BG17800A3 - Метод за получаване на 2-(5-нитро-2-фурил)-тиено (3,2-d)пиримидини - Google Patents
Метод за получаване на 2-(5-нитро-2-фурил)-тиено (3,2-d)пиримидиниInfo
- Publication number
- BG17800A3 BG17800A3 BG017732A BG1773270A BG17800A3 BG 17800 A3 BG17800 A3 BG 17800A3 BG 017732 A BG017732 A BG 017732A BG 1773270 A BG1773270 A BG 1773270A BG 17800 A3 BG17800 A3 BG 17800A3
- Authority
- BG
- Bulgaria
- Prior art keywords
- thieno
- pyrimidines
- furyl
- nitro
- preparation
- Prior art date
Links
- 150000003230 pyrimidines Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19691959403 DE1959403A1 (de) | 1969-11-26 | 1969-11-26 | Neue 2-(5-Nitro-2-furyl)-thieno[3,2-d]pyrimidine und Verfahren zu ihrer Herstellung |
DE19702050814 DE2050814A1 (de) | 1970-10-16 | 1970-10-16 | Neue Verfahren zur Herstellung von 2-(5-Nitro-2-furyl)-thieno eckige Klammer auf 3,2-d eckige Klammer zu pyrimidinen |
DE19702050815 DE2050815A1 (de) | 1970-10-16 | 1970-10-16 | Neue 2-(5-Nitro-2-furyl)-thieno eckige Klammer auf 3,2-d eckige Klammer zu pyrimidine |
DE19702050816 DE2050816A1 (de) | 1970-10-16 | 1970-10-16 | Neue 2-(Nitro-2-furyl>thieno eckige Klammer auf 3,2-d eckige Klammer zu pyrimidine |
Publications (1)
Publication Number | Publication Date |
---|---|
BG17800A3 true BG17800A3 (bg) | 1973-12-25 |
Family
ID=27430978
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BG016080A BG17799A3 (bg) | 1969-11-26 | 1970-11-17 | Метод за получаване на 2-/5-нитро-2-фурил/-тиено/3,2-d/ пиримидини |
BG017732A BG17800A3 (bg) | 1969-11-26 | 1970-11-17 | Метод за получаване на 2-(5-нитро-2-фурил)-тиено (3,2-d)пиримидини |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BG016080A BG17799A3 (bg) | 1969-11-26 | 1970-11-17 | Метод за получаване на 2-/5-нитро-2-фурил/-тиено/3,2-d/ пиримидини |
Country Status (13)
Country | Link |
---|---|
US (1) | US3661908A (ru) |
BE (1) | BE759493A (ru) |
BG (2) | BG17799A3 (ru) |
CA (1) | CA926865A (ru) |
CH (3) | CH559210A5 (ru) |
DK (1) | DK128781B (ru) |
FR (1) | FR2073416B1 (ru) |
GB (1) | GB1321316A (ru) |
IE (1) | IE34765B1 (ru) |
IL (1) | IL35729A (ru) |
NL (1) | NL7017210A (ru) |
NO (1) | NO129954B (ru) |
SE (1) | SE377938B (ru) |
Families Citing this family (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3932642A (en) * | 1971-04-10 | 1976-01-13 | Boehringer Ingelheim Gmbh | Biocidal compositions containing a 2- (5'-nitro-2'-furyl)-thieno(2,3-d) pyrimidine and methods of use |
US6187777B1 (en) | 1998-02-06 | 2001-02-13 | Amgen Inc. | Compounds and methods which modulate feeding behavior and related diseases |
US6608053B2 (en) * | 2000-04-27 | 2003-08-19 | Yamanouchi Pharmaceutical Co., Ltd. | Fused heteroaryl derivatives |
US20040138238A1 (en) * | 2002-08-08 | 2004-07-15 | Dhanoa Dale S. | Substituted aminopyrimidine compounds as neurokinin antagonists |
GB0423653D0 (en) * | 2004-10-25 | 2004-11-24 | Piramed Ltd | Pharmaceutical compounds |
TWI498332B (zh) * | 2006-04-26 | 2015-09-01 | Hoffmann La Roche | 作為pi3k抑制劑之嘧啶衍生物及相關製備方法、醫藥組合物、用途、套組及產物 |
AR060632A1 (es) * | 2006-04-26 | 2008-07-02 | Genentech Inc | Compuestos inhibidores de fosfoinositida 3- quinasa y metodos de uso |
NZ572812A (en) | 2006-04-26 | 2010-09-30 | Hoffmann La Roche | THIENO [3, 2-D] PYRIMIDINE Indazole DERIVATIVE USEFUL AS PI3K INHIBITOR |
NZ578162A (en) * | 2006-12-07 | 2011-12-22 | Genentech Inc | Phosphoinositide 3-kinase inhibitor compounds and methods of use |
