BR0112981A - Sais tartarato de derivado de tiazolidinadiona - Google Patents

Sais tartarato de derivado de tiazolidinadiona

Info

Publication number
BR0112981A
BR0112981A BR0112981-3A BR0112981A BR0112981A BR 0112981 A BR0112981 A BR 0112981A BR 0112981 A BR0112981 A BR 0112981A BR 0112981 A BR0112981 A BR 0112981A
Authority
BR
Brazil
Prior art keywords
tartrate salts
thiazolidinedione derivative
compound
derivative tartrate
salts
Prior art date
Application number
BR0112981-3A
Other languages
English (en)
Inventor
Bernadette Marie Choudary
Andrew Simon Craig
Tim Chien Ting Ho
Donald Colin Mackenzie
Deirdre O'keeffe
Original Assignee
Smithkline Beecham Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Plc filed Critical Smithkline Beecham Plc
Publication of BR0112981A publication Critical patent/BR0112981A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Cosmetics (AREA)

Abstract

"SAIS TARTARATO DE DERIVADO DE TIAZOLIDINADIONA". Um novo composto farmacêutico D (-)-tartarato de 5-[4-(N-metil-N-(2-piridil) amino) etoxi] benzil] tiazolidino-2,4-diona ou um seu solvato, um processo para preparação de um tal composto, uma composição farmacêutica compreendendo um tal composto e o uso de um tal composto em medicina.
BR0112981-3A 2000-08-04 2001-08-03 Sais tartarato de derivado de tiazolidinadiona BR0112981A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0019228.6A GB0019228D0 (en) 2000-08-04 2000-08-04 Novel pharmaceutical
PCT/GB2001/003515 WO2002012234A1 (en) 2000-08-04 2001-08-03 Tartrate salts of thiazolidinedione derivative

Publications (1)

Publication Number Publication Date
BR0112981A true BR0112981A (pt) 2003-08-26

Family

ID=9897030

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0112981-3A BR0112981A (pt) 2000-08-04 2001-08-03 Sais tartarato de derivado de tiazolidinadiona

Country Status (36)

Country Link
US (1) US20040048899A1 (pt)
EP (1) EP1305312B1 (pt)
JP (1) JP2004505972A (pt)
KR (1) KR100755173B1 (pt)
CN (1) CN1458931A (pt)
AP (1) AP1814A (pt)
AT (1) ATE393153T1 (pt)
AU (1) AU2001276509A1 (pt)
BG (1) BG107606A (pt)
BR (1) BR0112981A (pt)
CA (1) CA2417829A1 (pt)
CZ (1) CZ2003316A3 (pt)
DE (1) DE60133746T2 (pt)
DK (1) DK1305312T3 (pt)
DZ (1) DZ3467A1 (pt)
EA (1) EA004764B1 (pt)
EC (1) ECSP034469A (pt)
ES (1) ES2302506T3 (pt)
GB (1) GB0019228D0 (pt)
HK (1) HK1057359A1 (pt)
HR (1) HRP20030070A2 (pt)
HU (1) HUP0300777A3 (pt)
IL (2) IL154278A0 (pt)
MA (1) MA25898A1 (pt)
MX (1) MXPA03001087A (pt)
NO (1) NO324595B1 (pt)
NZ (1) NZ524032A (pt)
OA (1) OA12352A (pt)
PL (1) PL360703A1 (pt)
PT (1) PT1305312E (pt)
SI (1) SI1305312T1 (pt)
SK (1) SK1442003A3 (pt)
UA (1) UA76721C2 (pt)
WO (1) WO2002012234A1 (pt)
YU (1) YU16303A (pt)
ZA (1) ZA200300963B (pt)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
USRE39384E1 (en) 1993-09-01 2006-11-07 Smithkline Beecham P.L.C. Substituted thiazolidinedione derivatives
AR047530A1 (es) 2004-02-04 2006-01-25 Novartis Ag Formas de sal de 4-(4-metilpiperazin-1-ilmetil)-n-(4-metil-3-(4-piridin-3-il)pirimidin-2-ilamino)fenil)-benzamida
JP2008505075A (ja) * 2004-06-30 2008-02-21 イーライ リリー アンド カンパニー 1−(インドール−6−カルボニル−d−フェニルグリシニル)−4−(1−メチルピペリジン−4−イル)ピペラジンd−酒石酸塩
US7435741B2 (en) * 2006-05-09 2008-10-14 Teva Pharmaceutical Industries, Ltd. 2-N{5-[[4-[2-(methyl-2-pyridinylamino) ethoxy] phenyl]methyl]-2,4-thiazolidinedione} butanedioic acid, methods of preparation and compositions with rosiglitazone maleate
GB0616574D0 (en) * 2006-08-21 2006-09-27 Glaxo Group Ltd Compounds
DE102009053562A1 (de) 2009-11-18 2011-05-19 Alfred E. Tiefenbacher (Gmbh & Co. Kg) Rosiglitazonsuccinat enthaltende pharmazeutische Zusammensetzung
CN102532122B (zh) * 2010-12-29 2015-12-02 开封制药(集团)有限公司 酒石酸罗格列酮的制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0842925A1 (en) * 1987-09-04 1998-05-20 Beecham Group Plc Substituted thiazolidinedione derivatives
US6288095B1 (en) * 1987-09-04 2001-09-11 Beecham Group P.L.C. Compounds
GB9218830D0 (en) * 1992-09-05 1992-10-21 Smithkline Beecham Plc Novel compounds
US5741803A (en) * 1992-09-05 1998-04-21 Smithkline Beecham Plc Substituted thiazolidinedionle derivatives

