BE884189A - Nouveaux aryl-1 arylsulfonyl-4 gamma-aminopropoxy-3, 1h-pyrazoles, medicament en contenant et procede pour les preparer - Google Patents
Nouveaux aryl-1 arylsulfonyl-4 gamma-aminopropoxy-3, 1h-pyrazoles, medicament en contenant et procede pour les preparerInfo
- Publication number
- BE884189A BE884189A BE0/201309A BE201309A BE884189A BE 884189 A BE884189 A BE 884189A BE 0/201309 A BE0/201309 A BE 0/201309A BE 201309 A BE201309 A BE 201309A BE 884189 A BE884189 A BE 884189A
- Authority
- BE
- Belgium
- Prior art keywords
- aminopropoxy
- pyrazoles
- arylsulfonyl
- gamma
- preparing
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/28—Two oxygen or sulfur atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR7917507A FR2460299A1 (fr) | 1979-07-05 | 1979-07-05 | Nouveaux derives du pyrazole et leur application therapeutique |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BE884189A true BE884189A (fr) | 1981-01-05 |
Family
ID=9227565
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BE0/201309A BE884189A (fr) | 1979-07-05 | 1980-07-04 | Nouveaux aryl-1 arylsulfonyl-4 gamma-aminopropoxy-3, 1h-pyrazoles, medicament en contenant et procede pour les preparer |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US4337263A (Direct) |
| JP (1) | JPS5615271A (Direct) |
| BE (1) | BE884189A (Direct) |
| CA (1) | CA1152507A (Direct) |
| DE (1) | DE3025579A1 (Direct) |
| ES (1) | ES8102561A1 (Direct) |
| FR (1) | FR2460299A1 (Direct) |
| GB (2) | GB2063870B (Direct) |
| IT (1) | IT8068062A0 (Direct) |
| NL (1) | NL8003888A (Direct) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ZA857592B (en) * | 1984-10-17 | 1986-05-28 | Heumann Ludwig & Co Gmbh | Pyrazole derivatives,processes for their preparation and pharmaceutical preparations containing these compounds |
| US4964895A (en) * | 1987-06-08 | 1990-10-23 | Monsanto Company | Substituted 4-(4-nitrophenoxy) pyrazoles and their use as herbicides |
| US6005109A (en) * | 1997-10-30 | 1999-12-21 | Pflizer Inc. | Pyrazoles and pyrazolopyrimidines having CRF antagonistic activity |
| US6103900A (en) * | 1992-12-17 | 2000-08-15 | Pfizer Inc | Pyrazoles and pyrazolopyrimidines having CRF antagonistic activity |
| NZ257770A (en) * | 1992-12-17 | 1997-02-24 | Pfizer | 3- acylpyrazole and pyrazolo[3,4-d]pyrimidine derivatives |
| US5646152A (en) * | 1994-06-15 | 1997-07-08 | Pfizer Inc. | Methods of administering CRF antagonists |
| EP1634872A1 (en) * | 2004-08-27 | 2006-03-15 | Laboratorios Del Dr. Esteve, S.A. | Pyrazole derivatives as sigma receptor inhibitors |
| US7696199B2 (en) * | 2004-08-27 | 2010-04-13 | Laboratorios Del Dr. Esteve, S.A. | Sigma receptor inhibitors |
| MX2007002341A (es) * | 2004-08-27 | 2007-09-25 | Esteve Labor Dr | Inhibidores del receptor sigma. |
| WO2007098953A1 (en) * | 2006-03-01 | 2007-09-07 | Laboratorios Del Dr. Esteve, S.A. | Pyrazole derivatives as sigma receptor inhibitors |
| EP1829875A1 (en) | 2006-03-01 | 2007-09-05 | Laboratorios Del Dr. Esteve, S.A. | Pyrazole derivatives as sigma receptor inhibitors |
| EP1829866A1 (en) * | 2006-03-02 | 2007-09-05 | Laboratorios Del Dr. Esteve, S.A. | Sigma receptor inhibitors |
| EP1829867A1 (en) | 2006-03-03 | 2007-09-05 | Laboratorios Del Dr. Esteve, S.A. | Imidazole compounds having pharmaceutical activity towards the sigma receptor |
