BE866841A - Procede de preparation d'imidazoazines et -diazines substituees et leur utilisation - Google Patents
Procede de preparation d'imidazoazines et -diazines substituees et leur utilisationInfo
- Publication number
- BE866841A BE866841A BE187505A BE187505A BE866841A BE 866841 A BE866841 A BE 866841A BE 187505 A BE187505 A BE 187505A BE 187505 A BE187505 A BE 187505A BE 866841 A BE866841 A BE 866841A
- Authority
- BE
- Belgium
- Prior art keywords
- imidazoazines
- diazines
- substituted
- preparation
- Prior art date
Links
- -1 SUBSTITUTED Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/61—Halogen atoms or nitro radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Neurology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US05/796,958 US4166851A (en) | 1977-05-16 | 1977-05-16 | Certain imidazo(1,2a)pyridine derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BE866841A true BE866841A (fr) | 1978-11-09 |
Family
ID=25169498
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BE187505A BE866841A (fr) | 1977-05-16 | 1978-05-09 | Procede de preparation d'imidazoazines et -diazines substituees et leur utilisation |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US4166851A (en, 2012) |
| JP (1) | JPS53141292A (en, 2012) |
| BE (1) | BE866841A (en, 2012) |
| CH (1) | CH639662A5 (en, 2012) |
| DE (1) | DE2820938A1 (en, 2012) |
| DK (1) | DK180878A (en, 2012) |
| FR (1) | FR2391215A1 (en, 2012) |
| GB (1) | GB1601041A (en, 2012) |
| IE (1) | IE46882B1 (en, 2012) |
| IT (1) | IT1156737B (en, 2012) |
| LU (1) | LU79651A1 (en, 2012) |
| NL (1) | NL7804345A (en, 2012) |
| SE (1) | SE7804777L (en, 2012) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0006614A3 (en) * | 1978-06-27 | 1980-01-23 | Merck & Co. Inc. | Pyridyl- and imidazopyridyloxypropanolamines, process for preparing the same and pharmaceutical compositions containing the same |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4233301A (en) * | 1977-05-16 | 1980-11-11 | Merck & Co., Inc. | Novel imidazoazines and imidazodiazines |
| US4330543A (en) * | 1978-12-14 | 1982-05-18 | Merck & Co., Inc. | Imidazoazines and imidazodiazines |
| US4331679A (en) * | 1980-12-23 | 1982-05-25 | Merck Sharp & Dohme (I.A.) Corp. | (3-Aralkylamino-2-or-propoxy) heterocyclic compounds |
| US4442094A (en) * | 1980-12-23 | 1984-04-10 | Merck & Co., Inc. | (3-Aralkylamino-2-or-propoxy)heterocyclic compounds |
| US4349673A (en) * | 1980-12-23 | 1982-09-14 | Merck & Co., Inc. | Benzoxazines |
| US4656168A (en) * | 1980-12-23 | 1987-04-07 | Merck & Co., Inc. | (3-aralkylamino-2-or-propoxy)heterocyclic compounds in method of effecting bronchodilation |
| US4391806A (en) * | 1982-07-12 | 1983-07-05 | The Dow Chemical Company | Substituted tetrahydropyridazino-(1,6-A)benzimidazoles and use as bronchodilators |
| US4537889A (en) * | 1982-12-27 | 1985-08-27 | Eli Lilly And Company | Inotropic agents |
| US4636502A (en) * | 1982-12-27 | 1987-01-13 | Eli Lilly And Company | Methods of producing a positive inotropic effect or vasodilation by administration of 2-phenyl imidazo pyrimidines and pyrazines |
| RO87859B (ro) * | 1982-12-27 | 1985-12-31 | Eli Lilly And Company | Procedeu pentru prepararea unor derivati de inidazopirimidina pirezina si triazina |
| DE3446778A1 (de) * | 1984-12-21 | 1986-07-03 | Dr. Karl Thomae Gmbh, 7950 Biberach | Neue imidazoderivate, ihre herstellung und diese verbindungen enthaltende arzneimittel |
| GB8719368D0 (en) * | 1987-08-15 | 1987-09-23 | Wellcome Found | Heterocyclic compounds |
| PH27291A (en) * | 1989-01-31 | 1993-05-04 | Takeda Chemical Industries Ltd | Imidazolpyrimidazines their production and use |
| EP0440119A1 (en) * | 1990-01-31 | 1991-08-07 | Takeda Chemical Industries, Ltd. | Imidazopyridazine compounds, their production and use |
| US5244908A (en) * | 1990-07-30 | 1993-09-14 | Takeda Chemical Industries, Ltd. | Imidazopyridine derivatives and their pharmaceutical use |
| US5420133A (en) * | 1993-03-19 | 1995-05-30 | Merck & Co., Inc. | Quinazolinones substituted with phenoxyphenylacetic acid derivatives |
| DE10145457A1 (de) * | 2001-09-14 | 2003-04-03 | Basf Ag | Substituierte Imidazo[1,2-a]-5,6,7,8-tetrahydropyridin-8-one, Verfahren zu ihrer Herstellung, sowie deren Verwendung zur Herstellung von Imidazo[1,2,-a]pyridinen |
| US20070078136A1 (en) | 2005-09-22 | 2007-04-05 | Bristol-Myers Squibb Company | Fused heterocyclic compounds useful as kinase modulators |
