BE851278A - Preparations pharmaceutiques destinees a remedier a l'abus des stupefiants - Google Patents
Preparations pharmaceutiques destinees a remedier a l'abus des stupefiantsInfo
- Publication number
- BE851278A BE851278A BE174804A BE174804A BE851278A BE 851278 A BE851278 A BE 851278A BE 174804 A BE174804 A BE 174804A BE 174804 A BE174804 A BE 174804A BE 851278 A BE851278 A BE 851278A
- Authority
- BE
- Belgium
- Prior art keywords
- narcotics
- abuse
- remedy
- pharmaceutical preparations
- preparations intended
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Emergency Medicine (AREA)
- Psychiatry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Addiction (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US65699676A | 1976-02-11 | 1976-02-11 |
Publications (1)
Publication Number | Publication Date |
---|---|
BE851278A true BE851278A (fr) | 1977-08-10 |
Family
ID=24635439
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE174804A BE851278A (fr) | 1976-02-11 | 1977-02-10 | Preparations pharmaceutiques destinees a remedier a l'abus des stupefiants |
Country Status (13)
Country | Link |
---|---|
US (1) | US4126684A (fr) |
JP (1) | JPS5299228A (fr) |
AU (1) | AU515341B2 (fr) |
BE (1) | BE851278A (fr) |
CA (1) | CA1069050A (fr) |
DE (1) | DE2705051A1 (fr) |
FR (1) | FR2340727A1 (fr) |
GB (1) | GB1567543A (fr) |
IE (1) | IE44562B1 (fr) |
IL (1) | IL51415A (fr) |
NL (1) | NL7701494A (fr) |
PH (1) | PH13312A (fr) |
ZA (1) | ZA77773B (fr) |
Families Citing this family (49)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4457933A (en) * | 1980-01-24 | 1984-07-03 | Bristol-Myers Company | Prevention of analgesic abuse |
NL8006135A (nl) * | 1980-11-10 | 1982-06-01 | Univ Erasmus | Geneesmiddel met angst en angstequivalenten opheffende werking en werkwijze voor de bereiding van een dergelijk geneesmiddel. |
CH664085A5 (de) * | 1985-02-08 | 1988-02-15 | Ciba Geigy Ag | Pharmazeutische praeparate mit analgetischer wirksamkeit, sowie deren herstellung. |
GB8608818D0 (en) * | 1986-04-11 | 1986-05-14 | Reckitt & Colmann Prod Ltd | Pharmaceutical compositions |
IT1226800B (it) * | 1988-09-16 | 1991-02-19 | Prodotti Formenti | Composizioni farmaceutiche orali contenenti sali di destrorfano. |
FR2662354B1 (fr) * | 1990-05-23 | 1994-10-07 | Adir | Utilisation du baclofene pour l'obtention de medicaments destines au traitement de l'angine de poitrine. |
US5968551A (en) * | 1991-12-24 | 1999-10-19 | Purdue Pharma L.P. | Orally administrable opioid formulations having extended duration of effect |
US5321012A (en) * | 1993-01-28 | 1994-06-14 | Virginia Commonwealth University Medical College | Inhibiting the development of tolerance to and/or dependence on a narcotic addictive substance |
USRE39300E1 (en) | 1993-01-28 | 2006-09-19 | Virginia Commonwealth University Medical College Of Virginia | Inhibiting the development of tolerance to and/or dependence on an addictive substance |
US5914131A (en) * | 1994-07-07 | 1999-06-22 | Alza Corporation | Hydromorphone therapy |
US5529787A (en) * | 1994-07-07 | 1996-06-25 | Alza Corporation | Hydromorphone therapy |
US6375957B1 (en) | 1997-12-22 | 2002-04-23 | Euro-Celtique, S.A. | Opioid agonist/opioid antagonist/acetaminophen combinations |
ATE323491T1 (de) | 1997-12-22 | 2006-05-15 | Euro Celtique Sa | Peroral zu verabreichende arzneiform enthaltend eine kombination von einem opioid agonisten und naltrexon |
