BR0211762A - Certos policetìdeos substituìdos, composições farmacêuticas contendo os mesmos e seu uso no tratamento de tumores - Google Patents
Certos policetìdeos substituìdos, composições farmacêuticas contendo os mesmos e seu uso no tratamento de tumoresInfo
- Publication number
- BR0211762A BR0211762A BR0211762-2A BR0211762A BR0211762A BR 0211762 A BR0211762 A BR 0211762A BR 0211762 A BR0211762 A BR 0211762A BR 0211762 A BR0211762 A BR 0211762A
- Authority
- BR
- Brazil
- Prior art keywords
- tumors
- treatment
- pharmaceutical compositions
- compositions containing
- certain substituted
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
- C07D309/16—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D309/28—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D309/30—Oxygen atoms, e.g. delta-lactones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Oncology (AREA)
- Hematology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyrane Compounds (AREA)
Abstract
"CERTOS POLICETìDEOS SUBSTITUìDOS, COMPOSIçõES FARMACêUTICAS CONTENDO OS MESMOS E SEU USO NO TRATAMENTO DE TUMORES". A presente invenção refere-se a certos policetídeos substituídos da fórmula I, em que A, B, C, D, E, F e m são como definido aqui, composições farmacêuticas contendo os ditos compostos, o uso dos ditos compostos no tratamento de tumores.
Applications Claiming Priority (6)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US31030701P | 2001-08-06 | 2001-08-06 | |
US34453201P | 2001-10-25 | 2001-10-25 | |
US34118901P | 2001-12-13 | 2001-12-13 | |
US34904702P | 2002-01-16 | 2002-01-16 | |
US35899702P | 2002-02-22 | 2002-02-22 | |
PCT/EP2002/008734 WO2003014102A1 (en) | 2001-08-06 | 2002-08-05 | Certain substituted polyketides, pharmaceutical compositions containing them and their use in treating tumors |
Publications (1)
Publication Number | Publication Date |
---|---|
BR0211762A true BR0211762A (pt) | 2004-10-13 |
Family
ID=27540954
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0211762-2A BR0211762A (pt) | 2001-08-06 | 2002-08-05 | Certos policetìdeos substituìdos, composições farmacêuticas contendo os mesmos e seu uso no tratamento de tumores |
Country Status (7)
Country | Link |
---|---|
US (2) | US6972292B2 (pt) |
EP (1) | EP1417195A1 (pt) |
JP (1) | JP4243183B2 (pt) |
CN (1) | CN100522956C (pt) |
BR (1) | BR0211762A (pt) |
CA (1) | CA2454081A1 (pt) |
WO (1) | WO2003014102A1 (pt) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2005084349A2 (en) * | 2004-03-02 | 2005-09-15 | Kosan Biosciences, Inc. | Compounds useful for the synthesis of (+)-discodermolide and methods therefor |
US7214708B2 (en) * | 2004-11-18 | 2007-05-08 | Kosan Biosciences Incorporated | Synthetic discodermolide analogs |
JPWO2020017141A1 (ja) * | 2018-07-17 | 2021-09-24 | Eneos株式会社 | 反応性希釈剤、組成物、封止材、硬化物、基板、電子部品、エポキシ化合物、及び化合物の製造方法 |
CN113527238B (zh) * | 2021-08-02 | 2022-12-13 | 昆明学院 | 一种海绵内生真菌来源的聚酮化合物及其在制备抗炎药物中的应用 |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4939168A (en) * | 1989-08-11 | 1990-07-03 | Harbor Branch Oceanographics Institution, Inc. | Discodermolide compounds, compositions containing same and methods of preparation and use |
US5789605A (en) | 1996-12-03 | 1998-08-04 | Trustees Of The University Of Pennsylvania | Synthetic techniques and intermediates for polyhydroxy, dienyl lactones and mimics thereof |
US6870058B2 (en) | 1996-12-03 | 2005-03-22 | The Trustees Of The University Of Pennsylvania | Compounds which mimic the chemical and biological properties of discodermolide |
US6242616B1 (en) * | 1996-12-03 | 2001-06-05 | The Trustees Of The University Of Pennsylvania | Synthetic techniques and intermediates for polyhydroxy, dienyl lactone derivatives |
US6096904A (en) | 1996-12-03 | 2000-08-01 | The Trustees Of The University Of Pennsylvania | Synthetic techniques and intermediates for polyhydroxy, dienyl lactone derivatives |
US6127406A (en) | 1998-10-09 | 2000-10-03 | Harbor Branch Oceanographic Institution, Inc. | Discodermolide compounds and methods of use |
-
2002
- 2002-08-05 BR BR0211762-2A patent/BR0211762A/pt not_active IP Right Cessation
- 2002-08-05 US US10/212,535 patent/US6972292B2/en not_active Expired - Fee Related
- 2002-08-05 EP EP02794555A patent/EP1417195A1/en not_active Withdrawn
- 2002-08-05 CA CA002454081A patent/CA2454081A1/en not_active Abandoned
- 2002-08-05 JP JP2003519052A patent/JP4243183B2/ja not_active Expired - Fee Related
- 2002-08-05 WO PCT/EP2002/008734 patent/WO2003014102A1/en active Application Filing
- 2002-08-05 CN CNB028154991A patent/CN100522956C/zh not_active Expired - Fee Related
-
2004
- 2004-09-28 US US10/951,857 patent/US7192980B2/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
CN1538964A (zh) | 2004-10-20 |
WO2003014102B1 (en) | 2003-11-27 |
CN100522956C (zh) | 2009-08-05 |
JP2004537598A (ja) | 2004-12-16 |
CA2454081A1 (en) | 2003-02-20 |
WO2003014102A1 (en) | 2003-02-20 |
JP4243183B2 (ja) | 2009-03-25 |
EP1417195A1 (en) | 2004-05-12 |
US20030087934A1 (en) | 2003-05-08 |
US6972292B2 (en) | 2005-12-06 |
US7192980B2 (en) | 2007-03-20 |
US20050049249A1 (en) | 2005-03-03 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
B15K | Others concerning applications: alteration of classification |
Free format text: PARA.INT.CI.C07D 309/30, C07C 271/12, A61P 35/00 Ipc: C07D 309/30 (2011.01), C07C 271/12 (2011.01), A61P |
|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 9A ANUIDADE(S). |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2144 DE 07/02/2012. |