BR112014010719A2 - moduladores não competitivos de receptor nicotínico - Google Patents
moduladores não competitivos de receptor nicotínicoInfo
- Publication number
- BR112014010719A2 BR112014010719A2 BR112014010719A BR112014010719A BR112014010719A2 BR 112014010719 A2 BR112014010719 A2 BR 112014010719A2 BR 112014010719 A BR112014010719 A BR 112014010719A BR 112014010719 A BR112014010719 A BR 112014010719A BR 112014010719 A2 BR112014010719 A2 BR 112014010719A2
- Authority
- BR
- Brazil
- Prior art keywords
- nicotinic receptor
- receptor modulators
- competitive
- compounds
- competitive nicotinic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C211/00—Compounds containing amino groups bound to a carbon skeleton
- C07C211/33—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings
- C07C211/34—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of a saturated carbon skeleton
- C07C211/38—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of a saturated carbon skeleton containing condensed ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C215/00—Compounds containing amino and hydroxy groups bound to the same carbon skeleton
- C07C215/42—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having amino groups or hydroxy groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C215/00—Compounds containing amino and hydroxy groups bound to the same carbon skeleton
- C07C215/42—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having amino groups or hydroxy groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
- C07C215/44—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having amino groups or hydroxy groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton bound to carbon atoms of the same ring or condensed ring system
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Addiction (AREA)
- Psychiatry (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
resumo patente de invenção: "moduladores não competitivos de receptor nicotínico". a presente invenção se refere a compostos que modulam receptores nicotínicos como antagonistas não competitivos. a presente invenção refere-se ainda a métodos para a síntese dos mesmos. são ainda descritas composições farmacêuticas compreendendo os referidos compostos, bem como usos e métodos empregados no tratamento ou na prevenção de uma doença ou condição mediada por um receptor nicotínico neuronal.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201161554998P | 2011-11-03 | 2011-11-03 | |
PCT/US2012/062940 WO2013067105A2 (en) | 2011-11-03 | 2012-11-01 | Nicotinic receptor non-competitive modulators |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112014010719A2 true BR112014010719A2 (pt) | 2017-05-02 |
Family
ID=48193026
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112014010719A BR112014010719A2 (pt) | 2011-11-03 | 2012-11-01 | moduladores não competitivos de receptor nicotínico |
Country Status (14)
Country | Link |
---|---|
US (1) | US20140288185A1 (pt) |
EP (1) | EP2773609A4 (pt) |
JP (1) | JP2014532708A (pt) |
KR (1) | KR20140098115A (pt) |
AU (1) | AU2012332545A1 (pt) |
BR (1) | BR112014010719A2 (pt) |
CA (1) | CA2853282A1 (pt) |
CL (1) | CL2014001137A1 (pt) |
IL (1) | IL232240A0 (pt) |
MX (1) | MX2014005216A (pt) |
RU (1) | RU2014122338A (pt) |
SG (1) | SG11201401984VA (pt) |
WO (1) | WO2013067105A2 (pt) |
ZA (1) | ZA201403502B (pt) |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3290215A (en) * | 1963-10-29 | 1966-12-06 | Du Pont | Use of methanoindanamines as antiviral agents |
US3317387A (en) * | 1964-05-25 | 1967-05-02 | Du Pont | Method of reducing the severity of influenza virus infections |
TW200306189A (en) * | 2002-03-21 | 2003-11-16 | Merz Pharma Gmbh & Co Kgaa | Azabicyclic, azatricyclic and azaspirocyclic derivatives of aminocyclohexane NMDA, 5HT3, and neuronal nicotinic receptor antagonists |
SG185643A1 (en) * | 2010-05-27 | 2012-12-28 | Targacept Inc | Nicotinic receptor non-competitive antagonists |
-
2012
- 2012-11-01 WO PCT/US2012/062940 patent/WO2013067105A2/en active Application Filing
- 2012-11-01 CA CA2853282A patent/CA2853282A1/en not_active Abandoned
- 2012-11-01 RU RU2014122338/04A patent/RU2014122338A/ru not_active Application Discontinuation
- 2012-11-01 KR KR1020147015185A patent/KR20140098115A/ko not_active Application Discontinuation
- 2012-11-01 EP EP12846619.0A patent/EP2773609A4/en not_active Withdrawn
- 2012-11-01 BR BR112014010719A patent/BR112014010719A2/pt not_active Application Discontinuation
- 2012-11-01 MX MX2014005216A patent/MX2014005216A/es not_active Application Discontinuation
- 2012-11-01 JP JP2014540061A patent/JP2014532708A/ja active Pending
- 2012-11-01 US US14/355,316 patent/US20140288185A1/en not_active Abandoned
- 2012-11-01 AU AU2012332545A patent/AU2012332545A1/en not_active Abandoned
- 2012-11-01 SG SG11201401984VA patent/SG11201401984VA/en unknown
-
2014
- 2014-04-24 IL IL232240A patent/IL232240A0/en unknown
- 2014-04-30 CL CL2014001137A patent/CL2014001137A1/es unknown
- 2014-05-14 ZA ZA2014/03502A patent/ZA201403502B/en unknown
Also Published As
Publication number | Publication date |
---|---|
IL232240A0 (en) | 2014-06-30 |
RU2014122338A (ru) | 2015-12-10 |
US20140288185A1 (en) | 2014-09-25 |
MX2014005216A (es) | 2014-08-22 |
CA2853282A1 (en) | 2013-05-10 |
KR20140098115A (ko) | 2014-08-07 |
EP2773609A2 (en) | 2014-09-10 |
WO2013067105A3 (en) | 2013-07-11 |
AU2012332545A1 (en) | 2014-05-29 |
CL2014001137A1 (es) | 2014-08-18 |
SG11201401984VA (en) | 2014-05-29 |
WO2013067105A2 (en) | 2013-05-10 |
EP2773609A4 (en) | 2015-06-24 |
JP2014532708A (ja) | 2014-12-08 |
ZA201403502B (en) | 2015-12-23 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B11A | Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing | ||
B11Y | Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette] | ||
B350 | Update of information on the portal [chapter 15.35 patent gazette] |