BR0013349A - Processo para preparar uma formulação para liberação sustentada - Google Patents
Processo para preparar uma formulação para liberação sustentadaInfo
- Publication number
- BR0013349A BR0013349A BR0013349-3A BR0013349A BR0013349A BR 0013349 A BR0013349 A BR 0013349A BR 0013349 A BR0013349 A BR 0013349A BR 0013349 A BR0013349 A BR 0013349A
- Authority
- BR
- Brazil
- Prior art keywords
- preparing
- sustained release
- release formulation
- compound
- lgt
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
- A61K47/69—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit
- A61K47/6921—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit the form being a particulate, a powder, an adsorbate, a bead or a sphere
- A61K47/6927—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit the form being a particulate, a powder, an adsorbate, a bead or a sphere the form being a solid microparticle having no hollow or gas-filled cores
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
- A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
- A61K47/56—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule
- A61K47/59—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyureas or polyurethanes
- A61K47/593—Polyesters, e.g. PLGA or polylactide-co-glycolide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
- A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
- A61K47/62—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being a protein, peptide or polyamino acid
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Biological Depolymerization Polymers (AREA)
- Polyesters Or Polycarbonates (AREA)
Abstract
Patente de Invenção: "PROCESSO PARA PREPARAR UMA FORMULAçãO PARA LIBERAçãO SUSTENTADA". Esta invenção refere-se a um processo para preparar um complexo de liberação sustentada, Composto (I), o qual compreende o Composto (A), tendo fórmula (A), e um copolímero compreendendo ácido poli-(I)-láctico-glicólico-tartárico (P(I)LGT), em que o grupo amino do Composto (A) é ligado ionicamente a um grupo carboxila do P(I)LGT.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IE19990700A IES990700A2 (en) | 1999-08-18 | 1999-08-18 | Process to make a sustained release formulation |
PCT/IE2000/000099 WO2001012232A2 (en) | 1999-08-18 | 2000-08-14 | Process to make a sustained release formulation |
Publications (1)
Publication Number | Publication Date |
---|---|
BR0013349A true BR0013349A (pt) | 2002-04-23 |
Family
ID=11042112
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0013349-3A BR0013349A (pt) | 1999-08-18 | 2000-08-14 | Processo para preparar uma formulação para liberação sustentada |
Country Status (26)
Country | Link |
---|---|
US (1) | US6893645B1 (pt) |
EP (1) | EP1212095B1 (pt) |
JP (1) | JP3730917B2 (pt) |
CN (2) | CN1823736A (pt) |
AR (1) | AR022647A1 (pt) |
AT (1) | ATE243044T1 (pt) |
AU (1) | AU755229B2 (pt) |
BR (1) | BR0013349A (pt) |
CA (1) | CA2380902C (pt) |
CZ (1) | CZ294433B6 (pt) |
DE (1) | DE60003438T2 (pt) |
DK (1) | DK1212095T3 (pt) |
ES (1) | ES2195925T3 (pt) |
HK (1) | HK1044285A1 (pt) |
HU (1) | HUP0202895A3 (pt) |
IE (1) | IES990700A2 (pt) |
IL (1) | IL148044A0 (pt) |
MX (1) | MXPA02001415A (pt) |
NO (1) | NO20020762L (pt) |
NZ (1) | NZ517251A (pt) |
PL (1) | PL199862B1 (pt) |
PT (1) | PT1212095E (pt) |
RU (1) | RU2211694C1 (pt) |
TW (1) | TWI230069B (pt) |
WO (1) | WO2001012232A2 (pt) |
ZA (1) | ZA200202027B (pt) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
HUP0203060A3 (en) * | 1999-08-18 | 2003-11-28 | Sod Conseils Rech Applic | Sustained release complex of a peptide, process for its preparation and pharmaceutical composition containing the same |
US7109166B1 (en) | 1999-08-18 | 2006-09-19 | Societe De Conseils De Recherches Et D'applications Scientifiques, Sas | Sustained release formulation of a peptide |
EP1348444B1 (en) * | 1999-08-18 | 2006-04-12 | Societe De Conseils De Recherches Et D'applications Scientifiques S.A.S. | Sustained release formulation of a peptide complexed with a polymer |
