019-12-10 2020-12-07 Process and intermediate for the preparation of oxetan-2-ylmethanamine

Publications (1)

Publication Number Publication Date
BR112022008892A2 true BR112022008892A2 (pt) 2022-08-23

Family

ID=74003942

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112022008892A BR112022008892A2 (pt) 2019-12-10 2020-12-07 Processo e intermediário para a preparação de oxetan-2-ilmetanamina

Country Status (25)

Country Link
US (1) US20230013840A1 (pt)
EP (1) EP4073051B1 (pt)
JP (1) JP7292517B2 (pt)
KR (1) KR102635237B1 (pt)
CN (1) CN114728923A (pt)
AU (1) AU2020401539B2 (pt)
BR (1) BR112022008892A2 (pt)
CA (1) CA3160419A1 (pt)
CL (1) CL2022001511A1 (pt)
CO (1) CO2022008127A2 (pt)
DK (1) DK4073051T3 (pt)
EC (1) ECSP22046595A (pt)
FI (1) FI4073051T3 (pt)
HR (1) HRP20240343T1 (pt)
IL (1) IL292707A (pt)
LT (1) LT4073051T (pt)
MA (1) MA58104B1 (pt)
MX (1) MX2022006984A (pt)
PE (1) PE20230183A1 (pt)
PL (1) PL4073051T3 (pt)
PT (1) PT4073051T (pt)
RS (1) RS65238B1 (pt)
SI (1) SI4073051T1 (pt)
UA (1) UA127884C2 (pt)
WO (1) WO2021118906A1 (pt)

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7208140B2 (en) 2003-02-19 2007-04-24 Schering Aktiengesellschaft Trimeric macrocyclic substituted benzene derivatives
UA114601C2 (uk) 2011-05-06 2017-07-10 Егіш Дьйодьсердьяр Нільваношан Мюкеде Ресвеньтаршашаг Спосіб одержання ривароксабану та проміжних сполук, які одержано в даному способі
WO2013169531A1 (en) * 2012-05-09 2013-11-14 Boehringer Ingelheim International Gmbh Methods for making oxetan-3-ylmethanamines
PE20191501A1 (es) * 2016-12-16 2019-10-22 Pfizer Agonistas receptores de glp-1 y sus usos de los mismos
CN109265389B (zh) * 2018-08-31 2020-08-18 南京富润凯德生物医药有限公司 2-(氨基甲基)-1-氧杂-7-氮杂螺[3.5]壬烷衍生物、中间体及其制备方法

Also Published As

Publication number Publication date
UA127884C2 (uk) 2024-01-31
CL2022001511A1 (es) 2023-01-20
PT4073051T (pt) 2024-02-21
AU2020401539A1 (en) 2022-06-16
AU2020401539B2 (en) 2023-06-01
HRP20240343T1 (hr) 2024-05-24
EP4073051A1 (en) 2022-10-19
KR20220097941A (ko) 2022-07-08
PL4073051T3 (pl) 2024-05-20
KR102635237B1 (ko) 2024-02-13
PE20230183A1 (es) 2023-02-01
ECSP22046595A (es) 2022-07-29
CO2022008127A2 (es) 2022-06-10
MA58104B1 (fr) 2024-05-31
JP2023504581A (ja) 2023-02-03
IL292707A (en) 2022-07-01
MX2022006984A (es) 2022-07-13
CA3160419A1 (en) 2021-06-17
CN114728923A (zh) 2022-07-08
WO2021118906A1 (en) 2021-06-17
SI4073051T1 (sl) 2024-04-30
RS65238B1 (sr) 2024-03-29
JP7292517B2 (ja) 2023-06-16
US20230013840A1 (en) 2023-01-19
EP4073051B1 (en) 2024-02-07
FI4073051T3 (fi) 2024-03-28
LT4073051T (lt) 2024-03-12
DK4073051T3 (da) 2024-02-26

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