Also Published As

Publication number Publication date
BG107606A (bg) 2003-09-30
NO324595B1 (no) 2007-11-26
SK1442003A3 (en) 2004-05-04
OA12352A (en) 2006-05-16
DK1305312T3 (da) 2008-07-28
EP1305312B1 (en) 2008-04-23
IL154278A (en) 2009-02-11
ATE393153T1 (de) 2008-05-15
PT1305312E (pt) 2008-06-19
YU16303A (sh) 2006-01-16
NO20030507D0 (no) 2003-01-31
DE60133746D1 (de) 2008-06-05
MXPA03001087A (es) 2003-05-27
IL154278A0 (en) 2003-09-17
DE60133746T2 (de) 2009-05-14
PL360703A1 (en) 2004-09-20
AU2001276509A1 (en) 2002-02-18
GB0019228D0 (en) 2000-09-27
KR20030022357A (ko) 2003-03-15
EP1305312A1 (en) 2003-05-02
NO20030507L (no) 2003-03-26
NZ524032A (en) 2004-07-30
HRP20030070A2 (en) 2005-02-28
MA25898A1 (fr) 2003-10-01
KR100755173B1 (ko) 2007-09-03
CA2417829A1 (en) 2002-02-14
WO2002012234A1 (en) 2002-02-14
DZ3467A1 (fr) 2002-02-14
AP2003002738A0 (en) 2003-03-31
HK1057359A1 (en) 2004-04-02
CZ2003316A3 (en) 2004-03-17
ECSP034469A (es) 2003-06-25
CN1458931A (zh) 2003-11-26
HUP0300777A3 (en) 2005-04-28
AP1814A (en) 2008-01-04
ZA200300963B (en) 2004-04-19
UA76721C2 (uk) 2006-09-15
EA200300234A1 (ru) 2003-06-26
SI1305312T1 (sl) 2008-08-31
US20040048899A1 (en) 2004-03-11
ES2302506T3 (es) 2008-07-16
HUP0300777A2 (hu) 2003-11-28
JP2004505972A (ja) 2004-02-26
EA004764B1 (ru) 2004-08-26

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 9A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2082 DE 30/11/2010.