BR112014010997A2 - processo para o preparo de ß-glicosídeos de c-arila - Google Patents
processo para o preparo de ß-glicosídeos de c-arilaInfo
- Publication number
- BR112014010997A2 BR112014010997A2 BR112014010997A BR112014010997A BR112014010997A2 BR 112014010997 A2 BR112014010997 A2 BR 112014010997A2 BR 112014010997 A BR112014010997 A BR 112014010997A BR 112014010997 A BR112014010997 A BR 112014010997A BR 112014010997 A2 BR112014010997 A2 BR 112014010997A2
- Authority
- BR
- Brazil
- Prior art keywords
- glycosides
- aryl
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
- C07D309/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C07D309/08—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D309/10—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
- C07D407/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
- C07D407/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Saccharide Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyrane Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201161556780P | 2011-11-07 | 2011-11-07 | |
| US201261661793P | 2012-06-19 | 2012-06-19 | |
| PCT/IB2012/002894 WO2013068850A2 (en) | 2011-11-07 | 2012-11-07 | PROCESS FOR THE PREPARATION OF β-C-ARYL GLUCOSIDES |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR112014010997A2 true BR112014010997A2 (pt) | 2017-06-06 |
Family
ID=48290709
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR112014010997A BR112014010997A2 (pt) | 2011-11-07 | 2012-11-07 | processo para o preparo de ß-glicosídeos de c-arila |
Country Status (11)
| Country | Link |
|---|---|
| EP (1) | EP2776449B1 (pt) |
| JP (1) | JP6144686B2 (pt) |
| KR (1) | KR101756772B1 (pt) |
| CN (1) | CN103974964B (pt) |
| AU (1) | AU2012335280B2 (pt) |
| BR (1) | BR112014010997A2 (pt) |
| CA (1) | CA2854591A1 (pt) |
| IL (1) | IL232418A (pt) |
| IN (1) | IN2014CN04050A (pt) |
| TW (1) | TWI488861B (pt) |
| WO (1) | WO2013068850A2 (pt) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN104557894A (zh) * | 2013-10-18 | 2015-04-29 | 上海信谊药厂有限公司 | 坎格列汀晶型及其制备方法 |
| TWI592418B (zh) * | 2014-04-11 | 2017-07-21 | 台灣神隆股份有限公司 | β－Ｃ－芳基葡萄糖苷之製造方法 |
| CN105017237A (zh) * | 2014-04-29 | 2015-11-04 | 嘉实（湖南）医药科技有限公司 | 一种卡格列净的制备工艺 |
| EP2947077A1 (en) | 2014-05-19 | 2015-11-25 | LEK Pharmaceuticals d.d. | Stereoselective synthesis of intermediates in the preparation of ß-C-arylglucosides |
| US10370365B2 (en) | 2015-09-16 | 2019-08-06 | Optimus Drugs (P) Limited | Process for the preparation of Canagliflozin |
| CN105294624B (zh) * | 2015-11-16 | 2018-01-12 | 山东罗欣药业集团股份有限公司 | 一种达格列净的制备方法 |
| CN105486767B (zh) * | 2015-12-03 | 2018-03-13 | 上海应用技术学院 | 一种达格列净及其α‑异构体的分离方法 |
| CN105541815B (zh) * | 2015-12-24 | 2018-07-13 | 寿光富康制药有限公司 | 一种卡格列净的制备方法 |
| EP4114365A1 (en) | 2020-03-05 | 2023-01-11 | KRKA, d.d., Novo mesto | Pharmaceutical composition comprising sglt2 inhibitor |
| WO2021245253A1 (en) | 2020-06-05 | 2021-12-09 | Krka, D.D., Novo Mesto | Preparation of highly pure amorphous dapagliflozin |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5872599A (ja) * | 1981-10-27 | 1983-04-30 | Kanto Ishi Pharma Co Ltd | 複合糖質誘導体 |
| BR0317929A (pt) * | 2003-01-03 | 2006-04-11 | Bristol Myers Squibb Co | métodos de produzir inibidores de sglt2 de glicosìdeo de c-arila |
| AR056195A1 (es) * | 2005-09-15 | 2007-09-26 | Boehringer Ingelheim Int | Procedimientos para preparar derivados de (etinil-bencil)-benceno sustituidos de glucopiranosilo y compuestos intermedios de los mismos |
| WO2011064726A1 (en) | 2009-11-24 | 2011-06-03 | South African Medical Research Council | Method for the synthesis of aspalathin and analogues thereof |
-
2012
- 2012-11-07 JP JP2014539427A patent/JP6144686B2/ja not_active Expired - Fee Related
- 2012-11-07 EP EP12847376.6A patent/EP2776449B1/en not_active Not-in-force
- 2012-11-07 AU AU2012335280A patent/AU2012335280B2/en not_active Ceased
- 2012-11-07 CA CA2854591A patent/CA2854591A1/en not_active Abandoned
- 2012-11-07 BR BR112014010997A patent/BR112014010997A2/pt not_active Application Discontinuation
- 2012-11-07 WO PCT/IB2012/002894 patent/WO2013068850A2/en active Application Filing
- 2012-11-07 IN IN4050CHN2014 patent/IN2014CN04050A/en unknown
- 2012-11-07 KR KR1020147015420A patent/KR101756772B1/ko active IP Right Grant
- 2012-11-07 TW TW101141390A patent/TWI488861B/zh not_active IP Right Cessation
- 2012-11-07 CN CN201280054691.2A patent/CN103974964B/zh not_active Expired - Fee Related
-
2014
- 2014-05-01 IL IL232418A patent/IL232418A/en not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| AU2012335280B2 (en) | 2016-09-29 |
| CN103974964B (zh) | 2016-03-23 |
| WO2013068850A2 (en) | 2013-05-16 |
| EP2776449A4 (en) | 2015-10-07 |
| WO2013068850A3 (en) | 2013-08-22 |
| CA2854591A1 (en) | 2013-05-16 |
| IL232418A (en) | 2016-10-31 |
| IN2014CN04050A (pt) | 2015-07-10 |
| KR20140089427A (ko) | 2014-07-14 |
| AU2012335280A1 (en) | 2014-05-22 |
| WO2013068850A8 (en) | 2013-10-10 |
| TWI488861B (zh) | 2015-06-21 |
| TW201335175A (zh) | 2013-09-01 |
| KR101756772B1 (ko) | 2017-07-26 |
| CN103974964A (zh) | 2014-08-06 |
| EP2776449A2 (en) | 2014-09-17 |
| IL232418A0 (en) | 2014-06-30 |
| EP2776449B1 (en) | 2017-08-02 |
| JP6144686B2 (ja) | 2017-06-07 |
| JP2014532690A (ja) | 2014-12-08 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B11A | Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing | ||
| B11Y | Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette] |