KR101507182B1 (ko) * | 2006-12-07 | 2015-03-30 | 제넨테크, 인크. | 포스포이노시타이드 3-키나제 억제제 화합물 및 그의 사용 방법 |
EP2158207B1 (en) * | 2007-06-12 | 2011-05-25 | F. Hoffmann-La Roche AG | Thiazoliopyrimidines and their use as inhibitors of phosphatidylinositol-3 kinase |
ES2399774T3 (es) * | 2007-09-24 | 2013-04-03 | Genentech, Inc. | Compuestos de tiazolopirimidina inhibidores de PI3K y métodos de uso |
EP2214675B1 (en) | 2007-10-25 | 2013-11-20 | Genentech, Inc. | Process for making thienopyrimidine compounds |
GB0721095D0 (en) * | 2007-10-26 | 2007-12-05 | Piramed Ltd | Pharmaceutical compounds |
EP2405916B1 (en) | 2009-03-12 | 2018-02-07 | Genentech, Inc. | Combinations of phosphoinositide 3-kinase inhibitor compounds and chemotherapeutic agents for the treatment of hematopoietic malignancies |
CA2761445A1 (en) | 2009-05-27 | 2010-12-02 | Genentech, Inc. | Bicyclic pyrimidine pi3k inhibitor compounds selective for p110 delta, and methods of use |
WO2010136491A1 (en) * | 2009-05-27 | 2010-12-02 | F. Hoffmann-La Roche Ag | Bicyclic indole-pyrimidine pi3k inhibitor compounds selective for p110 delta, and methods of use |
US20110086837A1 (en) * | 2009-10-12 | 2011-04-14 | Genentech, Inc. | Combinations of a pi3k inhibitor and a mek inhibitor |
MX2012011887A (es) | 2010-04-16 | 2012-11-30 | Genentech Inc | Foxo 3a como biomarcador predictivo para la eficacia del inhibidor de la via de quinasa pi3k/akt. |
WO2012088254A1 (en) | 2010-12-22 | 2012-06-28 | Genentech, Inc. | Autophagy inducer and inhibitor combination therapy for the treatment of neoplasms |
WO2014130923A2 (en) | 2013-02-25 | 2014-08-28 | Genentech, Inc. | Methods and compositions for detecting and treating drug resistant akt mutant |
-
0
- BE BE759493D patent/BE759493A/xx unknown
-
1970
- 1970-11-17 BG BG016080A patent/BG17799A3/xx unknown
- 1970-11-17 BG BG017732A patent/BG17800A3/xx unknown
- 1970-11-18 US US90841A patent/US3661908A/en not_active Expired - Lifetime
- 1970-11-23 CH CH1731270A patent/CH559210A5/xx not_active IP Right Cessation
- 1970-11-23 CH CH1514674A patent/CH567029A5/xx not_active IP Right Cessation
- 1970-11-23 CH CH1514974A patent/CH568324A5/xx not_active IP Right Cessation
- 1970-11-25 NO NO04524/70A patent/NO129954B/no unknown
- 1970-11-25 GB GB5614670A patent/GB1321316A/en not_active Expired
- 1970-11-25 NL NL7017210A patent/NL7017210A/xx unknown
- 1970-11-25 DK DK601570AA patent/DK128781B/da unknown
- 1970-11-26 FR FR7042531A patent/FR2073416B1/fr not_active Expired
- 1970-11-26 CA CA099166A patent/CA926865A/en not_active Expired
- 1970-11-26 IE IE1519/70A patent/IE34765B1/xx unknown
- 1970-11-26 IL IL35729A patent/IL35729A/xx unknown
- 1970-11-26 SE SE7016054A patent/SE377938B/xx unknown
Also Published As
Publication number | Publication date |
---|---|
FR2073416B1 (ru) | 1975-04-18 |
NL7017210A (ru) | 1971-05-28 |
US3661908A (en) | 1972-05-09 |
IE34765L (en) | 1971-05-26 |
CH559210A5 (ru) | 1975-02-28 |
CA926865A (en) | 1973-05-22 |
GB1321316A (en) | 1973-06-27 |
BG17799A3 (bg) | 1973-12-25 |
DK128781B (da) | 1974-07-01 |
SE377938B (ru) | 1975-08-04 |
BE759493A (fr) | 1971-05-25 |
NO129954B (ru) | 1974-06-17 |
IL35729A0 (en) | 1971-01-28 |
FR2073416A1 (ru) | 1971-10-01 |
CH568324A5 (ru) | 1975-10-31 |
IE34765B1 (en) | 1975-08-06 |
CH567029A5 (ru) | 1975-09-30 |
IL35729A (en) | 1974-01-14 |
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