BE841540A - Derives de 4-aroyl-4-hydroxy-piperidines 1-substituees utilisables comme medicaments neuroleptiques, produits intermediaires, et procedes pour leur prep aration - Google Patents

Derives de 4-aroyl-4-hydroxy-piperidines 1-substituees utilisables comme medicaments neuroleptiques, produits intermediaires, et procedes pour leur prep aration

Info

Publication number
BE841540A
BE841540A BE166802A BE166802A BE841540A BE 841540 A BE841540 A BE 841540A BE 166802 A BE166802 A BE 166802A BE 166802 A BE166802 A BE 166802A BE 841540 A BE841540 A BE 841540A
Authority
BE
Belgium
Prior art keywords
products
neuroleptic
aroyl
piperidines
substitutes
Prior art date
Application number
BE166802A
Other languages
English (en)
French (fr)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of BE841540A publication Critical patent/BE841540A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40Oxygen atoms
    • C07D211/44Oxygen atoms attached in position 4
    • C07D211/48Oxygen atoms attached in position 4 having an acyclic carbon atom attached in position 4
    • C07D211/50Aroyl radical
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Anesthesiology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
BE166802A 1975-05-07 1976-05-06 Derives de 4-aroyl-4-hydroxy-piperidines 1-substituees utilisables comme medicaments neuroleptiques, produits intermediaires, et procedes pour leur prep aration BE841540A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB19222/75A GB1535791A (en) 1975-05-07 1975-05-07 Derivatives of 4-piperidinol

Publications (1)

Publication Number Publication Date
BE841540A true BE841540A (fr) 1976-09-01

Family

ID=10125766

Family Applications (1)

Application Number Title Priority Date Filing Date
BE166802A BE841540A (fr) 1975-05-07 1976-05-06 Derives de 4-aroyl-4-hydroxy-piperidines 1-substituees utilisables comme medicaments neuroleptiques, produits intermediaires, et procedes pour leur prep aration

Country Status (16)

Country Link
US (1) US4021564A (xx)
JP (2) JPS52279A (xx)
AT (1) AT349017B (xx)
BE (1) BE841540A (xx)
CA (1) CA1086742A (xx)
CH (1) CH626880A5 (xx)
DE (1) DE2617955A1 (xx)
DK (1) DK196376A (xx)
ES (1) ES447677A1 (xx)
FI (1) FI60558C (xx)
FR (1) FR2310131A1 (xx)
GB (1) GB1535791A (xx)
LU (1) LU74891A1 (xx)
NL (1) NL7604833A (xx)
NO (1) NO147150C (xx)
SE (1) SE7605204L (xx)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4200641A (en) * 1976-12-21 1980-04-29 Janssen Pharmaceutica, N.V. 1-[(Heterocyclyl)-alkyl]-4-diarylmethoxy piperidine derivatives
US4366162A (en) * 1977-11-09 1982-12-28 Ab Ferrosan Aryl ethers of N-alkyl-piperidines and acid addition salts thereof
US4284636A (en) * 1979-09-04 1981-08-18 Richardson-Merrell Inc. Cinnamoylpiperidinobutyrophenone antipsychotic agents
US4283404A (en) * 1979-09-04 1981-08-11 Richardson-Merrell Inc. Aroylethenylpiperidinobutyrophenone antipsychotic agents
ZA806501B (en) * 1979-10-27 1981-10-28 Richardson Merrell Inc 4-(4-alkyl-aroyl-1-piperidino)butyrophenone antipsychotic agents
JPS59190739U (ja) * 1983-06-01 1984-12-18 田川 桂子 延反機における生地繰出し装置
US4654336A (en) * 1985-04-22 1987-03-31 Hoechst-Roussel Pharmaceuticals Inc. Ethanobenzazepines
US5057611A (en) * 1985-04-22 1991-10-15 Hoechst-Roussel Pharmaceuticals Inc. Benzoylpiperidines
FR2581993B1 (fr) * 1985-05-14 1988-03-18 Synthelabo Derives de (benzoyl-4 piperidino)-2 phenyl-1 alcanols, leur preparation et leur application en therapeutique
US5171557A (en) * 1991-05-28 1992-12-15 Ford Motor Company Method for silicon nitride precursor solids recovery
US20210108967A1 (en) * 2019-10-14 2021-04-15 Justin Thrash TempTech

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3029244A (en) * 1959-08-31 1962-04-10 Research Corp Aroylpiperidinols and esters thereof
GB895309A (en) * 1959-11-18 1962-05-02 Res Lab Dr C Janssen Nv Pyrrolidine and piperidine derivatives
GB963639A (en) * 1960-10-20 1964-07-15 Arnold Heyworth Beckett New piperidine derivatives and processes for preparing the same
DE2116316A1 (de) * 1970-04-08 1971-10-28 Sandoz Ag, Basel (Schweiz) Verfahren zur Herstellung neuer heterocyclischer Verbindungen
JPS4718878U (xx) * 1971-04-05 1972-11-02

Also Published As

Publication number Publication date
US4021564A (en) 1977-05-03
JPS5654316B2 (xx) 1981-12-24
DK196376A (da) 1976-11-08
ES447677A1 (es) 1977-06-16
JPS5436277A (en) 1979-03-16
SE7605204L (sv) 1976-11-08
CH626880A5 (xx) 1981-12-15
CA1086742A (en) 1980-09-30
FI60558C (fi) 1982-02-10
JPS5531148B2 (xx) 1980-08-15
NO147150C (no) 1983-02-09
AT349017B (de) 1979-03-12
NO761565L (xx) 1976-11-09
NO147150B (no) 1982-11-01
FR2310131A1 (fr) 1976-12-03
FR2310131B1 (xx) 1979-01-12
NL7604833A (nl) 1976-11-09
ATA332076A (de) 1978-08-15
GB1535791A (en) 1978-12-13
JPS52279A (en) 1977-01-05
LU74891A1 (xx) 1977-01-14
DE2617955A1 (de) 1976-11-18
FI60558B (fi) 1981-10-30
FI761093A (xx) 1976-11-08

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: A.B. FERROSAN

Effective date: 19850506