BR112017011623A2 - composições farmacêuticas e processo para a preparação de uma composição - Google Patents
composições farmacêuticas e processo para a preparação de uma composiçãoInfo
- Publication number
- BR112017011623A2 BR112017011623A2 BR112017011623A BR112017011623A BR112017011623A2 BR 112017011623 A2 BR112017011623 A2 BR 112017011623A2 BR 112017011623 A BR112017011623 A BR 112017011623A BR 112017011623 A BR112017011623 A BR 112017011623A BR 112017011623 A2 BR112017011623 A2 BR 112017011623A2
- Authority
- BR
- Brazil
- Prior art keywords
- pharmaceutically acceptable
- compositions
- population
- composition
- present
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/12—Carboxylic acids; Salts or anhydrides thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
- A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
- A61K9/145—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1617—Organic compounds, e.g. phospholipids, fats
- A61K9/1623—Sugars or sugar alcohols, e.g. lactose; Derivatives thereof; Homeopathic globules
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Molecular Biology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Dispersion Chemistry (AREA)
- Emergency Medicine (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
a presente invenção refere-se a uma composição farmacêutica que compreende duas populações diferentes com a primeira população compreendendo oseltamivir ou um sal farmaceuticamente aceitável do mesmo e um ou mais excipientes farmaceuticamente aceitáveis e a segunda população compreendendo um ou mais excipientes farmaceuticamente aceitáveis. de preferência, as composições da segunda população não contêm oseltamivir ou um sal farmaceuticamente aceitável do mesmo. a presente invenção também descreve um novo método de enchimento da composição no recipiente. os inventores da presente invenção verificaram, surpreendentemente, que as composições são estáveis em condições de estabilidade a longo prazo e em tempo real. além disso, as composições são bioequivalentes à formulação de suspensão de mercado de fosfato de oseltamivir.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN1262KO2014 | 2014-12-01 | ||
PCT/IB2015/059198 WO2016088010A1 (en) | 2014-12-01 | 2015-11-30 | Oseltamivir compositions |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112017011623A2 true BR112017011623A2 (pt) | 2018-03-06 |
Family
ID=55069027
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112017011623A BR112017011623A2 (pt) | 2014-12-01 | 2015-11-30 | composições farmacêuticas e processo para a preparação de uma composição |
Country Status (3)
Country | Link |
---|---|
US (1) | US20170258749A1 (pt) |
BR (1) | BR112017011623A2 (pt) |
WO (1) | WO2016088010A1 (pt) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN110302151A (zh) * | 2019-07-16 | 2019-10-08 | 苏州二叶制药有限公司 | 含有磷酸奥司他韦的口服干混悬剂及其制备方法 |
CN111297823B (zh) * | 2020-03-04 | 2021-06-18 | 石药集团中奇制药技术(石家庄)有限公司 | 一种磷酸奥司他韦胶囊的制备方法 |
CN112121027B (zh) * | 2020-08-25 | 2023-01-17 | 北京民康百草医药科技有限公司 | 磷酸奥司他韦包衣颗粒的药物组合物、用途及制备方法 |
CN112494434A (zh) * | 2020-12-17 | 2021-03-16 | 江苏万珺医药科技有限公司 | 含有磷酸奥司他韦的干混悬剂及其制备方法 |
CN112717137B (zh) * | 2021-01-20 | 2022-12-30 | 澳美制药(苏州)有限公司 | 含有磷酸奥司他韦的药物组合物及其制备方法 |
CN115529815B (zh) * | 2021-04-27 | 2024-04-30 | 广州共禾医药科技有限公司 | 经直肠施用的奥司他韦或其药学上可接受的盐的药物组合物、及其制备方法和用途 |
CN116211810A (zh) * | 2023-03-21 | 2023-06-06 | 南京海鲸药业股份有限公司 | 一种磷酸奥司他韦干混悬剂的制备方法 |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5763483A (en) | 1995-12-29 | 1998-06-09 | Gilead Sciences, Inc. | Carbocyclic compounds |
US6605302B2 (en) * | 2001-07-17 | 2003-08-12 | Osmotica Corp. | Drug delivery device containing oseltamivir and an H1 antagonist |
WO2007097325A1 (ja) * | 2006-02-20 | 2007-08-30 | Chugai Seiyaku Kabushiki Kaisha | リン酸オセルタミビル含有医薬組成物 |
CN1820744B (zh) * | 2006-04-04 | 2011-01-26 | 中国人民解放军军事医学科学院毒物药物研究所 | 磷酸奥司他韦颗粒剂及其制备方法 |
US20120093738A1 (en) * | 2009-06-11 | 2012-04-19 | Rubicon Research Private Limited | Taste-masked oral formulations of influenza antivirals |
CN103315965B (zh) * | 2013-07-11 | 2015-08-05 | 河南中帅医药科技股份有限公司 | 一种适用于婴幼儿及儿童的口服固体颗粒及其制备方法 |
CN104138355A (zh) * | 2014-08-06 | 2014-11-12 | 广东东阳光药业有限公司 | 一种磷酸奥司他韦干混悬剂及其制备方法 |
-
2015
- 2015-11-30 WO PCT/IB2015/059198 patent/WO2016088010A1/en active Application Filing
- 2015-11-30 US US15/531,881 patent/US20170258749A1/en not_active Abandoned
- 2015-11-30 BR BR112017011623A patent/BR112017011623A2/pt not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
WO2016088010A1 (en) | 2016-06-09 |
US20170258749A1 (en) | 2017-09-14 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B11A | Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing | ||
B11Y | Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette] |