BE856464A - Nouveaux derives 16-acythio de l'acide fusidique, utiles notamment comme antimicrobiens et leur procede de preparation - Google Patents

Nouveaux derives 16-acythio de l'acide fusidique, utiles notamment comme antimicrobiens et leur procede de preparation

Info

Publication number
BE856464A
BE856464A BE179074A BE179074A BE856464A BE 856464 A BE856464 A BE 856464A BE 179074 A BE179074 A BE 179074A BE 179074 A BE179074 A BE 179074A BE 856464 A BE856464 A BE 856464A
Authority
BE
Belgium
Prior art keywords
acythio
antimicrobials
derivatives
useful
new
Prior art date
Application number
BE179074A
Other languages
English (en)
Original Assignee
Leo Pharm Prod Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Leo Pharm Prod Ltd filed Critical Leo Pharm Prod Ltd
Publication of BE856464A publication Critical patent/BE856464A/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
    • C07J41/0027—Azides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J13/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17
    • C07J13/007—Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17 with double bond in position 17 (20)
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/003—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring the S atom directly linked to a ring carbon atom of the cyclopenta(a)hydrophenanthrene skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J33/00—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J33/002—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J51/00—Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
BE179074A 1976-07-05 1977-07-04 Nouveaux derives 16-acythio de l'acide fusidique, utiles notamment comme antimicrobiens et leur procede de preparation BE856464A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB27921/76A GB1581335A (en) 1976-07-05 1976-07-05 16-s-acyl derivatives of fusidic acid

Publications (1)

Publication Number Publication Date
BE856464A true BE856464A (fr) 1978-01-04

Family

ID=10267438

Family Applications (1)

Application Number Title Priority Date Filing Date
BE179074A BE856464A (fr) 1976-07-05 1977-07-04 Nouveaux derives 16-acythio de l'acide fusidique, utiles notamment comme antimicrobiens et leur procede de preparation

Country Status (22)

Country Link
US (1) US4119717A (fr)
JP (1) JPS535152A (fr)
AT (1) AT354625B (fr)
AU (1) AU516152B2 (fr)
BE (1) BE856464A (fr)
CA (1) CA1100941A (fr)
DE (1) DE2730196A1 (fr)
DK (1) DK148390B (fr)
FI (1) FI58136C (fr)
FR (1) FR2357574A1 (fr)
GB (1) GB1581335A (fr)
GR (1) GR63210B (fr)
IE (1) IE45217B1 (fr)
IT (1) IT1083082B (fr)
LU (1) LU77683A1 (fr)
NL (1) NL7707221A (fr)
NZ (1) NZ184408A (fr)
PH (1) PH14058A (fr)
PT (1) PT66759B (fr)
SE (1) SE436752B (fr)
YU (1) YU165477A (fr)
ZA (1) ZA773739B (fr)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4162259A (en) * 1975-12-03 1979-07-24 Leo Pharmaceutical Products Ltd. A/S (Lovens Kemiske fabrik Produktionsaktienselskab) Fusidic acid derivatives
US4548922A (en) * 1983-06-06 1985-10-22 Beth Israel Hospital Drug administration
US4959358A (en) * 1983-06-06 1990-09-25 Beth Israel Hospital Assn. Drug administration
US4746508A (en) * 1983-06-06 1988-05-24 Beth Israel Hospital Assn. Drug administration
US4994439A (en) * 1989-01-19 1991-02-19 California Biotechnology Inc. Transmembrane formulations for drug administration
GB9518883D0 (en) * 1995-09-15 1995-11-15 Leo Pharm Prod Ltd Chemical compounds
MY140194A (en) * 2003-07-16 2009-11-30 Leo Pharma As Novel fusidic acid derivatives
AU2007299010B2 (en) * 2006-09-19 2013-01-31 Solvay Pharmaceuticals Gmbh Estratriene derivatives and their uses as 17beta-hydroxysteroid dehydrogenase inhibitors
PT106679B (pt) 2012-11-27 2015-03-25 Hovione Farmaciencia Sa Formulações tópicas de tetraciclinas, sua preparação e usos

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1490852A (en) * 1974-09-12 1977-11-02 Leo Pharm Prod Ltd Fusidic acid derivatives
GR60362B (en) * 1975-06-25 1978-05-19 Leo Pharm Prod Ltd Preparation process of new 16-ethers of fusidic acid derivatives
US4060606A (en) * 1975-06-25 1977-11-29 Leo Pharmaceutical Products Ltd. A/S 16-Ethers of fusidic acid derivatives

Also Published As

Publication number Publication date
FI58136B (fi) 1980-08-29
GR63210B (en) 1979-10-08
IE45217L (en) 1978-01-05
DE2730196A1 (de) 1978-01-19
IE45217B1 (en) 1982-07-14
FR2357574A1 (fr) 1978-02-03
FI772066A (fr) 1978-01-06
JPS535152A (en) 1978-01-18
DE2730196C2 (fr) 1987-03-05
AU516152B2 (en) 1981-05-21
AT354625B (de) 1979-01-25
FI58136C (fi) 1980-12-10
SE436752B (sv) 1985-01-21
PT66759A (en) 1977-08-01
US4119717A (en) 1978-10-10
LU77683A1 (fr) 1978-01-31
IT1083082B (it) 1985-05-21
JPS6238360B2 (fr) 1987-08-17
PH14058A (en) 1980-12-29
SE7707749L (sv) 1978-01-06
FR2357574B1 (fr) 1979-07-20
ATA455777A (de) 1979-06-15
YU165477A (en) 1982-06-30
ZA773739B (en) 1978-05-30
DK294177A (da) 1978-01-06
NZ184408A (en) 1980-04-28
NL7707221A (nl) 1978-01-09
AU2643877A (en) 1979-01-04
GB1581335A (en) 1980-12-10
DK148390B (da) 1985-06-24
PT66759B (en) 1978-12-14
CA1100941A (fr) 1981-05-12

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: LEO PHARMACEUTICAL PRODUCTS LTD A/S (LOVENS KEMIS

Effective date: 19860731