BG96204A - IMIDAZOQUINOXALINES, A NEW CLASS OF GAVA BRAIN RECEPTOR LIGANDS - Google Patents
IMIDAZOQUINOXALINES, A NEW CLASS OF GAVA BRAIN RECEPTOR LIGANDSInfo
- Publication number
- BG96204A BG96204A BG096204A BG9620492A BG96204A BG 96204 A BG96204 A BG 96204A BG 096204 A BG096204 A BG 096204A BG 9620492 A BG9620492 A BG 9620492A BG 96204 A BG96204 A BG 96204A
- Authority
- BG
- Bulgaria
- Prior art keywords
- imidazoquinoxalines
- gava
- new class
- receptor ligands
- brain receptor
- Prior art date
Links
- 210000004556 brain Anatomy 0.000 title abstract 2
- 239000003446 ligand Substances 0.000 title 1
- 239000000556 agonist Substances 0.000 abstract 2
- SVUOLADPCWQTTE-UHFFFAOYSA-N 1h-1,2-benzodiazepine Chemical compound N1N=CC=CC2=CC=CC=C12 SVUOLADPCWQTTE-UHFFFAOYSA-N 0.000 abstract 1
- YELMWJNXDALKFE-UHFFFAOYSA-N 3h-imidazo[4,5-f]quinoxaline Chemical class N1=CC=NC2=C(NC=N3)C3=CC=C21 YELMWJNXDALKFE-UHFFFAOYSA-N 0.000 abstract 1
- 206010012374 Depressed mood Diseases 0.000 abstract 1
- 206010041349 Somnolence Diseases 0.000 abstract 1
- 229940124277 aminobutyric acid Drugs 0.000 abstract 1
- 239000005557 antagonist Substances 0.000 abstract 1
- 229940049706 benzodiazepine Drugs 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 238000003745 diagnosis Methods 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 231100000252 nontoxic Toxicity 0.000 abstract 1
- 230000003000 nontoxic effect Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Имидазохиноксалините са силно селективни агонисти, антагонисти и инверсни агонисти на -аминобутировокисели мозъчни рецептори. Те се използват при диагностика и лечение на лошо настроение, сънливост и други подобни неразположения, при предозиране с лекарства от вида на бензодиазепините и за активизиране на паметта. Съединенията са с формула в която r1, r2, r3, r4, х и w имат различни значения. Изобретението се отнася и до техните фармацевтично приемливи нетоксични соли. 55 претенцииThe imidazoquinoxalines are highly selective agonists, antagonists and inverse agonists of -aminobutyric acid brain receptors. They are used in the diagnosis and treatment of low mood, drowsiness and other similar ailments, in overdose with drugs of the benzodiazepine type, and to activate memory. The compounds are of formula wherein r1, r2, r3, r4, x and w have different meanings. The invention also relates to their pharmaceutically acceptable non-toxic salts. 55 claims
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| BG96204A BG60518B1 (en) | 1992-04-09 | 1992-04-09 | Imidazoquinoxalines |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| BG96204A BG60518B1 (en) | 1992-04-09 | 1992-04-09 | Imidazoquinoxalines |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| BG96204A true BG96204A (en) | 1993-12-24 |
| BG60518B1 BG60518B1 (en) | 1995-07-28 |
Family
ID=3924369
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG96204A BG60518B1 (en) | 1992-04-09 | 1992-04-09 | Imidazoquinoxalines |
Country Status (1)
| Country | Link |
|---|---|
| BG (1) | BG60518B1 (en) |
-
1992
- 1992-04-09 BG BG96204A patent/BG60518B1/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| BG60518B1 (en) | 1995-07-28 |
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