BR112012010635A2 - hidratos cristalinos, composições farmaceuticas e seus métodos de preparação e métodos para uso dos mesmos - Google Patents
hidratos cristalinos, composições farmaceuticas e seus métodos de preparação e métodos para uso dos mesmosInfo
- Publication number
- BR112012010635A2 BR112012010635A2 BR112012010635A BR112012010635A BR112012010635A2 BR 112012010635 A2 BR112012010635 A2 BR 112012010635A2 BR 112012010635 A BR112012010635 A BR 112012010635A BR 112012010635 A BR112012010635 A BR 112012010635A BR 112012010635 A2 BR112012010635 A2 BR 112012010635A2
- Authority
- BR
- Brazil
- Prior art keywords
- methods
- preparation
- pharmaceutical compositions
- crystalline hydrates
- hydrates
- Prior art date
Links
- 150000004677 hydrates Chemical class 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/18—Oxygen atoms
- C07D263/20—Oxygen atoms attached in position 2
- C07D263/22—Oxygen atoms attached in position 2 with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to other ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4965—Non-condensed pyrazines
- A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Oncology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US25792409P | 2009-11-04 | 2009-11-04 | |
PCT/CN2010/078377 WO2011054292A1 (en) | 2009-11-04 | 2010-11-03 | Certain crystalline hydrates, pharmaceutical compositions thereof and methods for preparation and use thereof |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112012010635A2 true BR112012010635A2 (pt) | 2018-03-20 |
Family
ID=43969571
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112012010635A BR112012010635A2 (pt) | 2009-11-04 | 2010-11-03 | hidratos cristalinos, composições farmaceuticas e seus métodos de preparação e métodos para uso dos mesmos |
Country Status (11)
Country | Link |
---|---|
US (1) | US8916567B2 (pt) |
EP (1) | EP2496563A4 (pt) |
JP (1) | JP2013510098A (pt) |
KR (1) | KR20130028703A (pt) |
CN (1) | CN102256951B (pt) |
AU (1) | AU2010314593B2 (pt) |
BR (1) | BR112012010635A2 (pt) |
HK (1) | HK1164311A1 (pt) |
RU (1) | RU2012122767A (pt) |
WO (1) | WO2011054292A1 (pt) |
ZA (1) | ZA201203531B (pt) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2013182070A1 (zh) * | 2012-06-08 | 2013-12-12 | 四川贝力克生物技术有限责任公司 | 一种用于预防或治疗分支杆菌疾病的药物 |
CN107456442A (zh) * | 2016-06-03 | 2017-12-12 | 四川赛卓药业股份有限公司 | 一种噁唑烷酮化合物的亚微乳注射剂及其制备方法和用途 |
CN107648181B (zh) * | 2016-07-25 | 2021-05-04 | 广东赛法洛药业有限公司 | 一种利他唑酮磷脂复合物及其制备方法和应用 |
CN112409285A (zh) * | 2020-11-30 | 2021-02-26 | 山东金城昆仑药业有限公司 | 噁唑烷酮类化合物的晶型及其制备方法和应用 |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1993009103A1 (en) * | 1991-11-01 | 1993-05-13 | The Upjohn Company | Substituted aryl- and heteroarylphenyloxazolidinones useful as antibacterial agents |
ATE372966T1 (de) * | 1994-03-25 | 2007-09-15 | Isotechnika Inc | Verbesserung der effektivität von arzneimitteln duren deuterierung |
US6334997B1 (en) * | 1994-03-25 | 2002-01-01 | Isotechnika, Inc. | Method of using deuterated calcium channel blockers |
AU729745B2 (en) * | 1997-07-11 | 2001-02-08 | Pharmacia & Upjohn Company | Thiadiazolyl and oxadiazolyl phenyl oxazolidinone antibacterial agents |
GB9821938D0 (en) * | 1998-10-09 | 1998-12-02 | Zeneca Ltd | Chemical compounds |
CN1155585C (zh) * | 2001-12-19 | 2004-06-30 | 中国医学科学院医药生物技术研究所 | 3,5-取代噁唑烷酮衍生物及其制备方法和应用 |
US20070185132A1 (en) * | 2003-07-02 | 2007-08-09 | Yasumichi Fukuda | Cyclopropyl group substituted oxazolidinone antibiotics and derivatives thereo |
CA2572207A1 (en) * | 2004-06-29 | 2006-10-19 | Teva Pharmaceutical Industries Ltd. | Solid forms of linezolid and processes for preparation thereof |
CN100538355C (zh) * | 2007-03-19 | 2009-09-09 | 四川贝力克生物技术有限责任公司 | 3,5-取代噁唑烷酮类化合物的纯度的检测方法 |
CN100473385C (zh) * | 2007-03-19 | 2009-04-01 | 四川贝力克生物技术有限责任公司 | 3,5-取代噁唑烷酮类化合物的溶解方法 |
CN100582749C (zh) * | 2007-03-19 | 2010-01-20 | 四川贝力克生物技术有限责任公司 | 3,5-取代噁唑烷酮类化合物的含量测定方法 |
-
2010
- 2010-11-03 AU AU2010314593A patent/AU2010314593B2/en not_active Expired - Fee Related
- 2010-11-03 BR BR112012010635A patent/BR112012010635A2/pt not_active IP Right Cessation
- 2010-11-03 JP JP2012537290A patent/JP2013510098A/ja active Pending
- 2010-11-03 RU RU2012122767/04A patent/RU2012122767A/ru not_active Application Discontinuation
- 2010-11-03 CN CN2010800036817A patent/CN102256951B/zh active Active
- 2010-11-03 EP EP10827906A patent/EP2496563A4/en not_active Withdrawn
- 2010-11-03 WO PCT/CN2010/078377 patent/WO2011054292A1/en active Application Filing
- 2010-11-03 KR KR1020127014444A patent/KR20130028703A/ko not_active Application Discontinuation
- 2010-11-03 US US12/938,555 patent/US8916567B2/en not_active Expired - Fee Related
-
2012
- 2012-05-15 ZA ZA2012/03531A patent/ZA201203531B/en unknown
- 2012-05-22 HK HK12105009.4A patent/HK1164311A1/xx not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
HK1164311A1 (en) | 2012-09-21 |
US20110136822A1 (en) | 2011-06-09 |
EP2496563A1 (en) | 2012-09-12 |
US8916567B2 (en) | 2014-12-23 |
AU2010314593A1 (en) | 2012-06-14 |
EP2496563A4 (en) | 2013-04-03 |
AU2010314593B2 (en) | 2015-05-21 |
CN102256951A (zh) | 2011-11-23 |
ZA201203531B (en) | 2013-07-31 |
CN102256951B (zh) | 2013-07-17 |
RU2012122767A (ru) | 2013-12-10 |
WO2011054292A1 (en) | 2011-05-12 |
KR20130028703A (ko) | 2013-03-19 |
JP2013510098A (ja) | 2013-03-21 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] | ||
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2465 DE 03-04-2018 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |