BG96204A - Имидазохиноксалини,нов клас gава лиганди на мозъчни рецептори - Google Patents
Имидазохиноксалини,нов клас gава лиганди на мозъчни рецепториInfo
- Publication number
- BG96204A BG96204A BG096204A BG9620492A BG96204A BG 96204 A BG96204 A BG 96204A BG 096204 A BG096204 A BG 096204A BG 9620492 A BG9620492 A BG 9620492A BG 96204 A BG96204 A BG 96204A
- Authority
- BG
- Bulgaria
- Prior art keywords
- imidazoquinoxalines
- gava
- new class
- receptor ligands
- brain receptor
- Prior art date
Links
- 210000004556 brain Anatomy 0.000 title abstract 2
- 239000003446 ligand Substances 0.000 title 1
- 239000000556 agonist Substances 0.000 abstract 2
- SVUOLADPCWQTTE-UHFFFAOYSA-N 1h-1,2-benzodiazepine Chemical compound N1N=CC=CC2=CC=CC=C12 SVUOLADPCWQTTE-UHFFFAOYSA-N 0.000 abstract 1
- YELMWJNXDALKFE-UHFFFAOYSA-N 3h-imidazo[4,5-f]quinoxaline Chemical class N1=CC=NC2=C(NC=N3)C3=CC=C21 YELMWJNXDALKFE-UHFFFAOYSA-N 0.000 abstract 1
- 206010012374 Depressed mood Diseases 0.000 abstract 1
- 206010041349 Somnolence Diseases 0.000 abstract 1
- 229940124277 aminobutyric acid Drugs 0.000 abstract 1
- 239000005557 antagonist Substances 0.000 abstract 1
- 229940049706 benzodiazepine Drugs 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 238000003745 diagnosis Methods 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 231100000252 nontoxic Toxicity 0.000 abstract 1
- 230000003000 nontoxic effect Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Имидазохиноксалините са силно селективни агонисти, антагонисти и инверсни агонисти на -аминобутировокисели мозъчни рецептори. Те се използват при диагностика и лечение на лошо настроение, сънливост и други подобни неразположения, при предозиране с лекарства от вида на бензодиазепините и за активизиране на паметта. Съединенията са с формула в която r1, r2, r3, r4, х и w имат различни значения. Изобретението се отнася и до техните фармацевтично приемливи нетоксични соли. 55 претенции
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| BG96204A BG60518B1 (bg) | 1992-04-09 | 1992-04-09 | Имидазохиноксалини,нов клас gава лиганди на мозъчни рецептори |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| BG96204A BG60518B1 (bg) | 1992-04-09 | 1992-04-09 | Имидазохиноксалини,нов клас gава лиганди на мозъчни рецептори |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| BG96204A true BG96204A (bg) | 1993-12-24 |
| BG60518B1 BG60518B1 (bg) | 1995-07-28 |
Family
ID=3924369
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG96204A BG60518B1 (bg) | 1992-04-09 | 1992-04-09 | Имидазохиноксалини,нов клас gава лиганди на мозъчни рецептори |
Country Status (1)
| Country | Link |
|---|---|
| BG (1) | BG60518B1 (bg) |
-
1992
- 1992-04-09 BG BG96204A patent/BG60518B1/bg unknown
Also Published As
| Publication number | Publication date |
|---|---|
| BG60518B1 (bg) | 1995-07-28 |
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