HU228771B1 (en) * | 1998-05-15 | 2013-05-28 | Warner Lambert Co | Stabilized pharmaceutical preparations of gamma-aminobutyric acid derivatives and process for preparing the same |
HU228772B1 (en) * | 1998-05-15 | 2013-05-28 | Warner Lambert Co | Gamma-aminobutyric acid derivatives containing, solid compositions and process for preparing the same |
IT1313585B1 (it) * | 1999-07-30 | 2002-09-09 | Neuroscienze S C A R L | Uso di agonisti dei recettori gabab per la terapia di mantenimentodell'astinenza da nicotina in soggetti nicotino-dipendenti. |
ATE493130T1 (de) | 2001-05-11 | 2011-01-15 | Endo Pharmaceuticals Inc | Opioid enthaltende arzneiform gegen missbrauch |
US20040033253A1 (en) * | 2002-02-19 | 2004-02-19 | Ihor Shevchuk | Acyl opioid antagonists |
ES2627298T3 (es) * | 2002-04-05 | 2017-07-27 | Mundipharma Pharmaceuticals S.L. | Preparación farmacéutica que contiene oxicodona y naloxona |
US20030199439A1 (en) * | 2002-04-22 | 2003-10-23 | Simon David Lew | Compositions of alpha3beta4 receptor antagonists and opioid agonist analgesics |
US7109239B2 (en) * | 2003-08-20 | 2006-09-19 | Xenoport, Inc. | Acyloxyalkyl carbamate prodrugs, methods of synthesis and use |
EP2354120A1 (fr) | 2003-08-20 | 2011-08-10 | XenoPort, Inc. | Synthèse de promédicaments a base de carbamate d'acyloxyalkyle et leurs intermédiaires |
AU2004311879B2 (en) * | 2003-12-31 | 2010-08-05 | Cima Labs Inc. | Effervescent oral opiate dosage form |
EP1604667A1 (fr) * | 2004-06-08 | 2005-12-14 | Euro-Celtique S.A. | Opioides pour le traitement des impatiences des membres inférieurs |
EP1604666A1 (fr) | 2004-06-08 | 2005-12-14 | Euro-Celtique S.A. | Opioides pour le traitement de la bronchopneumopathie chronique obstructive |
WO2006050471A2 (fr) | 2004-11-03 | 2006-05-11 | Xenoport, Inc. | Prodrogues d'acyloxyalkyl carbamate de l'acide 3-aminopropylsulfinique, et procedes de synthese et d'utilisation |
WO2006050472A2 (fr) * | 2004-11-03 | 2006-05-11 | Xenoport, Inc. | Prodrogues d'acyloxyalkyl carbamate, et leurs procedes de synthese et d'utilisation |
AP2274A (en) * | 2005-01-28 | 2011-08-19 | Euro Celtiques Sa | Alcohol resistant dosage forms. |
EP1702558A1 (fr) | 2005-02-28 | 2006-09-20 | Euro-Celtique S.A. | Procédé et dispositif pour évaluer la fonction de l'activité intestinale |
EP1695700A1 (fr) * | 2005-02-28 | 2006-08-30 | Euro-Celtique S.A. | Forme posologique contenant de l'oxycodone et de la naloxone |
WO2008033572A1 (fr) * | 2006-09-15 | 2008-03-20 | Xenoport, Inc. | Promédicaments à base de carbamate d'acyloxyalkyle, procédés de synthèse et utilisation |
ES2365574T3 (es) * | 2007-01-11 | 2011-10-07 | Xenoport, Inc. | Formas de dosificación oral para liberación continua de un profármaco de r-baclofeno y procedimientos de tratamiento. |
TW200936123A (en) * | 2007-11-06 | 2009-09-01 | Xenoport Inc | Use of prodrugs of GABAb agonists for treating neuropathic and musculoskeletal pain |
WO2009094577A2 (fr) | 2008-01-25 | 2009-07-30 | Xenoport, Inc. | Formes mésophasiques de précurseurs d'acide (3s)-aminométhyl-5-méthyl-hexanoïque et procédés d'utilisation |
US7872046B2 (en) * | 2008-01-25 | 2011-01-18 | Xenoport, Inc. | Crystalline form of a (3S)-aminomethyl-5-methyl-hexanoic acid prodrug and methods of use |
TWI380812B (zh) * | 2008-01-25 | 2013-01-01 | Xenoport Inc | (3s)-胺甲基-5-甲基己酸前藥之晶形及使用方法 |
