BR112021019999A2 - Formulação de comprimido vaginal - Google Patents

Formulação de comprimido vaginal

Info

Publication number
BR112021019999A2
BR112021019999A2 BR112021019999A BR112021019999A BR112021019999A2 BR 112021019999 A2 BR112021019999 A2 BR 112021019999A2 BR 112021019999 A BR112021019999 A BR 112021019999A BR 112021019999 A BR112021019999 A BR 112021019999A BR 112021019999 A2 BR112021019999 A2 BR 112021019999A2
Authority
BR
Brazil
Prior art keywords
tablet formulation
vaginal tablet
vaginal
glucone
lactone
Prior art date
Application number
BR112021019999A
Other languages
English (en)
Inventor
Annette Säfholm
Helena Strevens
Nils-Olof Lindberg
Olov Sterner
Sophie Manner
Ulf Ellervik
Original Assignee
Gedea Biotech Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gedea Biotech Ab filed Critical Gedea Biotech Ab
Publication of BR112021019999A2 publication Critical patent/BR112021019999A2/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/365Lactones
    • A61K31/366Lactones having six-membered rings, e.g. delta-lactones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/365Lactones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0034Urogenital system, e.g. vagina, uterus, cervix, penis, scrotum, urethra, bladder; Personal lubricants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/02Drugs for genital or sexual disorders; Contraceptives for disorders of the vagina

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Reproductive Health (AREA)
  • Gynecology & Obstetrics (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)

Abstract

formulação de comprimido vaginal. a presente invenção se refere a uma composição farmacêutica que compreende glucona-d-lactona, que é adequado para uso no tratamento de infecções microbianas vaginais.
BR112021019999A 2019-04-05 2020-04-03 Formulação de comprimido vaginal BR112021019999A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP19167495 2019-04-05
PCT/EP2020/059582 WO2020201515A1 (en) 2019-04-05 2020-04-03 Vaginal tablet formulation

Publications (1)

Publication Number Publication Date
BR112021019999A2 true BR112021019999A2 (pt) 2021-12-07

Family

ID=66101895

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112021019999A BR112021019999A2 (pt) 2019-04-05 2020-04-03 Formulação de comprimido vaginal

Country Status (24)

Country Link
US (1) US20220193031A1 (pt)
EP (1) EP3976000B1 (pt)
JP (1) JP2022537478A (pt)
KR (1) KR20210148195A (pt)
CN (1) CN113660928B (pt)
AR (1) AR118580A1 (pt)
AU (1) AU2020252268A1 (pt)
BR (1) BR112021019999A2 (pt)
CA (1) CA3134086A1 (pt)
CL (1) CL2021002430A1 (pt)
CO (1) CO2021014253A2 (pt)
EA (1) EA202192716A1 (pt)
ES (1) ES2961736T3 (pt)
HU (1) HUE062772T2 (pt)
IL (1) IL286942A (pt)
MA (1) MA56011A (pt)
MX (1) MX2021012146A (pt)
PE (1) PE20220381A1 (pt)
PL (1) PL3976000T3 (pt)
SG (1) SG11202110236QA (pt)
TW (1) TW202103693A (pt)
UA (1) UA127823C2 (pt)
WO (1) WO2020201515A1 (pt)
ZA (1) ZA202106877B (pt)

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2165139T3 (es) * 1998-04-30 2002-03-01 Vesely Renata Maria Cavaliere Composiciones farmaceuticas que contienen lactobacillus brevis y lactobacillus salivarius para el tratamiento de infecciones vaginales.
US6287599B1 (en) * 2000-12-20 2001-09-11 Shire Laboratories, Inc. Sustained release pharmaceutical dosage forms with minimized pH dependent dissolution profiles
US20030017207A1 (en) * 2001-05-01 2003-01-23 Lin Shun Y. Compositions and methods for treating vulvovaginitis and vaginosis
ITBO20110461A1 (it) * 2011-07-29 2013-01-30 Alfa Wassermann Spa Composizioni farmaceutiche comprendenti rifaximina, processi per la loro preparazione e loro uso nel trattamento di infezioni vaginali.
MY198473A (en) 2016-04-06 2023-08-31 Gedea Biotech Ab Glucono delta-lactone for treatment of vaginal fungal infections
EP3691625A1 (en) 2017-10-06 2020-08-12 Gedea Biotech AB Gluconic acid derivatives for use in the treatment and/or prevention of microbial infections

Also Published As

Publication number Publication date
AR118580A1 (es) 2021-10-20
ES2961736T3 (es) 2024-03-13
PL3976000T3 (pl) 2023-12-04
KR20210148195A (ko) 2021-12-07
EP3976000C0 (en) 2023-08-02
EP3976000B1 (en) 2023-08-02
CA3134086A1 (en) 2020-10-08
JP2022537478A (ja) 2022-08-26
CL2021002430A1 (es) 2022-07-01
EA202192716A1 (ru) 2022-01-17
TW202103693A (zh) 2021-02-01
UA127823C2 (uk) 2024-01-10
PE20220381A1 (es) 2022-03-18
WO2020201515A1 (en) 2020-10-08
CO2021014253A2 (es) 2021-11-19
US20220193031A1 (en) 2022-06-23
IL286942A (en) 2021-12-01
CN113660928B (zh) 2024-04-05
MA56011A (fr) 2022-04-06
MX2021012146A (es) 2021-12-10
EP3976000A1 (en) 2022-04-06
ZA202106877B (en) 2023-03-29
SG11202110236QA (en) 2021-10-28
CN113660928A (zh) 2021-11-16
HUE062772T2 (hu) 2023-12-28
AU2020252268A1 (en) 2021-10-21

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