BR0116836A - Processo para a preparação de um derivado de pirazolo[4,3-d]-pirimidina - Google Patents

Processo para a preparação de um derivado de pirazolo[4,3-d]-pirimidina

Info

Publication number
BR0116836A
BR0116836A BR0116836-3A BR0116836A BR0116836A BR 0116836 A BR0116836 A BR 0116836A BR 0116836 A BR0116836 A BR 0116836A BR 0116836 A BR0116836 A BR 0116836A
Authority
BR
Brazil
Prior art keywords
pyrazolo
preparation
pyrimidine derivative
pirazole
methoxybenzylamino
Prior art date
Application number
BR0116836-3A
Other languages
English (en)
Inventor
Hans-Michael Eggenweiler
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of BR0116836A publication Critical patent/BR0116836A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Pulmonology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

"PROCESSO PARA A PREPARAçãO DE UM DERIVADO DE PIRAZOLO[4,3-D]-PIRIMIDINA". A invenção refere-se a um processo para a preparação do ácido [7-(3-cloro-4-metoxibenzilamino)-1-metil-3-propil-1H-pirazolo[4,3-d]piri midin-5-il-metóxi]acético e aos seus intermediários.
BR0116836-3A 2001-01-27 2001-12-29 Processo para a preparação de um derivado de pirazolo[4,3-d]-pirimidina BR0116836A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10103647A DE10103647A1 (de) 2001-01-27 2001-01-27 Verfahren zur Herstellung eines Pyrazolo (4,3-d) pyrimidinderivates
PCT/EP2001/015372 WO2002059126A1 (en) 2001-01-27 2001-12-29 Process for the preparation of a pyrazolo[4,3-d]pyrimidine derivative

Publications (1)

Publication Number Publication Date
BR0116836A true BR0116836A (pt) 2004-02-03

Family

ID=7671918

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0116836-3A BR0116836A (pt) 2001-01-27 2001-12-29 Processo para a preparação de um derivado de pirazolo[4,3-d]-pirimidina

Country Status (16)

Country Link
US (1) US6960661B2 (pt)
EP (1) EP1358189A1 (pt)
JP (1) JP2004517152A (pt)
KR (1) KR20030069224A (pt)
CN (1) CN1531536A (pt)
BR (1) BR0116836A (pt)
CA (1) CA2435884A1 (pt)
CZ (1) CZ20031782A3 (pt)
DE (1) DE10103647A1 (pt)
HU (1) HUP0303001A2 (pt)
MX (1) MXPA03006508A (pt)
PL (1) PL361914A1 (pt)
RU (1) RU2003124066A (pt)
SK (1) SK8302003A3 (pt)
WO (1) WO2002059126A1 (pt)
ZA (1) ZA200306649B (pt)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19942474A1 (de) * 1999-09-06 2001-03-15 Merck Patent Gmbh Pyrazolo[4,3-d]pyrimidine
PL362513A1 (en) * 2000-12-19 2004-11-02 Merck Patent Gmbh Pharmaceutical formulation containing pyrazolo[4,3-d]pyrimidines and antithrombotic agents, calcium-antagonists, prostaglandins or prostaglandin derivatives

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4666908A (en) 1985-04-05 1987-05-19 Warner-Lambert Company 5-Substituted pyrazolo[4,3-d]pyrimidine-7-ones and methods of use
DE19644228A1 (de) * 1996-10-24 1998-04-30 Merck Patent Gmbh Thienopyrimidine
DE19752952A1 (de) 1997-11-28 1999-06-02 Merck Patent Gmbh Thienopyrimidine
DE19942474A1 (de) * 1999-09-06 2001-03-15 Merck Patent Gmbh Pyrazolo[4,3-d]pyrimidine

Also Published As

Publication number Publication date
MXPA03006508A (es) 2003-10-15
US20040053945A1 (en) 2004-03-18
CZ20031782A3 (cs) 2003-10-15
EP1358189A1 (en) 2003-11-05
HUP0303001A2 (hu) 2003-12-29
WO2002059126A1 (en) 2002-08-01
PL361914A1 (en) 2004-10-04
US6960661B2 (en) 2005-11-01
JP2004517152A (ja) 2004-06-10
ZA200306649B (en) 2004-09-08
KR20030069224A (ko) 2003-08-25
CA2435884A1 (en) 2002-08-01
SK8302003A3 (en) 2003-10-07
CN1531536A (zh) 2004-09-22
RU2003124066A (ru) 2005-01-10
DE10103647A1 (de) 2002-08-01

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Legal Events

Date Code Title Description
B11A Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing
B11Y Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette]