BE899464A - Composition a liberation soutenue de propanolol. - Google Patents
Composition a liberation soutenue de propanolol.Info
- Publication number
- BE899464A BE899464A BE0/212794A BE212794A BE899464A BE 899464 A BE899464 A BE 899464A BE 0/212794 A BE0/212794 A BE 0/212794A BE 212794 A BE212794 A BE 212794A BE 899464 A BE899464 A BE 899464A
- Authority
- BE
- Belgium
- Prior art keywords
- propranolol
- propanolol
- sustained release
- release composition
- granule
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
- A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Abstract
L'invention concerne un granule contenant du propranolol à absorption soutenue, destiné à l'administration par la voie orale. Ce granule est constitué d'un noyau de propranolol ou d'un sel pharmaceutiquement acceptable de ce dernier et d'un acide organique, noyés dans une matière polymère selon un agencement à couches multiples, et d'une membrane externe qui permet la libération du propranolol à une vitesse réglée dans un milieu aqueux.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IE91583 | 1983-04-21 |
Publications (1)
Publication Number | Publication Date |
---|---|
BE899464A true BE899464A (fr) | 1984-08-16 |
Family
ID=11019730
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE0/212794A BE899464A (fr) | 1983-04-21 | 1984-04-19 | Composition a liberation soutenue de propanolol. |
Country Status (6)
Country | Link |
---|---|
US (1) | US4898737A (fr) |
EP (1) | EP0123470A1 (fr) |
JP (1) | JPS59205314A (fr) |
BE (1) | BE899464A (fr) |
CH (1) | CH661434A5 (fr) |
PH (1) | PH18946A (fr) |
Families Citing this family (38)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB2170104A (en) * | 1985-01-30 | 1986-07-30 | Warner Lambert Co | Coated pharmaceutical dosage forms |
US5188840A (en) * | 1985-09-26 | 1993-02-23 | Chugai Seiyaku Kabushiki Kaisha | Slow-release pharmaceutical agent |
SE450087B (sv) * | 1985-10-11 | 1987-06-09 | Haessle Ab | Korn med kontrollerad frisettning av farmaceutiskt aktiva emnen som anbringats teckande pa ett kompakt olosligt kernmaterial |
SE455836B (sv) * | 1985-10-11 | 1988-08-15 | Haessle Ab | Beredning med kontrollerad frisettning innehallande ett salt av metoprolol samt metod for framstellning av denna beredning |
IE58401B1 (en) * | 1986-06-20 | 1993-09-08 | Elan Corp Plc | Controlled absorption pharmaceutical composition |
IT1200217B (it) * | 1986-09-30 | 1989-01-05 | Valducci Roberto | Membrana per uso farmaceutico ed industriale |
CA1323833C (fr) * | 1987-04-28 | 1993-11-02 | Yatindra M. Joshi | Compositions pharmaceutiques sous forme de granules et methode de fabrication |
US4808413A (en) * | 1987-04-28 | 1989-02-28 | E. R. Squibb & Sons, Inc. | Pharmaceutical compositions in the form of beadlets and method |
GB8722306D0 (en) * | 1987-09-22 | 1987-10-28 | Aps Research Ltd | Sustained-release formulation |
SE8703881D0 (sv) * | 1987-10-08 | 1987-10-08 | Haessle Ab | New pharmaceutical preparation |
ATE241987T1 (de) * | 1987-10-16 | 2003-06-15 | Elan Corp Plc | Diltiazem-zusammensetzungen mit kontrollierter wirkstoffabsorption |
PH27186A (en) * | 1989-09-07 | 1993-04-16 | Ciba Geigy Ag | Double-coated granules of disodium pamidronate |
US5229135A (en) * | 1991-11-22 | 1993-07-20 | Prographarm Laboratories | Sustained release diltiazem formulation |
US5422122A (en) * | 1992-08-04 | 1995-06-06 | Eurand America, Incorporated | Controlled release potassium chloride tablet |
WO1994014421A2 (fr) * | 1992-12-23 | 1994-07-07 | Saitec S.R.L. | Procede de preparation de produits pharmaceutiques a liberation lente et produits ainsi obtenus |
JP2535141B2 (ja) * | 1995-01-17 | 1996-09-18 | 中外製薬株式会社 | フマル酸含有徐放性製剤 |
US8071128B2 (en) | 1996-06-14 | 2011-12-06 | Kyowa Hakko Kirin Co., Ltd. | Intrabuccally rapidly disintegrating tablet and a production method of the tablets |
US6066339A (en) * | 1997-10-17 | 2000-05-23 | Elan Corporation, Plc | Oral morphine multiparticulate formulation |
US6090411A (en) * | 1998-03-09 | 2000-07-18 | Temple University | Monolithic tablet for controlled drug release |
US6524620B2 (en) | 1998-07-20 | 2003-02-25 | Andrx Pharmaceuticals, Inc. | Diltiazem controlled release formulation and method of manufacture |
