BE883856A - Nouvelles aroyl-4 amidazolones-2 utiles comme medicaments leur procede de preparation et compositions therapeutiques les contenant - Google Patents

Nouvelles aroyl-4 amidazolones-2 utiles comme medicaments leur procede de preparation et compositions therapeutiques les contenant Download PDF

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Publication number
BE883856A
BE883856A BE0/201057A BE201057A BE883856A BE 883856 A BE883856 A BE 883856A BE 0/201057 A BE0/201057 A BE 0/201057A BE 201057 A BE201057 A BE 201057A BE 883856 A BE883856 A BE 883856A
Authority
BE
Belgium
Prior art keywords
emi
radical
methyl
carbon atoms
branched
Prior art date
Application number
BE0/201057A
Other languages
English (en)
French (fr)
Inventor
R Dage
R Schnettler
J Grisar
Original Assignee
Richardson Merrell Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richardson Merrell Inc filed Critical Richardson Merrell Inc
Publication of BE883856A publication Critical patent/BE883856A/fr

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/70—One oxygen atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Cardiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BE0/201057A 1979-06-18 1980-06-17 Nouvelles aroyl-4 amidazolones-2 utiles comme medicaments leur procede de preparation et compositions therapeutiques les contenant BE883856A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US4980879A 1979-06-18 1979-06-18

Publications (1)

Publication Number Publication Date
BE883856A true BE883856A (fr) 1980-10-16

Family

ID=21961857

Family Applications (1)

Application Number Title Priority Date Filing Date
BE0/201057A BE883856A (fr) 1979-06-18 1980-06-17 Nouvelles aroyl-4 amidazolones-2 utiles comme medicaments leur procede de preparation et compositions therapeutiques les contenant

Country Status (4)

Country Link
JP (1) JPS565463A (enrdf_load_stackoverflow)
BE (1) BE883856A (enrdf_load_stackoverflow)
HU (1) HU192634B (enrdf_load_stackoverflow)
ZA (1) ZA803332B (enrdf_load_stackoverflow)

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4405628A (en) * 1981-03-05 1983-09-20 Merrell Dow Pharmaceuticals Inc. 4-Pyridylimidazolones and method of use
EP3763365A1 (en) 2019-07-09 2021-01-13 Breakthrough Medical Research B.V. Aroylimidazolones for the treatment of thaumetopoea exposure
WO2022018085A1 (en) 2020-07-20 2022-01-27 Breakthrough Medical Research B.V. Pde3 inhibitors for treating viral infections

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PH18106A (en) * 1981-02-18 1985-03-21 Merrell Dow Pharma Novel-4-aroylimidazol-2-ones
ZA821347B (en) * 1981-03-05 1983-01-26 Merrell Dow Pharma Novel aroylimidazole-2-ones
JPS6191249A (ja) * 1984-10-11 1986-05-09 Nippon Zeon Co Ltd ダストカバ−ブ−ツ用ゴム組成物
JPS6126662A (ja) * 1984-07-17 1986-02-05 Nippon Zeon Co Ltd ダストカバ−ブ−ツ用ゴム組成物

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4405628A (en) * 1981-03-05 1983-09-20 Merrell Dow Pharmaceuticals Inc. 4-Pyridylimidazolones and method of use
EP3763365A1 (en) 2019-07-09 2021-01-13 Breakthrough Medical Research B.V. Aroylimidazolones for the treatment of thaumetopoea exposure
WO2022018085A1 (en) 2020-07-20 2022-01-27 Breakthrough Medical Research B.V. Pde3 inhibitors for treating viral infections

Also Published As

Publication number Publication date
ZA803332B (en) 1981-01-28
HUT36099A (en) 1985-08-28
JPH0223548B2 (enrdf_load_stackoverflow) 1990-05-24
HU192634B (en) 1987-06-29
JPS565463A (en) 1981-01-20

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Legal Events

Date Code Title Description
CCPA Application for a supplementary protection certificate

Free format text: 093C0168

CCPV Grant of a supplementary protection certificate

Free format text: 093C0168, EXPIRES 20021027

RE20 Patent expired

Owner name: MERRELL DOW PHARMACEUTICALS INC.

Effective date: 20000617