BR112018004310A2 - derivados de espinosina e método de preparação - Google Patents
derivados de espinosina e método de preparaçãoInfo
- Publication number
- BR112018004310A2 BR112018004310A2 BR112018004310A BR112018004310A BR112018004310A2 BR 112018004310 A2 BR112018004310 A2 BR 112018004310A2 BR 112018004310 A BR112018004310 A BR 112018004310A BR 112018004310 A BR112018004310 A BR 112018004310A BR 112018004310 A2 BR112018004310 A2 BR 112018004310A2
- Authority
- BR
- Brazil
- Prior art keywords
- preparation
- spinosine
- derivatives
- spinosine derivatives
- arachnid
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/02—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms
- A01N43/04—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom
- A01N43/22—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom rings with more than six members
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N45/00—Biocides, pest repellants or attractants, or plant growth regulators, containing compounds having three or more carbocyclic rings condensed among themselves, at least one ring not being a six-membered ring
- A01N45/02—Biocides, pest repellants or attractants, or plant growth regulators, containing compounds having three or more carbocyclic rings condensed among themselves, at least one ring not being a six-membered ring having three carbocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D313/00—Heterocyclic compounds containing rings of more than six members having one oxygen atom as the only ring hetero atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H1/00—Processes for the preparation of sugar derivatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N2300/00—Combinations or mixtures of active ingredients covered by classes A01N27/00 - A01N65/48 with other active or formulation relevant ingredients, e.g. specific carrier materials or surfactants, covered by classes A01N25/00 - A01N65/48
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biotechnology (AREA)
- Biochemistry (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Environmental Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Zoology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Dermatology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Saccharide Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Compositions Of Macromolecular Compounds (AREA)
- Medicinal Preparation (AREA)
Abstract
são fornecidas composições e métodos para a produção de derivados de espinosina. o método produz derivados de espinosina que exibem atividade em relação a insetos, aracnídeos e nematoides e que são úteis nos mercados da agricultura e da saúde animal.
Applications Claiming Priority (6)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201562214083P | 2015-09-03 | 2015-09-03 | |
US201662290676P | 2016-02-03 | 2016-02-03 | |
US201662303015P | 2016-03-03 | 2016-03-03 | |
US201662303078P | 2016-03-03 | 2016-03-03 | |
US201662380664P | 2016-08-29 | 2016-08-29 | |
PCT/US2016/049879 WO2017040769A1 (en) | 2015-09-03 | 2016-09-01 | Spinosyn derivatives as insecticides |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112018004310A2 true BR112018004310A2 (pt) | 2018-10-09 |
Family
ID=56940400
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112018004313A BR112018004313A2 (pt) | 2015-09-03 | 2016-09-01 | derivados de espinosina |
BR112018004310A BR112018004310A2 (pt) | 2015-09-03 | 2016-09-01 | derivados de espinosina e método de preparação |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112018004313A BR112018004313A2 (pt) | 2015-09-03 | 2016-09-01 | derivados de espinosina |
Country Status (12)
Country | Link |
---|---|
US (3) | US10570166B2 (pt) |
EP (3) | EP3344612B1 (pt) |
JP (3) | JP2018531912A (pt) |
