BE869133A - NEW DERIVATIVES OF INDOLE, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS - Google Patents

NEW DERIVATIVES OF INDOLE, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS

Info

Publication number
BE869133A
BE869133A BE189392A BE189392A BE869133A BE 869133 A BE869133 A BE 869133A BE 189392 A BE189392 A BE 189392A BE 189392 A BE189392 A BE 189392A BE 869133 A BE869133 A BE 869133A
Authority
BE
Belgium
Prior art keywords
indole
preparation
application
medicinal products
new derivatives
Prior art date
Application number
BE189392A
Other languages
French (fr)
Original Assignee
Sandoz Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from CH907777A external-priority patent/CH632246A5/en
Application filed by Sandoz Sa filed Critical Sandoz Sa
Publication of BE869133A publication Critical patent/BE869133A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/30Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/42Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/12Radicals substituted by oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/30Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Indole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
BE189392A 1977-07-21 1978-07-19 NEW DERIVATIVES OF INDOLE, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS BE869133A (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
CH907077 1977-07-21
CH906577 1977-07-21
CH907777A CH632246A5 (en) 1977-07-21 1977-07-21 Process for preparing novel 3-aminopropoxyindoles
CH907377 1977-07-21

Publications (1)

Publication Number Publication Date
BE869133A true BE869133A (en) 1979-01-19

Family

ID=27429188

Family Applications (1)

Application Number Title Priority Date Filing Date
BE189392A BE869133A (en) 1977-07-21 1978-07-19 NEW DERIVATIVES OF INDOLE, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS

Country Status (18)

Country Link
JP (1) JPS5422364A (en)
AU (1) AU523105B2 (en)
BE (1) BE869133A (en)
CA (1) CA1098909A (en)
DE (1) DE2830211A1 (en)
DK (1) DK312878A (en)
ES (1) ES471863A1 (en)
FI (1) FI782229A (en)
FR (1) FR2398058A1 (en)
GB (1) GB2001971B (en)
IE (1) IE47131B1 (en)
IL (1) IL55170A (en)
IT (1) IT1105092B (en)
NL (1) NL7807626A (en)
NZ (1) NZ187909A (en)
PT (1) PT68317A (en)
SE (1) SE435374B (en)
SU (1) SU843740A3 (en)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2905877A1 (en) * 1979-02-16 1980-08-28 Boehringer Mannheim Gmbh NEW AMINOPROPANOL DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND MEDICINAL PRODUCTS CONTAINING THESE COMPOUNDS
EP0025111B1 (en) * 1979-08-10 1984-07-25 Sandoz Ag 3-aminopropoxyaryl derivatives, their preparation and pharmaceutical compositions containing them
DE3030047A1 (en) * 1980-08-08 1982-03-11 Boehringer Mannheim Gmbh, 6800 Mannheim NEW AMINOPROPANOL DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND MEDICINAL PRODUCTS CONTAINING THESE COMPOUNDS
DE3029980A1 (en) * 1980-08-08 1982-03-11 Boehringer Mannheim Gmbh, 6800 Mannheim INDOLDER DERIVATIVES AND METHOD FOR THEIR PRODUCTION
DE3131146A1 (en) * 1981-08-06 1983-02-24 Boehringer Mannheim Gmbh, 6800 Mannheim NEW HETEROARYLOXYPROPANOLAMINE, METHOD FOR THE PRODUCTION THEREOF AND MEDICINAL PRODUCTS CONTAINING THESE COMPOUNDS
ZA967892B (en) * 1995-09-21 1998-03-18 Lilly Co Eli Selective β3 adrenergic agonists.
US6818660B2 (en) 1996-04-09 2004-11-16 Nps Pharmaceuticals, Inc. Calcilytic compounds
AU726659B2 (en) * 1996-04-09 2000-11-16 Nps Pharmaceuticals, Inc. Calcilytic compounds
ES2171839T3 (en) * 1996-09-05 2002-09-16 Lilly Co Eli CARBAZOL ANALOGS AS BETA3 SELECTIVE ADRENERGIC AGONISTS.
TW483881B (en) 1996-12-03 2002-04-21 Nps Pharma Inc Calcilytic compounds
US7202261B2 (en) 1996-12-03 2007-04-10 Nps Pharmaceuticals, Inc. Calcilytic compounds
AU1580001A (en) * 1999-11-15 2001-05-30 Eli Lilly And Company Process for the preparation of aryloxy propanolamines
US11173144B2 (en) 2016-05-13 2021-11-16 The Board Of Trustees Of The Leland Stanford Junior University Adrenergic receptor modulating compounds and methods of using the same

