BE884189A - Nouveaux aryl-1 arylsulfonyl-4 gamma-aminopropoxy-3, 1h-pyrazoles, medicament en contenant et procede pour les preparer - Google Patents

Nouveaux aryl-1 arylsulfonyl-4 gamma-aminopropoxy-3, 1h-pyrazoles, medicament en contenant et procede pour les preparer

Info

Publication number
BE884189A
BE884189A BE0/201309A BE201309A BE884189A BE 884189 A BE884189 A BE 884189A BE 0/201309 A BE0/201309 A BE 0/201309A BE 201309 A BE201309 A BE 201309A BE 884189 A BE884189 A BE 884189A
Authority
BE
Belgium
Prior art keywords
aminopropoxy
pyrazoles
arylsulfonyl
gamma
preparing
Prior art date
Application number
BE0/201309A
Other languages
English (en)
French (fr)
Inventor
H Techer
G Monnier
M Pesson
Original Assignee
Bellon Labor Sa Roger
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bellon Labor Sa Roger filed Critical Bellon Labor Sa Roger
Publication of BE884189A publication Critical patent/BE884189A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/28Two oxygen or sulfur atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BE0/201309A 1979-07-05 1980-07-04 Nouveaux aryl-1 arylsulfonyl-4 gamma-aminopropoxy-3, 1h-pyrazoles, medicament en contenant et procede pour les preparer BE884189A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7917507A FR2460299A1 (fr) 1979-07-05 1979-07-05 Nouveaux derives du pyrazole et leur application therapeutique

Publications (1)

Publication Number Publication Date
BE884189A true BE884189A (fr) 1981-01-05

Family

ID=9227565

Family Applications (1)

Application Number Title Priority Date Filing Date
BE0/201309A BE884189A (fr) 1979-07-05 1980-07-04 Nouveaux aryl-1 arylsulfonyl-4 gamma-aminopropoxy-3, 1h-pyrazoles, medicament en contenant et procede pour les preparer

Country Status (10)

Country Link
US (1) US4337263A (Direct)
JP (1) JPS5615271A (Direct)
BE (1) BE884189A (Direct)
CA (1) CA1152507A (Direct)
DE (1) DE3025579A1 (Direct)
ES (1) ES8102561A1 (Direct)
FR (1) FR2460299A1 (Direct)
GB (2) GB2063870B (Direct)
IT (1) IT8068062A0 (Direct)
NL (1) NL8003888A (Direct)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA857592B (en) * 1984-10-17 1986-05-28 Heumann Ludwig & Co Gmbh Pyrazole derivatives,processes for their preparation and pharmaceutical preparations containing these compounds
US4964895A (en) * 1987-06-08 1990-10-23 Monsanto Company Substituted 4-(4-nitrophenoxy) pyrazoles and their use as herbicides
US6005109A (en) * 1997-10-30 1999-12-21 Pflizer Inc. Pyrazoles and pyrazolopyrimidines having CRF antagonistic activity
US6103900A (en) * 1992-12-17 2000-08-15 Pfizer Inc Pyrazoles and pyrazolopyrimidines having CRF antagonistic activity
NZ257770A (en) * 1992-12-17 1997-02-24 Pfizer 3- acylpyrazole and pyrazolo[3,4-d]pyrimidine derivatives
US5646152A (en) * 1994-06-15 1997-07-08 Pfizer Inc. Methods of administering CRF antagonists
EP1634872A1 (en) * 2004-08-27 2006-03-15 Laboratorios Del Dr. Esteve, S.A. Pyrazole derivatives as sigma receptor inhibitors
US7696199B2 (en) * 2004-08-27 2010-04-13 Laboratorios Del Dr. Esteve, S.A. Sigma receptor inhibitors
MX2007002341A (es) * 2004-08-27 2007-09-25 Esteve Labor Dr Inhibidores del receptor sigma.
WO2007098953A1 (en) * 2006-03-01 2007-09-07 Laboratorios Del Dr. Esteve, S.A. Pyrazole derivatives as sigma receptor inhibitors
EP1829875A1 (en) 2006-03-01 2007-09-05 Laboratorios Del Dr. Esteve, S.A. Pyrazole derivatives as sigma receptor inhibitors
EP1829866A1 (en) * 2006-03-02 2007-09-05 Laboratorios Del Dr. Esteve, S.A. Sigma receptor inhibitors
EP1829867A1 (en) 2006-03-03 2007-09-05 Laboratorios Del Dr. Esteve, S.A. Imidazole compounds having pharmaceutical activity towards the sigma receptor
EP2529793B1 (en) * 2007-06-08 2016-08-10 Georgia State University Research Foundation, Inc. Compositions for regulating or modulating quorum sensing in bacteria, methods of using the compounds, and methods of regulating or modulating quorum sensing in bacteria
EP2116539A1 (en) 2008-04-25 2009-11-11 Laboratorios Del. Dr. Esteve, S.A. 1-aryl-3-aminoalkoxy-pyrazoles as sigma ligands enhancing analgesic effects of opioids and attenuating the dependency thereof
EP2353591A1 (en) 2010-02-04 2011-08-10 Laboratorios Del. Dr. Esteve, S.A. Sigma ligands for potentiating the analgesic effect of opioids and opiates in post-operative pain and attenuating the dependency thereof
EP2388005A1 (en) 2010-05-21 2011-11-23 Laboratorios Del. Dr. Esteve, S.A. Sigma ligands for the prevention and/or treatment of emesis induced by chemotherapy or radiotherapy
EP2395003A1 (en) 2010-05-27 2011-12-14 Laboratorios Del. Dr. Esteve, S.A. Pyrazole compounds as sigma receptor inhibitors
EP2415471A1 (en) 2010-08-03 2012-02-08 Laboratorios Del. Dr. Esteve, S.A. Use of sigma ligands in opioid-induced hyperalgesia
EP2524694A1 (en) 2011-05-19 2012-11-21 Laboratorios Del. Dr. Esteve, S.A. Use of sigma ligands in diabetes type-2 associated pain
TW201607538A (zh) 2013-12-17 2016-03-01 以斯提夫博士實驗室股份有限公司 血清素-去甲腎上腺素再攝取抑制劑(SNRIS)和σ受體配體組合物

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI34517A (fi) 1962-12-08 1964-10-10 Laeaeketehdas Orion Oy 5-pyratsolyylialkamiinieetterien valmistusmenetelmä
JPS4832112B1 (Direct) * 1969-10-03 1973-10-04
DE2409753A1 (de) * 1974-03-01 1975-09-11 Basf Ag Substituierte pyrazole
FR2301250A1 (fr) 1975-02-21 1976-09-17 Bellon Labor Sa Roger Nouveaux diaryl-1, 4o-aminoalcoxy-3 pyrazoles et leurs sels

Also Published As

Publication number Publication date
JPS5615271A (en) 1981-02-14
IT8068062A0 (it) 1980-07-04
NL8003888A (nl) 1981-01-07
GB2063870B (en) 1983-06-22
US4337263A (en) 1982-06-29
GB2054566A (en) 1981-02-18
GB2054566B (en) 1983-05-18
DE3025579A1 (de) 1981-01-15
CA1152507A (fr) 1983-08-23
GB2063870A (en) 1981-06-10
ES492986A0 (es) 1981-02-16
ES8102561A1 (es) 1981-02-16
FR2460299B1 (Direct) 1983-01-14
FR2460299A1 (fr) 1981-01-23

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