| EP2529793B1 (en) * | 2007-06-08 | 2016-08-10 | Georgia State University Research Foundation, Inc. | Compositions for regulating or modulating quorum sensing in bacteria, methods of using the compounds, and methods of regulating or modulating quorum sensing in bacteria |
| EP2116539A1 (en) | 2008-04-25 | 2009-11-11 | Laboratorios Del. Dr. Esteve, S.A. | 1-aryl-3-aminoalkoxy-pyrazoles as sigma ligands enhancing analgesic effects of opioids and attenuating the dependency thereof |
| EP2353591A1 (en) | 2010-02-04 | 2011-08-10 | Laboratorios Del. Dr. Esteve, S.A. | Sigma ligands for potentiating the analgesic effect of opioids and opiates in post-operative pain and attenuating the dependency thereof |
| EP2388005A1 (en) | 2010-05-21 | 2011-11-23 | Laboratorios Del. Dr. Esteve, S.A. | Sigma ligands for the prevention and/or treatment of emesis induced by chemotherapy or radiotherapy |
| EP2395003A1 (en) | 2010-05-27 | 2011-12-14 | Laboratorios Del. Dr. Esteve, S.A. | Pyrazole compounds as sigma receptor inhibitors |
| EP2415471A1 (en) | 2010-08-03 | 2012-02-08 | Laboratorios Del. Dr. Esteve, S.A. | Use of sigma ligands in opioid-induced hyperalgesia |
| EP2524694A1 (en) | 2011-05-19 | 2012-11-21 | Laboratorios Del. Dr. Esteve, S.A. | Use of sigma ligands in diabetes type-2 associated pain |
| TW201607538A (zh) | 2013-12-17 | 2016-03-01 | 以斯提夫博士實驗室股份有限公司 | 血清素-去甲腎上腺素再攝取抑制劑(SNRIS)和σ受體配體組合物 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FI34517A (fi) | 1962-12-08 | 1964-10-10 | Laeaeketehdas Orion Oy | 5-pyratsolyylialkamiinieetterien valmistusmenetelmä |
| JPS4832112B1 (Direct) * | 1969-10-03 | 1973-10-04 | ||
| DE2409753A1 (de) * | 1974-03-01 | 1975-09-11 | Basf Ag | Substituierte pyrazole |
| FR2301250A1 (fr) | 1975-02-21 | 1976-09-17 | Bellon Labor Sa Roger | Nouveaux diaryl-1, 4o-aminoalcoxy-3 pyrazoles et leurs sels |
-
1979
- 1979-07-05 FR FR7917507A patent/FR2460299A1/fr active Granted
-
1980
- 1980-06-24 GB GB8100028A patent/GB2063870B/en not_active Expired
- 1980-06-24 GB GB8020609A patent/GB2054566B/en not_active Expired
- 1980-06-30 US US06/164,566 patent/US4337263A/en not_active Expired - Lifetime
- 1980-07-01 ES ES492986A patent/ES8102561A1/es not_active Expired
- 1980-07-03 CA CA000355323A patent/CA1152507A/fr not_active Expired
- 1980-07-04 BE BE0/201309A patent/BE884189A/fr unknown
- 1980-07-04 NL NL8003888A patent/NL8003888A/xx not_active Application Discontinuation
- 1980-07-04 IT IT8068062A patent/IT8068062A0/it unknown
- 1980-07-05 DE DE19803025579 patent/DE3025579A1/de not_active Withdrawn
- 1980-07-05 JP JP9216580A patent/JPS5615271A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| JPS5615271A (en) | 1981-02-14 |
| IT8068062A0 (it) | 1980-07-04 |
| NL8003888A (nl) | 1981-01-07 |
| GB2063870B (en) | 1983-06-22 |
| US4337263A (en) | 1982-06-29 |
| GB2054566A (en) | 1981-02-18 |
| GB2054566B (en) | 1983-05-18 |
| DE3025579A1 (de) | 1981-01-15 |
| CA1152507A (fr) | 1983-08-23 |
| GB2063870A (en) | 1981-06-10 |
| ES492986A0 (es) | 1981-02-16 |
| ES8102561A1 (es) | 1981-02-16 |
| FR2460299B1 (Direct) | 1983-01-14 |
| FR2460299A1 (fr) | 1981-01-23 |
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