US20100137442A2 (en) * | 2008-02-01 | 2010-06-03 | Xenoport, Inc. | Sustained Release Particulate Oral Dosage Forms of (R)-Baclofen and Methods of Treatment |
WO2010017504A1 (fr) * | 2008-08-07 | 2010-02-11 | Xenoport, Inc. | Procédés de synthèse de promédicaments de 1-(acyloxy)-alkylcarbamate |
US7989641B2 (en) | 2008-08-07 | 2011-08-02 | Xenoport, Inc. | Methods of synthesizing N-hydroxysuccinimidyl carbonates |
KR20110117216A (ko) | 2009-03-03 | 2011-10-26 | 제노포트 인코포레이티드 | R-바클로펜 전구약물의 서방형 경구 투약 형태 |
KR20110133602A (ko) | 2009-03-10 | 2011-12-13 | 유로-셀티큐 에스.에이. | 옥시코돈 및 날록손을 포함하는 즉시 방출 제약 조성물 |
CA2758245A1 (fr) * | 2009-04-17 | 2010-10-21 | Xenoport, Inc. | Derives d'acide gamma-aminobutyrique comme ligands des recepteurs gabab |
WO2013023155A1 (fr) | 2011-08-11 | 2013-02-14 | Xenoport, Inc. | Formes cristallines anhydres et hémihydratées d'un promédicament (r)-baclofène, procédés de synthèse et procédés d'utilisation |
JP2016525138A (ja) | 2013-07-23 | 2016-08-22 | ユーロ−セルティーク エス.エイ. | 疼痛および腸内ディスバイオシスをもたらす疾患および/または腸内細菌移行に対するリスクを高める疾患に罹患している患者における痛みの治療への使用のためのオキシコドンおよびナロキソンの組み合わせ |
JP6539274B2 (ja) | 2013-08-12 | 2019-07-03 | ファーマシューティカル マニュファクチュアリング リサーチ サービシズ,インコーポレーテッド | 押出成形された即放性乱用抑止性丸剤 |
WO2015095391A1 (fr) | 2013-12-17 | 2015-06-25 | Pharmaceutical Manufacturing Research Services, Inc. | Comprimé extrudé anti-abus à libération prolongée |
US9492444B2 (en) | 2013-12-17 | 2016-11-15 | Pharmaceutical Manufacturing Research Services, Inc. | Extruded extended release abuse deterrent pill |
JP6371463B2 (ja) | 2014-07-17 | 2018-08-08 | ファーマシューティカル マニュファクチュアリング リサーチ サービシズ,インコーポレーテッド | 即時放出性乱用抑止性液体充填剤形 |
US20160106737A1 (en) | 2014-10-20 | 2016-04-21 | Pharmaceutical Manufacturing Research Services, Inc. | Extended Release Abuse Deterrent Liquid Fill Dosage Form |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CH449645A (de) * | 1963-07-09 | 1968-01-15 | Ciba Geigy | Verfahren zur Herstellung neuer Aminosäuren |
US3773955A (en) * | 1970-08-03 | 1973-11-20 | Bristol Myers Co | Analgetic compositions |
-
1976
- 1976-12-08 US US05/748,591 patent/US4126684A/en not_active Expired - Lifetime
-
1977
- 1977-02-04 GB GB4685/77A patent/GB1567543A/en not_active Expired
- 1977-02-08 FR FR7703465A patent/FR2340727A1/fr not_active Withdrawn
- 1977-02-08 DE DE19772705051 patent/DE2705051A1/de not_active Withdrawn
- 1977-02-09 CA CA271,439A patent/CA1069050A/fr not_active Expired
- 1977-02-10 AU AU22171/77A patent/AU515341B2/en not_active Expired
- 1977-02-10 IL IL51415A patent/IL51415A/xx unknown
- 1977-02-10 PH PH19441A patent/PH13312A/en unknown
- 1977-02-10 JP JP1311077A patent/JPS5299228A/ja active Pending
- 1977-02-10 ZA ZA770773A patent/ZA77773B/xx unknown
- 1977-02-10 BE BE174804A patent/BE851278A/fr unknown
- 1977-02-10 IE IE280/77A patent/IE44562B1/en unknown
- 1977-02-11 NL NL7701494A patent/NL7701494A/xx not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
AU515341B2 (en) | 1981-04-02 |
DE2705051A1 (de) | 1977-08-18 |
ZA77773B (en) | 1977-12-28 |
NL7701494A (nl) | 1977-08-15 |
IE44562L (en) | 1977-08-11 |
PH13312A (en) | 1980-03-06 |
AU2217177A (en) | 1978-08-17 |
IL51415A (en) | 1979-11-30 |
IE44562B1 (en) | 1982-01-13 |
CA1069050A (fr) | 1980-01-01 |
GB1567543A (en) | 1980-05-14 |
IL51415A0 (en) | 1977-04-29 |
FR2340727A1 (fr) | 1977-09-09 |
JPS5299228A (en) | 1977-08-19 |
US4126684A (en) | 1978-11-21 |
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