JP5183068B2 (ja) * | 2003-12-22 | 2013-04-17 | フィンレイ,ウォーレン,エイチ | 大気噴出凍結乾燥法による粉末形成 |
JP2008518026A (ja) | 2004-10-27 | 2008-05-29 | ユニバーシティ・オブ・デンバー | 副腎皮質刺激ホルモンアナログおよびこれに関連する方法 |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5863985A (en) * | 1995-06-29 | 1999-01-26 | Kinerton Limited | Ionic molecular conjugates of biodegradable polyesters and bioactive polypeptides |
CA2150574A1 (en) * | 1993-01-06 | 1994-07-21 | Shalaby W. Shalaby | Ionic molecular conjugates of biodegradable polyesters and bioactive polypeptides |
US6221958B1 (en) * | 1993-01-06 | 2001-04-24 | Societe De Conseils De Recherches Et D'applications Scientifiques, Sas | Ionic molecular conjugates of biodegradable polyesters and bioactive polypeptides |
ATE284413T1 (de) | 1993-08-09 | 2004-12-15 | Sod Conseils Rech Applic | Therapeutische peptid derivate |
IE960308A1 (en) * | 1996-04-23 | 1997-11-05 | Kinerton Ltd | Sustained release ionic conjugate |
WO1998008528A1 (en) * | 1996-08-30 | 1998-03-05 | Biomeasure Incorporated | Method of inhibiting fibrosis with a somatostatin agonist |
US5972893A (en) * | 1997-05-06 | 1999-10-26 | Cedars-Sinai Medical Center | Method of treating hyperprolactinemia and prolactinomas |
PL342135A1 (en) | 1998-01-29 | 2001-05-21 | Kinerton Ltd | Method of obtaining absorbable microparticle |
EP1043079A4 (en) | 1998-08-28 | 2005-03-16 | Mitutoyo Corp | AUTOMATIC DEVICE FOR WASHING WORKPIECES BEFORE MEASURING AND AUTOMATIC PRODUCTION SYSTEM EQUIPPED WITH THIS AUTOMATIC WASHING DEVICE |
HUP0203060A3 (en) * | 1999-08-18 | 2003-11-28 | Sod Conseils Rech Applic | Sustained release complex of a peptide, process for its preparation and pharmaceutical composition containing the same |
-
1999
- 1999-08-18 IE IE19990700A patent/IES990700A2/xx not_active IP Right Cessation
-
2000
- 2000-08-07 TW TW089115867A patent/TWI230069B/zh not_active IP Right Cessation
- 2000-08-14 EP EP00951802A patent/EP1212095B1/en not_active Expired - Lifetime
- 2000-08-14 HU HU0202895A patent/HUP0202895A3/hu unknown
- 2000-08-14 PT PT00951802T patent/PT1212095E/pt unknown
- 2000-08-14 CN CNA2005100488321A patent/CN1823736A/zh active Pending
- 2000-08-14 WO PCT/IE2000/000099 patent/WO2001012232A2/en active IP Right Grant
- 2000-08-14 AT AT00951802T patent/ATE243044T1/de not_active IP Right Cessation
- 2000-08-14 CA CA002380902A patent/CA2380902C/en not_active Expired - Fee Related
- 2000-08-14 IL IL14804400A patent/IL148044A0/xx not_active IP Right Cessation
- 2000-08-14 AU AU64647/00A patent/AU755229B2/en not_active Ceased
- 2000-08-14 BR BR0013349-3A patent/BR0013349A/pt not_active IP Right Cessation
- 2000-08-14 PL PL354263A patent/PL199862B1/pl not_active IP Right Cessation
- 2000-08-14 MX MXPA02001415A patent/MXPA02001415A/es not_active Application Discontinuation
- 2000-08-14 NZ NZ517251A patent/NZ517251A/en unknown
- 2000-08-14 US US10/049,692 patent/US6893645B1/en not_active Expired - Fee Related
- 2000-08-14 JP JP2001516575A patent/JP3730917B2/ja not_active Expired - Fee Related
- 2000-08-14 ES ES00951802T patent/ES2195925T3/es not_active Expired - Lifetime
- 2000-08-14 DE DE60003438T patent/DE60003438T2/de not_active Expired - Lifetime
- 2000-08-14 CN CNB008113963A patent/CN1246040C/zh not_active Expired - Fee Related
- 2000-08-14 CZ CZ2002266A patent/CZ294433B6/cs not_active IP Right Cessation
- 2000-08-14 RU RU2002106809/04A patent/RU2211694C1/ru not_active IP Right Cessation
- 2000-08-14 DK DK00951802T patent/DK1212095T3/da active
- 2000-08-17 AR ARP000104254A patent/AR022647A1/es not_active Application Discontinuation
-
2002
- 2002-02-15 NO NO20020762A patent/NO20020762L/no not_active Application Discontinuation
- 2002-03-12 ZA ZA200202027A patent/ZA200202027B/xx unknown
- 2002-08-10 HK HK02105860A patent/HK1044285A1/xx not_active IP Right Cessation
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 6A, 7A E 8A ANUIDADES. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO PUBLICADO NA RPI 1962 DE 12/08/2008. |
|
B15K | Others concerning applications: alteration of classification |
Ipc: A61K 47/69 (2017.01), A61K 47/59 (2017.01), A61K 4 |