BR112019004946A2 - método para produzir compostos bicíclicos halogenados - Google Patents

método para produzir compostos bicíclicos halogenados

Info

Publication number
BR112019004946A2
BR112019004946A2 BR112019004946A BR112019004946A BR112019004946A2 BR 112019004946 A2 BR112019004946 A2 BR 112019004946A2 BR 112019004946 A BR112019004946 A BR 112019004946A BR 112019004946 A BR112019004946 A BR 112019004946A BR 112019004946 A2 BR112019004946 A2 BR 112019004946A2
Authority
BR
Brazil
Prior art keywords
bicyclic compounds
producing halogenated
halogenated bicyclic
halogen
formula
Prior art date
Application number
BR112019004946A
Other languages
English (en)
Other versions
BR112019004946B1 (pt
Inventor
Wilcke David
Hager Dominik
Hoffmeister Laura
Mosrin Marc
Willot Matthieu
Kausch-Busies Nina
Fischer Rüdiger
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of BR112019004946A2 publication Critical patent/BR112019004946A2/pt
Publication of BR112019004946B1 publication Critical patent/BR112019004946B1/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F3/00—Compounds containing elements of Groups 2 or 12 of the Periodic Table
    • C07F3/06—Zinc compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

a presente invenção se refere a um processo para preparar sistemas bicíclicos halogenados da fórmula (ii) procedendo a partir dos compostos da estrutura q-h através de intermediários da fórmula (iiia) ou (iiib) em que q é um elemento estrutural em que o símbolo # indica a ligação ao resto da molécula e a, q1, q2, q3, q4, q5 e q6 têm as definições dadas na descrição, hal é halogênio, e r2 é halogênio ou -o-pivaloíla.
BR112019004946-0A 2016-09-14 2017-09-06 Processo para produção de compostos bicíclicos halogenados, e seus intermediários BR112019004946B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP16188760 2016-09-14
EP16188760.9 2016-09-14
PCT/EP2017/072363 WO2018050515A1 (de) 2016-09-14 2017-09-06 Verfahren zur herstellung von halogenierten bizyklen

Publications (2)

Publication Number Publication Date
BR112019004946A2 true BR112019004946A2 (pt) 2019-06-25
BR112019004946B1 BR112019004946B1 (pt) 2023-01-10

Family

ID=56943355

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112019004946-0A BR112019004946B1 (pt) 2016-09-14 2017-09-06 Processo para produção de compostos bicíclicos halogenados, e seus intermediários

Country Status (12)

Country Link
US (1) US20190375766A1 (pt)
EP (1) EP3512847B1 (pt)
JP (1) JP7066683B2 (pt)
KR (1) KR102471278B1 (pt)
CN (1) CN109715627A (pt)
BR (1) BR112019004946B1 (pt)
DK (1) DK3512847T3 (pt)
ES (1) ES2919558T3 (pt)
IL (1) IL265257B (pt)
MX (1) MX2019002937A (pt)
TW (1) TWI749060B (pt)
WO (1) WO2018050515A1 (pt)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR102420235B1 (ko) * 2016-08-16 2022-07-12 바이엘 크롭사이언스 악티엔게젤샤프트 3H-이미다졸[4,5-c]피리딘 유도체와 유기금속 아연-아민 염기의 반응에 의한 2-(3,6-디할로피리딘-2-일)-3H-이미다졸[4,5-c]피리딘 유도체 및 관련 화합물의 제조 방법
TWI820231B (zh) * 2018-10-11 2023-11-01 德商拜耳廠股份有限公司 用於製備經取代咪唑衍生物之方法

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4472409A (en) * 1981-11-05 1984-09-18 Byk Gulden Lomberg Chemische Fabrik Gesellschaft Mit Beschrankter Haftung 2-Pyridylmethyl thio(sulfinyl)benzimidazoles with gastric acid secretion inhibiting effects
JPS5910590A (ja) * 1982-07-08 1984-01-20 Ishihara Sangyo Kaisha Ltd 置換酢酸アニリド系化合物およびそれらを含有する除草剤
JPS61106563A (ja) * 1984-10-30 1986-05-24 Oouchi Shinko Kagaku Kogyo Kk ２−クロルベンゾチアゾ−ル誘導体の製造方法
GB0027561D0 (en) 2000-11-10 2000-12-27 Merck Sharp & Dohme Therapeutic agents
EP1879896A1 (en) 2005-04-05 2008-01-23 Eli Lilly And Company Imidazopyridazine compounds
US9108959B2 (en) 2011-03-03 2015-08-18 Merck Sharp & Dohme Corp. Process for the preparation of an orexin receptor antagonist
BR112014029501B1 (pt) * 2012-05-31 2020-05-19 Sumitomo Chemical Co composto heterocíclico fundido, seu uso, agente de controle de pragas e método para o controle de pragas
US20150289512A1 (en) 2012-11-09 2015-10-15 Sumitomo Chemical Company, Limited Method for promoting plant growth
US8846657B2 (en) 2012-12-20 2014-09-30 Merck Sharp & Dohme Corp. Substituted imidazopyridines as HDM2 inhibitors
AU2014296184B2 (en) 2013-07-31 2017-04-27 Gilead Sciences, Inc. Syk inhibitors
KR101698640B1 (ko) * 2013-09-26 2017-01-20 주식회사 엘지화학 헤테로환 화합물 및 이를 포함하는 유기 발광 소자
AU2014348191B2 (en) * 2013-11-18 2019-03-28 Forma Therapeutics Inc. Tetrahydroquinoline compositions as BET bromodomain inhibitors

Also Published As

Publication number Publication date
IL265257A (en) 2019-05-30
CN109715627A (zh) 2019-05-03
MX2019002937A (es) 2019-06-06
TW201825485A (zh) 2018-07-16
JP7066683B2 (ja) 2022-05-13
IL265257B (en) 2021-12-01
EP3512847A1 (de) 2019-07-24
TWI749060B (zh) 2021-12-11
WO2018050515A1 (de) 2018-03-22
BR112019004946B1 (pt) 2023-01-10
KR20190045332A (ko) 2019-05-02
JP2019529405A (ja) 2019-10-17
ES2919558T3 (es) 2022-07-27
KR102471278B1 (ko) 2022-11-25
US20190375766A1 (en) 2019-12-12
EP3512847B1 (de) 2022-03-30
DK3512847T3 (da) 2022-06-27

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Legal Events

Date Code Title Description
B350 Update of information on the portal [chapter 15.35 patent gazette]
B06W Patent application suspended after preliminary examination (for patents with searches from other patent authorities) chapter 6.23 patent gazette]
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

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