BE859987A - Nouvelles aza-8 purinones-6 - Google Patents
Nouvelles aza-8 purinones-6Info
- Publication number
- BE859987A BE859987A BE181957A BE181957A BE859987A BE 859987 A BE859987 A BE 859987A BE 181957 A BE181957 A BE 181957A BE 181957 A BE181957 A BE 181957A BE 859987 A BE859987 A BE 859987A
- Authority
- BE
- Belgium
- Prior art keywords
- purinones
- aza
- news
- news aza
- Prior art date
Links
- VTXJIDBQMAXDIY-QKBMRJQYSA-N C[C@H]1CN[C@]2(C[C@H]3O[C@]4(CC(=C)[C@H]5O[C@@](O)([C@H](O)[C@@H]6C[C@H]7O[C@@]8(CC[C@]9(CC=C[C@H](O9)\C=C\CCC(O)=O)O8)[C@H](C)C[C@H]7O6)[C@H](C)[C@H](O)[C@@H]5C)C[C@@H](C)C[C@@H](O4)[C@H]3O2)[C@@H](C)C1 Chemical compound C[C@H]1CN[C@]2(C[C@H]3O[C@]4(CC(=C)[C@H]5O[C@@](O)([C@H](O)[C@@H]6C[C@H]7O[C@@]8(CC[C@]9(CC=C[C@H](O9)\C=C\CCC(O)=O)O8)[C@H](C)C[C@H]7O6)[C@H](C)[C@H](O)[C@@H]5C)C[C@@H](C)C[C@@H](O4)[C@H]3O2)[C@@H](C)C1 VTXJIDBQMAXDIY-QKBMRJQYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Pulmonology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB44008/76A GB1561345A (en) | 1976-10-22 | 1976-10-22 | 8 - azapuring - 6 - ones |
Publications (1)
Publication Number | Publication Date |
---|---|
BE859987A true BE859987A (fr) | 1978-04-21 |
Family
ID=10431345
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE181957A BE859987A (fr) | 1976-10-22 | 1977-10-21 | Nouvelles aza-8 purinones-6 |
Country Status (15)
Country | Link |
---|---|
US (1) | US4167568A (cs) |
JP (1) | JPS5395993A (cs) |
AU (1) | AU510478B2 (cs) |
BE (1) | BE859987A (cs) |
CA (1) | CA1111027A (cs) |
CH (1) | CH628898A5 (cs) |
DE (1) | DE2747199A1 (cs) |
DK (1) | DK142766B (cs) |
GB (1) | GB1561345A (cs) |
HU (1) | HU180009B (cs) |
IE (1) | IE45810B1 (cs) |
LU (1) | LU78363A1 (cs) |
NL (1) | NL7711332A (cs) |
SE (1) | SE7711836L (cs) |
ZA (1) | ZA776258B (cs) |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8817651D0 (en) * | 1988-07-25 | 1988-09-01 | Smith Kline French Lab | Chemical compounds |
US5250534A (en) * | 1990-06-20 | 1993-10-05 | Pfizer Inc. | Pyrazolopyrimidinone antianginal agents |
GB9114760D0 (en) * | 1991-07-09 | 1991-08-28 | Pfizer Ltd | Therapeutic agents |
US5294612A (en) * | 1992-03-30 | 1994-03-15 | Sterling Winthrop Inc. | 6-heterocyclyl pyrazolo [3,4-d]pyrimidin-4-ones and compositions and method of use thereof |
BR9816155B1 (pt) | 1997-11-12 | 2010-07-27 | imidazotriazinonas 2-fenil-substituìdas como inibidores de fosfodiesterase, bem como medicamento e uso farmacêutico compreendendo as mesmas. | |
ATE348618T1 (de) * | 2001-05-09 | 2007-01-15 | Bayer Healthcare Ag | Neue verwendung von 2-(2-ethoxy-5-(4-methyl- piperazin-1-sulfonyl)-phenyl)-5-methyl-7-propyl 3h-imidazo(5,1-f)(1,2,4)triazin-4-on |
DE10232113A1 (de) | 2002-07-16 | 2004-01-29 | Bayer Ag | Vardenafil Hydrochlorid Trihydrat enthaltende Arzneimittel |
DE102005001989A1 (de) * | 2005-01-15 | 2006-07-20 | Bayer Healthcare Ag | Intravenöse Formulierungen von PDE-Inhibitoren |
DE102005009240A1 (de) * | 2005-03-01 | 2006-09-07 | Bayer Healthcare Ag | Arzneiformen mit verbesserten pharmakokinetischen Eigenschaften |
DE102005009241A1 (de) * | 2005-03-01 | 2006-09-07 | Bayer Healthcare Ag | Arzneiformen mit kontrollierter Bioverfügbarkeit |
KR20080056250A (ko) * | 2005-09-29 | 2008-06-20 | 바이엘 헬스케어 아게 | 비뇨기 장애의 치료를 위한 pde 억제제 및 이들의 조합 |
TWI845600B (zh) | 2019-01-24 | 2024-06-21 | 美商普羅米修斯生物科學股份有限公司 | Gpr35調節劑 |
WO2022020617A1 (en) * | 2020-07-23 | 2022-01-27 | Prometheus Biosciences, Inc. | Therapeutic agents targeting gpr35 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1421970A (en) * | 1973-06-12 | 1976-01-21 | May & Baker Ltd | 8-azapurin-6-one derivatives |
GB1493685A (en) * | 1970-12-15 | 1977-11-30 | May & Baker Ltd | 8-azapurinones |
US3819631A (en) * | 1970-12-15 | 1974-06-25 | May & Baker Ltd | Azapurinones |
US4052390A (en) * | 1973-06-12 | 1977-10-04 | May & Baker Limited | Azapurinones |
-
1976
- 1976-10-22 GB GB44008/76A patent/GB1561345A/en not_active Expired
-
1977
- 1977-10-14 NL NL7711332A patent/NL7711332A/xx not_active Application Discontinuation
- 1977-10-19 HU HU77MA2922A patent/HU180009B/hu unknown
- 1977-10-20 JP JP12634477A patent/JPS5395993A/ja active Pending
- 1977-10-20 ZA ZA00776258A patent/ZA776258B/xx unknown
- 1977-10-20 AU AU29911/77A patent/AU510478B2/en not_active Expired
- 1977-10-20 SE SE7711836A patent/SE7711836L/xx not_active Application Discontinuation
- 1977-10-20 IE IE2139/77A patent/IE45810B1/en unknown
- 1977-10-20 US US05/843,786 patent/US4167568A/en not_active Expired - Lifetime
- 1977-10-20 DK DK467177AA patent/DK142766B/da not_active IP Right Cessation
- 1977-10-20 DE DE19772747199 patent/DE2747199A1/de not_active Withdrawn
- 1977-10-21 CA CA289,249A patent/CA1111027A/fr not_active Expired
- 1977-10-21 CH CH1286877A patent/CH628898A5/fr not_active IP Right Cessation
- 1977-10-21 LU LU78363A patent/LU78363A1/xx unknown
- 1977-10-21 BE BE181957A patent/BE859987A/xx not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
CH628898A5 (fr) | 1982-03-31 |
DE2747199A1 (de) | 1978-04-27 |
DK467177A (cs) | 1978-04-23 |
SE7711836L (sv) | 1978-04-23 |
LU78363A1 (cs) | 1978-06-12 |
JPS5395993A (en) | 1978-08-22 |
HU180009B (en) | 1983-01-28 |
AU510478B2 (en) | 1980-06-26 |
DK142766B (da) | 1981-01-19 |
DK142766C (cs) | 1981-08-17 |
IE45810B1 (en) | 1982-12-01 |
CA1111027A (fr) | 1981-10-20 |
ZA776258B (en) | 1978-07-26 |
NL7711332A (nl) | 1978-04-25 |
IE45810L (en) | 1978-04-22 |
US4167568A (en) | 1979-09-11 |
AU2991177A (en) | 1979-04-26 |
GB1561345A (en) | 1980-02-20 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RE | Patent lapsed |
Owner name: MAY & BAKER LTD Effective date: 19841021 |