DE19845358A1 (de) * | 1998-10-02 | 2000-04-06 | Roehm Gmbh | Überzogene Arzneiformen mit kontrollierter Wirkstoffabgabe |
US7052706B2 (en) * | 2001-06-08 | 2006-05-30 | Nostrum Pharmaceuticals, Inc. | Control release formulation containing a hydrophobic material as the sustained release agent |
US9358214B2 (en) * | 2001-10-04 | 2016-06-07 | Adare Pharmaceuticals, Inc. | Timed, sustained release systems for propranolol |
US7022342B2 (en) | 2002-03-28 | 2006-04-04 | Andrx Corporation, Inc. | Controlled release oral dosage form of beta-adrenergic blocking agents |
US9107804B2 (en) | 2002-12-10 | 2015-08-18 | Nortec Development Associates, Inc. | Method of preparing biologically active formulations |
US8367111B2 (en) | 2002-12-31 | 2013-02-05 | Aptalis Pharmatech, Inc. | Extended release dosage forms of propranolol hydrochloride |
US7632521B2 (en) * | 2003-07-15 | 2009-12-15 | Eurand, Inc. | Controlled release potassium chloride tablets |
WO2005123042A1 (fr) * | 2004-06-10 | 2005-12-29 | Glatt Air Techniques, Inc. | Preparation pharmaceutique a liberation lente |
US8747895B2 (en) * | 2004-09-13 | 2014-06-10 | Aptalis Pharmatech, Inc. | Orally disintegrating tablets of atomoxetine |
US9884014B2 (en) * | 2004-10-12 | 2018-02-06 | Adare Pharmaceuticals, Inc. | Taste-masked pharmaceutical compositions |
CA2584957C (fr) | 2004-10-21 | 2015-08-25 | Eurand Pharmaceuticals Limited | Compositions pharmaceutiques a saveur masquee avec substances porogenes gastrosolubles |
US20060099259A1 (en) * | 2004-11-05 | 2006-05-11 | Grant Heinicke | Propranolol formulations |
US20060099258A1 (en) * | 2004-11-05 | 2006-05-11 | Grant Heinicke | Propranolol formulations |
US20060105038A1 (en) * | 2004-11-12 | 2006-05-18 | Eurand Pharmaceuticals Limited | Taste-masked pharmaceutical compositions prepared by coacervation |
BRPI0609505A2 (pt) * | 2005-03-29 | 2010-04-13 | Rihm Gmbh | forma farmacêutica em multipartìculas compreendendo péletes com uma matriz que influencia o fornecimento de uma substáncia moduladora |
US9161918B2 (en) * | 2005-05-02 | 2015-10-20 | Adare Pharmaceuticals, Inc. | Timed, pulsatile release systems |
US20080187579A1 (en) * | 2007-02-01 | 2008-08-07 | Pavan Bhat | Extended-release dosage form |
WO2011067667A2 (fr) | 2009-12-02 | 2011-06-09 | Eurand Pharmaceuticals Limited | Microcapsules de fexofénadine et compositions les contenant |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS52139715A (en) * | 1976-05-14 | 1977-11-21 | Nippon Kayaku Co Ltd | Coated granules of alkali polyacrylate |
GB1561204A (en) * | 1977-06-01 | 1980-02-13 | Ici Ltd | Sustained release pharmaceutical composition |
IE48715B1 (en) * | 1978-12-22 | 1985-05-01 | Elan Corp Plc | New galencial forms for administration of medicaments by oral route,with programmed release and processes for preparing same |
US4248856A (en) * | 1979-07-10 | 1981-02-03 | American Home Products Corporation | Sustained release pharmaceutical compositions |
US4309406A (en) * | 1979-07-10 | 1982-01-05 | American Home Products Corporation | Sustained release pharmaceutical compositions |
US4248858A (en) * | 1979-08-09 | 1981-02-03 | American Home Products Corporation | Sustained release pharmaceutical compositions |
US4309404A (en) * | 1979-08-09 | 1982-01-05 | American Home Products Corporation | Sustained release pharmaceutical compositions |
US4248857A (en) * | 1979-08-09 | 1981-02-03 | American Home Products Corporation | Sustained release pharmaceutical compositions |
-
1984
- 1984-04-05 PH PH30502A patent/PH18946A/en unknown
- 1984-04-06 EP EP84302385A patent/EP0123470A1/fr not_active Ceased
- 1984-04-16 CH CH1893/84A patent/CH661434A5/fr not_active IP Right Cessation
- 1984-04-19 BE BE0/212794A patent/BE899464A/fr not_active IP Right Cessation
- 1984-04-21 JP JP59081019A patent/JPS59205314A/ja active Pending
-
1988
- 1988-04-27 US US07/188,090 patent/US4898737A/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
CH661434A5 (fr) | 1987-07-31 |
PH18946A (en) | 1985-11-14 |
JPS59205314A (ja) | 1984-11-20 |
EP0123470A1 (fr) | 1984-10-31 |
US4898737A (en) | 1990-02-06 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RE | Patent lapsed |
Owner name: ELAN CORP. P.L.C. Effective date: 19920430 |