BG60271B1 - 13-алкил-23-имино и 13-хало-23-имино производни на ll-f28249 и приложението им като ендо- и ектопаразитицидни, инсектицидни, акарицидни и нематоцидни средства - Google Patents

13-алкил-23-имино и 13-хало-23-имино производни на ll-f28249 и приложението им като ендо- и ектопаразитицидни, инсектицидни, акарицидни и нематоцидни средства

Info

Publication number
BG60271B1
BG60271B1 BG092811A BG9281190A BG60271B1 BG 60271 B1 BG60271 B1 BG 60271B1 BG 092811 A BG092811 A BG 092811A BG 9281190 A BG9281190 A BG 9281190A BG 60271 B1 BG60271 B1 BG 60271B1
Authority
BG
Bulgaria
Prior art keywords
imino
halo
alkyl
endo
ektoparasiticide
Prior art date
Application number
BG092811A
Other languages
English (en)
Other versions
BG60271B2 (bg
Inventor
Brian Buckwalter
Shin-Shyong Tseng
Timothy Barden
Original Assignee
Wyeth Holdings Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US07/405,808 external-priority patent/US5030650A/en
Priority claimed from US07/455,686 external-priority patent/US5055486A/en
Application filed by Wyeth Holdings Corporation filed Critical Wyeth Holdings Corporation
Publication of BG60271B1 publication Critical patent/BG60271B1/bg
Publication of BG60271B2 publication Critical patent/BG60271B2/bg

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/22—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains four or more hetero rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Environmental Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Biotechnology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Biochemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Molecular Biology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Някои 13-алкил-23-иминои 13-хало-23-иминопроизводни на ll-f28249 съединения, получени от ферментационен бульон на sтrертомyсеs сyаnеоgrisеus, подвид nоnсyаnоgеnus, с депозитен <216> nrrl-15773, са полезни за борба с ендои ектопаразитни инфекции по топлокръвни животни, както и за контролиране на насекоми, акари и нематоди по културни растения. 12 претенции
BG92811A 1989-09-11 1990-09-10 13-алкил-23-имино и 13-хало-23-имино производни на ll-f28249 и приложението им като ендо- и ектопаразитицидни, инсектицидни, акарицидни и нематоцидни средства BG60271B2 (bg)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US07/405,808 US5030650A (en) 1989-09-11 1989-09-11 13-halo-23-imino derivatives of LL-F28249 compounds and their use as endo- and ectoparasiticidal, insecticidal, acaricidal and nematocidal agents
US07/455,686 US5055486A (en) 1989-12-22 1989-12-22 13-alkyl-23-imino derivative of LL-F28249 compounds and their use as endo- and ectoparasiticidal, insecticidal, acaricidal and nematocidal agents

Publications (2)

Publication Number Publication Date
BG60271B1 true BG60271B1 (bg) 1994-03-31
BG60271B2 BG60271B2 (bg) 1994-03-31

Family

ID=27019245

Family Applications (1)

Application Number Title Priority Date Filing Date
BG92811A BG60271B2 (bg) 1989-09-11 1990-09-10 13-алкил-23-имино и 13-хало-23-имино производни на ll-f28249 и приложението им като ендо- и ектопаразитицидни, инсектицидни, акарицидни и нематоцидни средства

Country Status (21)

Country Link
EP (1) EP0423445B1 (bg)
JP (1) JP3026827B2 (bg)
KR (2) KR0160972B1 (bg)
CN (2) CN1032004C (bg)
AT (1) ATE130006T1 (bg)
AU (1) AU631454B2 (bg)
BG (1) BG60271B2 (bg)
BR (1) BR9004494A (bg)
DE (1) DE69023454T2 (bg)
DK (1) DK0423445T3 (bg)
ES (1) ES2081880T3 (bg)
GR (1) GR3018033T3 (bg)
HU (1) HU217357B (bg)
IE (1) IE71210B1 (bg)
IL (1) IL109791A (bg)
PL (1) PL164168B1 (bg)
PT (1) PT95241B (bg)
RU (1) RU2070885C1 (bg)
SI (1) SI9011710B (bg)
UA (1) UA41246C2 (bg)
YU (1) YU47592B (bg)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4988824A (en) * 1989-09-11 1991-01-29 Maulding Donald R Process for the preparation of 23-(C1-C6 alkyloxime)-LL-F28249 compounds
US5229416A (en) * 1992-04-29 1993-07-20 Merck & Co., Inc. Avermectin difluoro derivatives
DE19654079A1 (de) 1996-12-23 1998-06-25 Bayer Ag Endo-ekto-parasitizide Mittel
DE102004053964A1 (de) 2004-11-09 2006-05-11 Bayer Healthcare Ag Mittel gegen Demodikose
CN105085540B (zh) * 2015-08-12 2017-07-07 内蒙古佳瑞米精细化工有限公司 一种制备高含量尼莫克汀的方法
WO2019152808A1 (en) 2018-02-01 2019-08-08 Yale University Compositions and methods for inhibition of nuclear-penetrating antibodies

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ221077A (en) * 1986-07-18 1990-06-26 Ciba Geigy Ag 13b-alkyl milbemycins and use as parasiticides
ES2058082T3 (es) * 1986-09-12 1994-11-01 American Cyanamid Co Derivados 23-oxo (ceto) y 23-imino de compuestos ll-f28249.
US4831016A (en) * 1986-10-31 1989-05-16 Merck & Co., Inc. Reduced avermectin derivatives
US4886829A (en) * 1987-03-06 1989-12-12 American Cyanamid Company 23-Oxo (keto) and 23-imino derivatives of mono- and diepoxy LL-F28249 compounds
US4806527A (en) * 1987-03-16 1989-02-21 Merck & Co., Inc. Avermectin derivatives
US5830875A (en) * 1989-10-30 1998-11-03 Merck & Co., Inc. 24-and 25-substituted avermectin and milbemycin derivatives

Also Published As

Publication number Publication date
SI9011710B (sl) 2000-12-31
EP0423445A1 (en) 1991-04-24
CN1032004C (zh) 1996-06-12
DE69023454T2 (de) 1996-06-05
JPH03106886A (ja) 1991-05-07
AU631454B2 (en) 1992-11-26
EP0423445B1 (en) 1995-11-08
DE69023454D1 (de) 1995-12-14
HU217357B (hu) 2000-01-28
UA41246C2 (uk) 2001-09-17
CN1050193A (zh) 1991-03-27
JP3026827B2 (ja) 2000-03-27
PT95241A (pt) 1991-06-25
BR9004494A (pt) 1991-09-10
RU2070885C1 (ru) 1996-12-27
SI9011710A (sl) 1998-02-28
AU6235790A (en) 1991-03-14
PL286823A1 (en) 1991-10-07
YU171090A (sh) 1992-12-21
BG60271B2 (bg) 1994-03-31
PT95241B (pt) 1997-06-30
IL109791A (en) 1996-06-18
DK0423445T3 (da) 1995-12-11
PL164168B1 (pl) 1994-06-30
IE71210B1 (en) 1997-02-12
CN1053556C (zh) 2000-06-21
ATE130006T1 (de) 1995-11-15
HUT54691A (en) 1991-03-28
KR910006491A (ko) 1991-04-29
ES2081880T3 (es) 1996-03-16
YU47592B (sh) 1995-10-24
CN1115600A (zh) 1996-01-31
IE903274A1 (en) 1991-03-27
GR3018033T3 (en) 1996-02-29
KR0160972B1 (ko) 1998-12-01
KR0168751B1 (ko) 1999-01-15

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