BE868881A - Alpha-halogenomethyl-amino-acides et leurs derives, leur preparation et leur utilisation - Google Patents

Alpha-halogenomethyl-amino-acides et leurs derives, leur preparation et leur utilisation

Info

Publication number
BE868881A
BE868881A BE189190A BE189190A BE868881A BE 868881 A BE868881 A BE 868881A BE 189190 A BE189190 A BE 189190A BE 189190 A BE189190 A BE 189190A BE 868881 A BE868881 A BE 868881A
Authority
BE
Belgium
Prior art keywords
halogenomethyl
alpha
derivatives
acids
amino
Prior art date
Application number
BE189190A
Other languages
English (en)
French (fr)
Original Assignee
Merrell Toraude & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merrell Toraude & Co filed Critical Merrell Toraude & Co
Publication of BE868881A publication Critical patent/BE868881A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06191Dipeptides containing heteroatoms different from O, S, or N
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Peptides Or Proteins (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
BE189190A 1977-07-11 1978-07-10 Alpha-halogenomethyl-amino-acides et leurs derives, leur preparation et leur utilisation BE868881A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US81424377A 1977-07-11 1977-07-11

Publications (1)

Publication Number Publication Date
BE868881A true BE868881A (fr) 1978-11-03

Family

ID=25214519

Family Applications (1)

Application Number Title Priority Date Filing Date
BE189190A BE868881A (fr) 1977-07-11 1978-07-10 Alpha-halogenomethyl-amino-acides et leurs derives, leur preparation et leur utilisation

Country Status (16)

Country Link
JP (1) JPS5484544A (de)
AU (1) AU525684B2 (de)
BE (1) BE868881A (de)
CH (1) CH636846A5 (de)
DE (1) DE2828738A1 (de)
DK (1) DK309378A (de)
ES (3) ES471595A1 (de)
FR (1) FR2397391A1 (de)
GB (1) GB2005659B (de)
IE (1) IE46932B1 (de)
IL (1) IL54913A0 (de)
IT (1) IT1105534B (de)
NL (1) NL7807454A (de)
NZ (1) NZ187538A (de)
SE (1) SE7807690L (de)
ZA (1) ZA783273B (de)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2457279A2 (fr) * 1977-07-11 1980-12-19 Merrell Toraude & Co A-halogenomethylphenylalanines et leurs derives, utiles notamment pour traiter la maladie de parkinson ou un etat de psychose, et leur procede de preparation
EP0040150A1 (de) * 1980-05-09 1981-11-18 Merrell Toraude Et Compagnie Fluormethylierter Tyrosin-Methylester

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE3282T1 (de) * 1978-07-24 1983-05-15 Merck & Co. Inc. Alpha-difluormethyl-alpha-aminosaeuren und sie enthaltende pharmazeutische zusammensetzung.
FR2450247A1 (fr) * 1979-02-28 1980-09-26 Tamsir Ndike Wade Esters et acides aliphatiques a-amines b,b-difluores
IE49522B1 (en) * 1979-04-26 1985-10-16 Merrell Toraude & Co Alpha-halomethylaminoacids
ZA815807B (en) * 1980-08-23 1982-08-25 Merrell Toraude & Co Preparation of aminoacetonitrile derivatives
JP2022510425A (ja) * 2018-12-06 2022-01-26 センダ バイオサイエンシーズ, インコーポレイテッド パーキンソン病を治療するためのデカルボキシラーゼ阻害剤

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3046300A (en) * 1960-10-21 1962-07-24 Merck & Co Inc alpha-trifluoromethyloxyphenylalanines
IE47542B1 (en) * 1977-06-01 1984-04-18 Merck & Co Inc Di-and tri-fluoromethyl amino acids and amines,compositions and processes for preparing said compounds
FR2392958A1 (fr) * 1977-06-01 1978-12-29 Merck & Co Inc Nouveaux amino-acides fluores utiles comme medicament

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2457279A2 (fr) * 1977-07-11 1980-12-19 Merrell Toraude & Co A-halogenomethylphenylalanines et leurs derives, utiles notamment pour traiter la maladie de parkinson ou un etat de psychose, et leur procede de preparation
EP0040150A1 (de) * 1980-05-09 1981-11-18 Merrell Toraude Et Compagnie Fluormethylierter Tyrosin-Methylester

Also Published As

Publication number Publication date
ES478517A1 (es) 1979-07-16
GB2005659A (en) 1979-04-25
DK309378A (da) 1979-01-12
FR2397391B1 (de) 1981-02-20
SE7807690L (sv) 1979-01-12
ZA783273B (en) 1979-06-27
CH636846A5 (de) 1983-06-30
IE781167L (en) 1979-01-11
IL54913A0 (en) 1978-08-31
GB2005659B (en) 1982-02-17
DE2828738A1 (de) 1979-02-01
IT1105534B (it) 1985-11-04
NZ187538A (en) 1982-08-17
ES478516A1 (es) 1979-07-16
AU525684B2 (en) 1982-11-25
AU3731278A (en) 1980-01-03
NL7807454A (nl) 1979-01-15
FR2397391A1 (fr) 1979-02-09
IE46932B1 (en) 1983-11-02
JPS5484544A (en) 1979-07-05
IT7850230A0 (it) 1978-07-10
ES471595A1 (es) 1979-10-01
JPS6326101B2 (de) 1988-05-27

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: MERRELL TORAUDE ET CIE

Effective date: 19930731