| WO2010017047A1 (en) * | 2008-08-05 | 2010-02-11 | Merck & Co., Inc. | Therapeutic compounds |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR208397A1 (es) * | 1973-02-20 | 1976-12-27 | Ciba Geigy Ag | Procedimiento para la elaboracion de compuestos de 1-piridiloxi-2-hidroxi-3-amino-propano1-piraziniloxi-2-hidroxi-3-amino-propano y 1-pirimidiniloxi-2-hidroxi-3-amino-propan |
| CH614711A5 (en, 2012) * | 1975-04-08 | 1979-12-14 | Sandoz Ag | |
| US4071630A (en) * | 1975-04-08 | 1978-01-31 | Sandoz Ltd. | 1-Substituted-amino-3-(4-furo[3,2-c]pyridinyloxy)-2-propanols |
-
1977
- 1977-05-16 US US05/796,958 patent/US4166851A/en not_active Expired - Lifetime
-
1978
- 1978-04-24 NL NL7804345A patent/NL7804345A/xx not_active Application Discontinuation
- 1978-04-26 DK DK180878A patent/DK180878A/da not_active Application Discontinuation
- 1978-04-26 SE SE7804777A patent/SE7804777L/xx unknown
- 1978-05-08 IE IE923/78A patent/IE46882B1/en unknown
- 1978-05-09 BE BE187505A patent/BE866841A/xx not_active IP Right Cessation
- 1978-05-12 LU LU79651A patent/LU79651A1/xx unknown
- 1978-05-12 DE DE19782820938 patent/DE2820938A1/de not_active Ceased
- 1978-05-12 IT IT49338/78A patent/IT1156737B/it active
- 1978-05-12 CH CH522978A patent/CH639662A5/de not_active IP Right Cessation
- 1978-05-12 GB GB19246/78A patent/GB1601041A/en not_active Expired
- 1978-05-12 FR FR7814248A patent/FR2391215A1/fr active Granted
- 1978-05-16 JP JP5723378A patent/JPS53141292A/ja active Granted
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0006614A3 (en) * | 1978-06-27 | 1980-01-23 | Merck & Co. Inc. | Pyridyl- and imidazopyridyloxypropanolamines, process for preparing the same and pharmaceutical compositions containing the same |
Also Published As
| Publication number | Publication date |
|---|---|
| US4166851A (en) | 1979-09-04 |
| IT1156737B (it) | 1987-02-04 |
| SE7804777L (sv) | 1978-11-17 |
| GB1601041A (en) | 1981-10-21 |
| IE780923L (en) | 1978-11-16 |
| IT7849338A0 (it) | 1978-05-12 |
| JPS623153B2 (en, 2012) | 1987-01-23 |
| DE2820938A1 (de) | 1978-11-23 |
| CH639662A5 (de) | 1983-11-30 |
| NL7804345A (nl) | 1978-11-20 |
| FR2391215B1 (en, 2012) | 1981-12-11 |
| IE46882B1 (en) | 1983-10-19 |
| JPS53141292A (en) | 1978-12-08 |
| LU79651A1 (fr) | 1979-02-02 |
| FR2391215A1 (fr) | 1978-12-15 |
| DK180878A (da) | 1978-11-17 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| FR2449699B1 (fr) | Polyetherpolyamides et leur procede de preparation | |
| BE891094Q (fr) | N-benzoyl-n'-pyridyloxy-phenylurees et leur procede de preparation | |
| BE866226A (fr) | Procede pour la preparation de thymosine alpha1 et d'un analogue | |
| BE866841A (fr) | Procede de preparation d'imidazoazines et -diazines substituees et leur utilisation | |
| LU79597A1 (fr) | Procede de preparation de n-alkyl-n-acyl-thienamycines et leur utilisation | |
| BE869163A (fr) | Thioethers basiques et leur procede de preparation | |
| BE863872A (fr) | Steroides-11 beta-substitues et procede de leur preparation | |
| BE866957A (fr) | Procede de preparation d'homopolymerisats et de copolymerisats d'alpha-mono-olefines | |
| BE850855A (fr) | Procede de preparation d'homopolymeres et copolymeres d'alpha-mono-olefines | |
| BE865136A (fr) | Composes de 2-phenoxy-5-trifluoromethylpyridine et leur procede de preparation | |
| BE869074A (fr) | Diurethannes, leur procede de preparation et leur utilisation | |
| BE865805A (fr) | 1,2,3-thiadiazol-3-in-5-ylidene-urees, leur procede de preparation et leur utilisation | |
| FR2305416A1 (fr) | Procede de preparation de tricosene-(9) et d'heneicosene-(9) | |
| BE856220A (fr) | Polyether-polyureides et procede de leur preparation | |
| BE872294A (fr) | Procede de preparation de 3-iodorifamycine s et de 3-bromorifamycine s | |
| BE884286A (fr) | Acylurees, leur procede de preparation et leur utilisation | |
| BE885946A (fr) | Nouvelles pyridothienotriazines et leur procede de preparation | |
| BE857100A (fr) | Procede de preparation d'homopolymeres et de copolymeres d'&-mono-olefines | |
| BE878127A (fr) | Amides 1,2,3-triazolecarboxyliques, leur procede de preparation et leur utilisation | |
| BE884652R (fr) | Phenoxyalcoyl trialcoxysilanes et leur procede de preparation | |
| RO75387A (ro) | Procedeu pentru prepararea unor derivatidde 4"-aminooleandomicina | |
| BE858806A (fr) | Procede pour la preparation de glycol-aldehyde et d'ethylene-glycol | |
| BE867086A (fr) | Composes d'azacyclyle et procede pour leur preparation | |
| BE854237A (fr) | 1,2,3-thiadiazol-5-yl-urees, leur procede de preparation et leur utilisation | |
| RO78342A (ro) | Procedeu de preparare a unor imino-eteri de benztiazoline si benzoxazoline |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RE | Patent lapsed |
Owner name: MERCK & CO. INC. Effective date: 19850509 |