KR (3) | KR20180048871A (pt) |
CN (3) | CN108026063A (pt) |
AU (3) | AU2016317854A1 (pt) |
BR (2) | BR112018004313A2 (pt) |
CA (3) | CA2997499A1 (pt) |
CL (2) | CL2018000525A1 (pt) |
IL (2) | IL257759A (pt) |
MX (3) | MX2018002540A (pt) |
WO (4) | WO2017040769A1 (pt) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2018531912A (ja) | 2015-09-03 | 2018-11-01 | アグリメティス,エルエルシー | 殺虫剤としてのスピノシン誘導体 |
WO2018132288A1 (en) * | 2017-01-13 | 2018-07-19 | Agrimetis, Llc | Aziridine spinosyn derivatives and methods of making |
BR112020012018A2 (pt) * | 2017-12-15 | 2020-11-24 | Tarsus Pharmaceuticals, Inc. | formulações de parasiticida de isoxazolina e métodos para tratar blefarite |
AR116524A1 (es) * | 2018-10-04 | 2021-05-19 | Elanco Tiergesundheit Ag | Potenciación de tratamiento de helmintos |
EP4079744A1 (en) | 2021-04-23 | 2022-10-26 | Acies Bio d.o.o. | Novel spinosyn prodrugs |
AR125402A1 (es) | 2021-04-23 | 2023-07-12 | Acies Bio D O O | Profármacos nuevos de espinosinas |
EP4101858A1 (en) | 2021-06-08 | 2022-12-14 | Acies Bio d.o.o. | Novel spinosyn compounds |
Family Cites Families (30)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE1049845B (de) | 1957-01-04 | 1959-02-05 | Consortium Elektrochem Ind | Verfahren zur Herstellung von Carbonylverbindungen |
US5362634A (en) | 1989-10-30 | 1994-11-08 | Dowelanco | Process for producing A83543 compounds |
US5728554A (en) | 1995-04-11 | 1998-03-17 | Cytel Corporation | Enzymatic synthesis of glycosidic linkages |
US6030815A (en) | 1995-04-11 | 2000-02-29 | Neose Technologies, Inc. | Enzymatic synthesis of oligosaccharides |
US5922577A (en) | 1995-04-11 | 1999-07-13 | Cytel Corporation | Enzymatic synthesis of glycosidic linkages |
US5876980A (en) | 1995-04-11 | 1999-03-02 | Cytel Corporation | Enzymatic synthesis of oligosaccharides |
CN1130369C (zh) * | 1995-06-14 | 2003-12-10 | 道农业科学公司 | 对刺糖多孢菌素化合物的合成修饰 |
US6001981A (en) * | 1996-06-13 | 1999-12-14 | Dow Agrosciences Llc | Synthetic modification of Spinosyn compounds |
US6143526A (en) | 1998-03-09 | 2000-11-07 | Baltz; Richard H. | Biosynthetic genes for spinosyn insecticide production |
WO2000001347A2 (en) | 1998-07-02 | 2000-01-13 | Eli Lilly And Company | Formulations for controlling human lice |
AU770879B2 (en) | 1999-08-12 | 2004-03-04 | Eli Lilly And Company | Ectoparasiticidal aqueous suspension formulations of spinosyns |
US6927210B1 (en) | 1999-08-12 | 2005-08-09 | Eli Lilly And Company | Ectoparasiticidal aqueous suspension formulations of spinosyns |
TWI275592B (en) * | 2001-03-21 | 2007-03-11 | Dow Agrosciences Llc | Synthetic derivatives of 21-butenyl and related spinosyns |
US6919464B1 (en) | 2001-03-21 | 2005-07-19 | Dow Agrosciences Llc | Synthetic derivatives of 21-butenyl and related spinosyns |
US20030225006A1 (en) * | 2002-02-19 | 2003-12-04 | Burns Lesley S | Novel spinosyn-producing polyketide synthases |
MXPA05010773A (es) | 2003-04-09 | 2005-12-12 | Neose Technologies Inc | Metodos de glicopegilacion y proteinas/peptidos producidos por los metodos. |
PL1744763T3 (pl) | 2004-04-29 | 2010-06-30 | Elanco Us Inc | Spinozyny do gojenia ran |
US8470381B2 (en) | 2008-09-22 | 2013-06-25 | Christine Kritikou | Spinosyn antifouling compositions, methods of use thereof and articles protected from attachment of biofouling organisms |
WO2010150100A1 (en) | 2009-06-24 | 2010-12-29 | Entarco Sa | The use of spinosyns and spinosyn compositions against diseases caused by protozoans, viral infections and cancer |
WO2011091122A1 (en) | 2010-01-25 | 2011-07-28 | Eli Lilly And Company | Methods for internally controlling or treating equine bot larvae |
AU2011323082B2 (en) | 2010-11-05 | 2015-06-11 | Eli Lilly And Company | Methods for inhibiting insect infestations |
