BE867517A - Derives amines spiranniques, leur preparation et leur utilisation comme medicaments - Google Patents

Derives amines spiranniques, leur preparation et leur utilisation comme medicaments

Info

Publication number
BE867517A
BE867517A BE188062A BE188062A BE867517A BE 867517 A BE867517 A BE 867517A BE 188062 A BE188062 A BE 188062A BE 188062 A BE188062 A BE 188062A BE 867517 A BE867517 A BE 867517A
Authority
BE
Belgium
Prior art keywords
spirannic
preparation
amine derivatives
medicinal products
medicinal
Prior art date
Application number
BE188062A
Other languages
English (en)
French (fr)
Original Assignee
Sumitomo Chemical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sumitomo Chemical Co filed Critical Sumitomo Chemical Co
Publication of BE867517A publication Critical patent/BE867517A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/10Spiro-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Cardiology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
BE188062A 1978-02-13 1978-05-26 Derives amines spiranniques, leur preparation et leur utilisation comme medicaments BE867517A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP1577878A JPS54109983A (en) 1978-02-13 1978-02-13 Novel spiroamine derivative and its preparation

Publications (1)

Publication Number Publication Date
BE867517A true BE867517A (fr) 1978-09-18

Family

ID=11898262

Family Applications (1)

Application Number Title Priority Date Filing Date
BE188062A BE867517A (fr) 1978-02-13 1978-05-26 Derives amines spiranniques, leur preparation et leur utilisation comme medicaments

Country Status (13)

Country Link
US (1) US4233307A (xx)
JP (1) JPS54109983A (xx)
AT (1) AT356108B (xx)
AU (1) AU511735B2 (xx)
BE (1) BE867517A (xx)
CA (1) CA1092106A (xx)
CH (1) CH635841A5 (xx)
DE (1) DE2822227A1 (xx)
ES (1) ES470155A1 (xx)
FR (1) FR2442845A1 (xx)
IT (1) IT7849577A0 (xx)
NL (1) NL7805814A (xx)
SE (1) SE7805949L (xx)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4337260A (en) * 1981-09-10 1982-06-29 Yoshitomi Pharmaceutical Industries, Ltd. Imidazopyridine-spiro-piperidine compounds
IL96507A0 (en) * 1989-12-08 1991-08-16 Merck & Co Inc Nitrogen-containing spirocycles and pharmaceutical compositions containing them
AU680020B2 (en) * 1993-06-07 1997-07-17 Merck & Co., Inc. Spiro-substituted azacycles as neurokinin antagonists
WO1995027712A1 (fr) * 1994-04-07 1995-10-19 Cemaf Nouveaux derives de spiro[indole-pyrrolidine] agonistes melatoninergiques, leur procede de preparation et leur utilisation a titre de medicament
FR2724170B1 (fr) * 1994-09-02 1997-05-30 Cemaf Nouveaux derives de spiro(indole-pyrrolidine) agonistes de la melatonine, leur procede de preparation et leur utilisation a titre de medicament
US5607936A (en) * 1994-09-30 1997-03-04 Merck & Co., Inc. Substituted aryl piperazines as neurokinin antagonists
US5962462A (en) * 1996-12-13 1999-10-05 Merck & Co., Inc. Spiro-substituted azacycles as modulators of chemokine receptor activity
US6013652A (en) * 1997-12-04 2000-01-11 Merck & Co., Inc. Spiro-substituted azacycles as neurokinin antagonists
EP1426375A3 (en) * 1999-07-21 2004-12-15 AstraZeneca AB Analgesic spiroindole derivatives
GB0213715D0 (en) * 2002-06-14 2002-07-24 Syngenta Ltd Chemical compounds
AU2003268512A1 (en) * 2002-09-09 2004-03-29 Janssen Pharmaceutica N.V. Hydroxy alkyl substituted 1,3,8-triazaspiro[4.5]decan-4-one derivatives useful for the treatment of ORL-1 receptor mediated disorders
TW200621244A (en) * 2004-08-19 2006-07-01 Vertex Pharma Modulators of muscarinic receptors
US7786141B2 (en) * 2004-08-19 2010-08-31 Vertex Pharmaceuticals Incorporated Dihydrospiroindene modulators of muscarinic receptors
NZ555444A (en) * 2004-11-29 2011-01-28 Vertex Pharma Modulators of muscarinic receptors
AU2006252781A1 (en) * 2005-06-02 2006-12-07 Janssen Pharmaceutica, N.V. Novel 3-spirocyclic indolyl derivatives useful as ORL-1 receptor modulators
WO2007028638A1 (en) * 2005-09-09 2007-03-15 Euro-Celtique S.A. Fused and spirocycle compounds and the use thereof
EP1973543A2 (en) * 2005-12-22 2008-10-01 Vertex Pharmaceuticals Incorporated Modulators of muscarinic receptors
EP1988892A2 (en) 2006-02-22 2008-11-12 Vertex Pharmaceuticals Incorporated Modulators of muscarinic receptors
NZ570497A (en) * 2006-02-22 2011-09-30 Vertex Pharma Spiro condensed 4,4'-quinilino-piperidines derivatives as modulators of muscarinic receptors
EP2040706A2 (en) * 2006-06-29 2009-04-01 Vertex Pharmceuticals Incorporated Modulators of muscarinic receptors
AU2007284548A1 (en) * 2006-08-15 2008-02-21 Vertex Pharmaceuticals Incorporated Modulators of muscarinic receptors
EP2051715A2 (en) * 2006-08-18 2009-04-29 Vertex Pharmceuticals Incorporated Modulators of muscarinic receptors
EA200970517A1 (ru) * 2006-11-28 2009-12-30 Янссен Фармацевтика Н.В. Соли 3-(3-амино-2-(r)-гидроксипропил)-1-(4-фторфенил)-8-(8-метилнафталин-1-илметил)-1,3,8-триазаспиро[4,5]декан-4-она
JP5490677B2 (ja) * 2007-04-09 2014-05-14 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ 不安及び鬱病の処置のためのorl−1受容体リガンドとしての1,3,8−三置換−1,3,8−トリアザ−スピロ[4.5]デカン−4−オン誘導体
WO2008142859A1 (ja) * 2007-05-18 2008-11-27 Kowa Company, Ltd. 新規なスピロオキシインドール化合物及びこれを含有する医薬
EP2207549A1 (en) 2007-10-03 2010-07-21 Vertex Pharmceuticals Incorporated Modulators of muscarinic receptors
US11976067B2 (en) * 2022-01-18 2024-05-07 Maze Therapeutics, Inc. APOL1 inhibitors and methods of use

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3299075A (en) * 1964-03-12 1967-01-17 Smith Kline French Lab Spiro [3h-indole-3, 3'-pyrrolidine and piperidine] derivatives

Also Published As

Publication number Publication date
ES470155A1 (es) 1979-01-01
AT356108B (de) 1980-04-10
AU3616978A (en) 1979-11-22
AU511735B2 (en) 1980-09-04
CH635841A5 (de) 1983-04-29
SE7805949L (sv) 1979-08-14
JPS54109983A (en) 1979-08-29
FR2442845B1 (xx) 1981-07-24
FR2442845A1 (fr) 1980-06-27
NL7805814A (nl) 1979-08-15
ATA388878A (de) 1979-09-15
IT7849577A0 (it) 1978-05-26
CA1092106A (en) 1980-12-23
DE2822227A1 (de) 1979-08-16
US4233307A (en) 1980-11-11

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: SUMITOMO CHEMICAL CY LTD

Effective date: 19850526