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1547056A (en) * 1966-12-13 1968-11-22 Sandoz Sa Indole derivatives and their preparation
FR2019185A1 (en) * 1968-09-30 1970-06-26 Sandoz Sa 4-(2-hydroxy-3-amino-propoxy)-indole-2-carboxy- - lic acids and esters and 2-hydroxymethylindoles as beta
US3699123A (en) * 1970-03-24 1972-10-17 Sandoz Ltd 4-(3-amino-2-hydroxy-propoxy) indole derivatives
US4076829A (en) * 1974-11-16 1978-02-28 Boehringer Mannheim Gmbh Aminopropanol compounds and compositions for the treatment of cardiac and circulatory diseases
DE2508251C2 (en) * 1975-02-26 1983-12-29 Boehringer Mannheim Gmbh, 6800 Mannheim Derivatives of indole, processes for their preparation and medicaments containing them
DE2633839A1 (en) * 1975-08-07 1977-02-24 Sandoz Ag NEW 4-AMINOPROPOXYINDOLDE DERIVATIVES, THEIR PRODUCTION AND USE
DE2635209C2 (en) * 1975-08-15 1983-01-27 Sandoz-Patent-GmbH, 7850 Lörrach 4- (2-Benzoyloxy-3-tert-butylamino-propoxy) -2-methylindole, its (S) -enantiomer, their acid addition salts, processes for their preparation and medicaments containing these compounds

Also Published As

Publication number Publication date
IE781448L (en) 1979-01-21
IL55170A (en) 1982-07-30
DK312878A (en) 1979-01-22
PT68317A (en) 1978-08-01
SE435374B (en) 1984-09-24
FR2398058A1 (en) 1979-02-16
AU3818278A (en) 1980-01-24
SU843740A3 (en) 1981-06-30
FI782229A (en) 1979-01-22
FR2398058B1 (en) 1982-08-06
GB2001971A (en) 1979-02-14
NZ187909A (en) 1981-04-24
IT7850299A0 (en) 1978-07-14
IL55170A0 (en) 1978-09-29
NL7807626A (en) 1979-01-23
AU523105B2 (en) 1982-07-15
GB2001971B (en) 1982-02-10
CA1098909A (en) 1981-04-07
IT1105092B (en) 1985-10-28
IE47131B1 (en) 1983-12-28
SE7807753L (en) 1979-01-22
ES471863A1 (en) 1979-10-01
DE2830211A1 (en) 1979-02-01
JPS5422364A (en) 1979-02-20

Similar Documents

Publication Publication Date Title
BE838509A (en) NEW ISOXAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS
FR2336135A1 (en) NEW ERGOLINE DERIVATIVES, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS
BE869133A (en) NEW DERIVATIVES OF INDOLE, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS
FR2333504A1 (en) NEW INDAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS
BE839967R (en) NEW ISOQUINOLEINE DERIVATIVES, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS
FR2339598A1 (en) NEW DERIVATIVES OF PYRROLIDINE, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS
BE860613A (en) NEW DERIVATIVES OF MORPHANTHRIDINE, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS
FR2341577A1 (en) NEW DERIVATIVES OF PIPERAZINE, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS
FR2320090A1 (en) NEW DERIVATIVES OF INDOLE, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS
LU81027A1 (en) NEW DERIVATIVES OF N-PHENYLALANINE, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS
BE863215A (en) NEW DERIVATIVES OF BENZO (F) ISOQUINOLEINE, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS
FR2310756A1 (en) NEW DERIVATIVES OF QUINAZOLINE, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS
BE839969A (en) NEW ISOQUINOLEINE DERIVATIVES, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS
BE859084A (en) NEW DERIVATIVES OF IMIDAZO (5,1-A) ISOQUINOLEINE, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS
FR2335225A1 (en) NEW ISOQUINOLEINE DERIVATIVES, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS
BE850050R (en) NEW ERGOLINE DERIVATIVES, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS
BE865267A (en) NEW DERIVATIVES OF RYE ERGOT, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS
FR2323386A1 (en) NEW DERIVATIVES OF BENZO-CYCLOHEPTA-PYRIDINE, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS
BE844881A (en) NEW DERIVATIVES OF MORPHANTHRIDINE, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS
FR2302090A1 (en) NEW DERIVATIVES OF INDOLINE, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS
FR2313936A1 (en) NEW DERIVATIVES OF BENZO (G) ISOQUINOLEINE, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS
BE855168R (en) NEW DERIVATIVES OF INDOLINE, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS
BE854323A (en) NEW DERIVATIVES OF INDOLINE, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS
BE843039A (en) NEW BENZO-CYCLOCHEPTA-THIOPHENE DERIVATIVES, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS
FR2313048A1 (en) NEW DERIVATIVES OF INDOLINE, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS

Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: SANDOZ S.A.

Effective date: 19860731