EP2654757A1 (en) | 2010-12-22 | 2013-10-30 | Entarco SA | The use of spinosyns and spinosyn compositions as local anesthetics and as antiarrhythmic agents |
WO2012141754A2 (en) | 2010-12-29 | 2012-10-18 | Dow Agrosciences Llc | Methods of controlling insects |
US9631195B2 (en) | 2011-12-28 | 2017-04-25 | Dow Agrosciences Llc | Identification and characterization of the spinactin biosysnthesis gene cluster from spinosyn producing saccharopolyspora spinosa |
US9895388B1 (en) * | 2012-07-27 | 2018-02-20 | ParaPRO | Methods and compositions useful for controlling cutaneous mites |
CN102977166B (zh) * | 2012-12-05 | 2015-07-29 | 湖南化工研究院 | 13-硫醚取代多杀菌素衍生物及其制备方法 |
CA2896790C (en) * | 2013-01-22 | 2022-05-10 | Actelion Pharmaceuticals Ltd | Heterocyclic amide derivatives as p2x7 receptor antagonists |
EP3060054A4 (en) | 2013-10-22 | 2017-04-05 | Dow AgroSciences LLC | Synergistic pesticidal compositions and related methods |
US9873639B1 (en) | 2015-07-17 | 2018-01-23 | Joe Doccola | Agricultural biomass as a matrix for release of plant active compounds |
JP2018531912A (ja) | 2015-09-03 | 2018-11-01 | アグリメティス,エルエルシー | 殺虫剤としてのスピノシン誘導体 |
-
2016
- 2016-09-01 JP JP2018512332A patent/JP2018531912A/ja not_active Withdrawn
- 2016-09-01 WO PCT/US2016/049879 patent/WO2017040769A1/en active Application Filing
- 2016-09-01 CN CN201680056085.2A patent/CN108026063A/zh active Pending
- 2016-09-01 KR KR1020187008942A patent/KR20180048871A/ko unknown
- 2016-09-01 WO PCT/US2016/049870 patent/WO2017040763A1/en active Application Filing
- 2016-09-01 BR BR112018004313A patent/BR112018004313A2/pt not_active Application Discontinuation
- 2016-09-01 MX MX2018002540A patent/MX2018002540A/es unknown
- 2016-09-01 JP JP2018512331A patent/JP2018532708A/ja not_active Withdrawn
- 2016-09-01 EP EP16767424.1A patent/EP3344612B1/en active Active
- 2016-09-01 AU AU2016317854A patent/AU2016317854A1/en not_active Abandoned
- 2016-09-01 MX MX2018002538A patent/MX2018002538A/es unknown
- 2016-09-01 KR KR1020187008943A patent/KR20180050340A/ko unknown
- 2016-09-01 BR BR112018004310A patent/BR112018004310A2/pt not_active Application Discontinuation
- 2016-09-01 CN CN201680061132.2A patent/CN108137529A/zh active Pending
- 2016-09-01 US US15/757,204 patent/US10570166B2/en active Active
- 2016-09-01 AU AU2016317848A patent/AU2016317848A1/en not_active Abandoned
- 2016-09-01 CA CA2997499A patent/CA2997499A1/en not_active Abandoned
- 2016-09-01 EP EP16767084.3A patent/EP3344611B1/en active Active
- 2016-09-01 CA CA2997540A patent/CA2997540A1/en not_active Abandoned
- 2016-09-01 US US15/757,317 patent/US10717756B2/en active Active
- 2016-09-02 US US15/757,307 patent/US10711026B2/en active Active
- 2016-09-02 JP JP2018512326A patent/JP2018532707A/ja not_active Withdrawn
- 2016-09-02 KR KR1020187008941A patent/KR20180041755A/ko unknown
- 2016-09-02 CN CN201680057361.7A patent/CN108137528A/zh active Pending
- 2016-09-02 AU AU2016315860A patent/AU2016315860A1/en not_active Abandoned
- 2016-09-02 EP EP16766747.6A patent/EP3344610B1/en active Active
- 2016-09-02 WO PCT/US2016/050034 patent/WO2017040882A1/en active Application Filing
- 2016-09-02 CA CA2997639A patent/CA2997639A1/en not_active Abandoned
- 2016-09-02 MX MX2018002539A patent/MX2018002539A/es unknown
- 2016-09-02 WO PCT/US2016/050028 patent/WO2017040878A1/en active Application Filing
-
2018
- 2018-02-27 CL CL2018000525A patent/CL2018000525A1/es unknown
- 2018-02-27 IL IL257759A patent/IL257759A/en unknown
- 2018-02-27 CL CL2018000527A patent/CL2018000527A1/es unknown
- 2018-02-27 IL IL257760A patent/IL257760A/en unknown
Also Published As
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B06U | Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette] | ||
B11B | Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements |