BR0214225A - Processos para a preparação e para a formação de um composto, e, composto - Google Patents

Processos para a preparação e para a formação de um composto, e, composto

Info

Publication number
BR0214225A
BR0214225A BR0214225-2A BR0214225A BR0214225A BR 0214225 A BR0214225 A BR 0214225A BR 0214225 A BR0214225 A BR 0214225A BR 0214225 A BR0214225 A BR 0214225A
Authority
BR
Brazil
Prior art keywords
compound
preparation
processes
formation
formula
Prior art date
Application number
BR0214225-2A
Other languages
English (en)
Inventor
Duncan Michael Gill
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of BR0214225A publication Critical patent/BR0214225A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/08Bridged systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/44Iso-indoles; Hydrogenated iso-indoles
    • C07D209/48Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D265/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/281,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/301,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D265/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/281,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/301,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
    • C07D265/321,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings with oxygen atoms directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

"PROCESSOS PARA A PREPARAçãO E PARA A FORMAçãO DE UM COMPOSTO, E, COMPOSTO". é fornecido um processo para a preparação de um composto de fórmula (I), cujo processo compreende a reação de um composto de fórmula (II), com cada um: (a) um formaldeído e um composto de fórmula (III), R^ a^-OH III e/ou (b) um derivado protegido de um formaldeìdo, em que R^ 1^, R^ 2^ e R^ a^ possuem os significados dados na descrição.
BR0214225-2A 2001-11-22 2002-11-20 Processos para a preparação e para a formação de um composto, e, composto BR0214225A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE0103908 2001-11-22
PCT/GB2002/005262 WO2003045956A1 (en) 2001-11-22 2002-11-20 Process for the preparation of 2-or-9-oxa-3, 7-diazabicyclo (3.3.1) nonanes from 2-aminomethyl-2, 3-dihydrooxazines, intermediates therefore, and processes for preparing such intermediates

Publications (1)

Publication Number Publication Date
BR0214225A true BR0214225A (pt) 2004-09-21

Family

ID=20286082

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0214225-2A BR0214225A (pt) 2001-11-22 2002-11-20 Processos para a preparação e para a formação de um composto, e, composto

Country Status (13)

Country Link
US (1) US20050014940A1 (pt)
EP (1) EP1468001A1 (pt)
JP (1) JP2005514376A (pt)
KR (1) KR20040054790A (pt)
CN (1) CN1589272A (pt)
AU (1) AU2002343067A1 (pt)
BR (1) BR0214225A (pt)
CA (1) CA2465840A1 (pt)
IL (1) IL161751A0 (pt)
MX (1) MXPA04004708A (pt)
NO (1) NO20042593L (pt)
WO (1) WO2003045956A1 (pt)
ZA (1) ZA200403782B (pt)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE9903759D0 (sv) * 1999-10-18 1999-10-18 Astra Ab Pharmaceutically active compounds

Also Published As

Publication number Publication date
US20050014940A1 (en) 2005-01-20
EP1468001A1 (en) 2004-10-20
IL161751A0 (en) 2005-11-20
MXPA04004708A (es) 2004-08-19
AU2002343067A1 (en) 2003-06-10
ZA200403782B (en) 2005-03-17
CA2465840A1 (en) 2003-06-05
KR20040054790A (ko) 2004-06-25
JP2005514376A (ja) 2005-05-19
CN1589272A (zh) 2005-03-02
WO2003045956A1 (en) 2003-06-05
NO20042593L (no) 2004-08-20

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 4A, 5A, 6A E 7A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 DA RPI 2034 DE 29/12/2009.