BR112017020081B1 - Composto análogo deuterado de etifoxina, composição farmacêutica que o compreende e usos do referido composto - Google Patents
Composto análogo deuterado de etifoxina, composição farmacêutica que o compreende e usos do referido composto Download PDFInfo
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
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| US201562135979P | 2015-03-20 | 2015-03-20 | |
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| EP3347006B1 (en) * | 2015-03-20 | 2022-07-27 | GABA Therapeutics Inc. | Deuterated analogs of etifoxine, their derivatives and uses therof |
| US10420773B2 (en) | 2017-09-26 | 2019-09-24 | Ovid Therapeutics Inc. | Methods of treating developmental disorders and/or seizure disorders with etifoxine |
| JP2021519276A (ja) * | 2018-03-23 | 2021-08-10 | コンサート ファーマシューティカルズ インコーポレイテッド | Ｄ−β−ヒドロキシ酪酸の重水素化類似体およびその使用 |
| AU2019270173A1 (en) * | 2018-05-18 | 2020-12-03 | Ovid Therapeutics Inc. | Methods of treating attention deficit hyperactivity disorder |
| CN112125862A (zh) * | 2019-06-25 | 2020-12-25 | 上海安谱实验科技股份有限公司 | 一种稳定同位素标记的阿特拉津-d5及其合成方法 |
| WO2021097427A1 (en) | 2019-11-15 | 2021-05-20 | Karuna Therapeutics, Inc. | Xanomeline derivatives and methods for treating neurological disorders |
| KR20240050372A (ko) * | 2021-09-14 | 2024-04-18 | 난징 미노바 파마슈티컬 컴퍼니, 리미티드 | 수용성 알로프레그나놀론 유도체 및 이의 제조 방법과 용도 |
| WO2023218251A1 (en) * | 2022-05-10 | 2023-11-16 | Clearsynth Labs Limied | Novel deuterium-enriched nefazodone analogues and method for preparing thereof |
| EP4608408A2 (en) * | 2022-10-24 | 2025-09-03 | GABA Therapeutics Inc. | Deuterated analogs of etifoxine and methods of administration without autoinduction of metabolism |
| WO2025085958A1 (en) * | 2023-10-23 | 2025-05-01 | Glomesh Intl Pty Ltd | A module for mounting items |
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| FR2888748B1 (fr) | 2005-07-19 | 2007-10-12 | Biocodex | Composes neuroprotecteurs et compositions pharmaceutiques les comprenant |
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| US8110569B2 (en) * | 2006-03-20 | 2012-02-07 | The Regents Of The University Of California | Enantiomerically pure S-etifoxine, pharmaceutical compositions thereof and methods of their use |
| JP2011001308A (ja) * | 2009-06-19 | 2011-01-06 | Research Foundation Itsuu Laboratory | 重水素化カルボスチリル化合物 |
| SG10201505236YA (en) * | 2010-07-09 | 2015-08-28 | Teva Pharma | Deuterated n-ethyl-n-phenyl-1,2-dihydro-4-hydroxy-5-chloro-1-methyl-2-oxoquinoline-3-carboxamide, salts and uses thereof |
| US20140121407A1 (en) | 2011-07-05 | 2014-05-01 | Research Foundation Itsuu Laboratory | Deuterated phenylpropionic acid derivative |
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| EP3347006B1 (en) * | 2015-03-20 | 2022-07-27 | GABA Therapeutics Inc. | Deuterated analogs of etifoxine, their derivatives and uses therof |
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