BE834247A - Nouveaux composes chimiques utiles en therapeutique humaine - Google Patents

Nouveaux composes chimiques utiles en therapeutique humaine

Info

Publication number
BE834247A
BE834247A BE160739A BE160739A BE834247A BE 834247 A BE834247 A BE 834247A BE 160739 A BE160739 A BE 160739A BE 160739 A BE160739 A BE 160739A BE 834247 A BE834247 A BE 834247A
Authority
BE
Belgium
Prior art keywords
chemical compounds
compounds useful
new chemical
human therapeutics
therapeutics
Prior art date
Application number
BE160739A
Other languages
English (en)
French (fr)
Inventor
Katsuu Arimura
Mitsuhiru Konishi
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of BE834247A publication Critical patent/BE834247A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56Nitrogen atoms
    • C07D211/58Nitrogen atoms attached in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BE160739A 1974-10-12 1975-10-06 Nouveaux composes chimiques utiles en therapeutique humaine BE834247A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP49117503A JPS5152176A (de) 1974-10-12 1974-10-12

Publications (1)

Publication Number Publication Date
BE834247A true BE834247A (fr) 1976-02-02

Family

ID=14713345

Family Applications (1)

Application Number Title Priority Date Filing Date
BE160739A BE834247A (fr) 1974-10-12 1975-10-06 Nouveaux composes chimiques utiles en therapeutique humaine

Country Status (7)

Country Link
JP (1) JPS5152176A (de)
AU (1) AU8564375A (de)
BE (1) BE834247A (de)
DE (1) DE2545501A1 (de)
FR (1) FR2287228A1 (de)
NL (1) NL7511857A (de)
SE (1) SE7511408L (de)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4203988A (en) 1975-11-12 1980-05-20 Merck & Co., Inc. Pyridinyl ureas and pharmaceutical use

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1561023A (en) * 1977-04-22 1980-02-13 Beecham Group Ltd 2-methoxy - 5 - chloro aniline derivatives
US4806552A (en) * 1980-03-01 1989-02-21 John Wyeth & Brother, Limited Pyridyl- and/or pyridoyl-(piperid-4-yl) ureas and analogues thereof
US4722930A (en) * 1980-03-01 1988-02-02 John Wyeth And Brother Limited 3-benzoyl-1-[(oxo or thioheteroaryl-ylalkyl)-piperid-4-yl]ureas and derivatives
NZ196324A (en) * 1980-03-01 1983-09-02 Wyeth John & Brother Ltd Piperidine derivatives and pharmaceutical compositions piperidine and pyridinium intermediates
FI95572C (fi) * 1987-06-22 1996-02-26 Eisai Co Ltd Menetelmä lääkeaineena käyttökelpoisen piperidiinijohdannaisten tai sen farmaseuttisen suolan valmistamiseksi
AUPP818099A0 (en) * 1999-01-14 1999-02-11 Fujisawa Pharmaceutical Co., Ltd. New n-containing heterocyclic compounds
FR2802206B1 (fr) * 1999-12-14 2005-04-22 Sod Conseils Rech Applic Derives de 4-aminopiperidine et leur utilisation en tant que medicament
US6476050B2 (en) 2000-03-14 2002-11-05 Sepracor, Inc. 3-substituted piperidines comprising urea functionality, and methods of use thereof
ES2314362T3 (es) 2003-01-16 2009-03-16 Acadia Pharmaceuticals Inc. Agonistas inversos selectivos de los receptores 2a o 2c de serotonina utilizados como agentes terapeuticos contra enfermedades neurodegenerativas.
US20050261278A1 (en) 2004-05-21 2005-11-24 Weiner David M Selective serotonin receptor inverse agonists as therapeutics for disease
US7820695B2 (en) 2004-05-21 2010-10-26 Acadia Pharmaceuticals, Inc. Selective serotonin receptor inverse agonists as therapeutics for disease
JP2010522198A (ja) 2007-03-19 2010-07-01 アカドイア プハルマセウチカルス インコーポレーテッド 5−ht2aインバースアゴニスト及びアンタゴニストの抗精神病薬との併用
SI3325444T1 (sl) 2015-07-20 2021-11-30 Acadia Pharmaceuticals Inc. Postopki za pripravo N-(4-fluorobenzil)-N-(1-metilpiperidin-4-il)-N'- (4-(2-metilpropiloksi)fenilmetil)karbamida in njegove tartratne soli in polimorfne oblike C
US10953000B2 (en) 2016-03-25 2021-03-23 Acadia Pharmaceuticals Inc. Combination of pimavanserin and cytochrome P450 modulators
WO2017165635A1 (en) 2016-03-25 2017-09-28 Acadia Pharmaceuticals Inc. Combination of pimavanserin and cytochrome p450 modulators
EP3558311A1 (de) 2016-12-20 2019-10-30 Acadia Pharmaceuticals Inc. Pimavanserin allein oder in kombination zur verwendung in der behandlung von morbus-alzheimer-psychose
WO2018200977A1 (en) 2017-04-28 2018-11-01 Acadia Pharmaceuticals Inc. Pimavanserin for treating impulse control disorder
EP3675827A1 (de) 2017-08-30 2020-07-08 Acadia Pharmaceuticals Inc. Formulierungen von pimavanserin
WO2024067304A1 (zh) * 2022-09-28 2024-04-04 瀚远医药有限公司 一种具有Sigma2和5HT2A抑制活性的化合物及用途

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4203988A (en) 1975-11-12 1980-05-20 Merck & Co., Inc. Pyridinyl ureas and pharmaceutical use

Also Published As

Publication number Publication date
NL7511857A (nl) 1976-04-14
FR2287228A1 (fr) 1976-05-07
AU8564375A (en) 1977-04-21
DE2545501A1 (de) 1976-04-22
SE7511408L (sv) 1976-04-13
JPS5152176A (de) 1976-05-08

Similar Documents

Publication Publication Date Title
BE834247A (fr) Nouveaux composes chimiques utiles en therapeutique humaine
KE2908A (en) Improvements in or relating to the processing of radiation-sensitive members
IT1047093B (it) Uretandossazolidine e procedimento per produrle
BR7500044A (pt) Aperfeicoamentos em oxigenador de sangue
IT977396B (it) Pila di misura per determinare la concentrazione dell ossigeno in miscugli gassosi
SE405447B (sv) Bubbelblodsyrsettare
IT1049058B (it) Composizione catalitica e procedimento per ottenerla
BE856636A (fr) Nouvelles 7-b-oxyiminoacylcephalosporines, leurs procedes de preparation et leurs applications en therapeutique
IT1051791B (it) Dispositivo per la codificazione in facsilile
IT1035815B (it) Perfezionamenti in scale o relativi ad esse
HK61978A (en) Improvements in or relating to radiograph
IT1051792B (it) Dispositivo per la codificazione in facsilile
AT339492B (de) Hautfeuchthaltemittel
NL7514448A (nl) 1-alkyl-2-(fenoxymethyl)-5-nitro-imidazolen en hun bereiding.
BE843931A (fr) Nouveaux composes chimiques et leurs applications en therapeutique cardio-vasculaire
FR2281746A1 (fr) Nouveaux composes chimiques et leur application en therapeutique humaine
AT336802B (de) Hautfeuchthaltemittel
TR18322A (tr) N-n-diallildikloroasetamid'in
IT1044466B (it) Procedimento e impianto per produrre polivimilcloruro in emulsione
NL7514580A (nl) In water onoplosbare disazomethineverbindingen en hun bereiding en toepassing.
IT1041179B (it) Composti alluminorganici e metodo per produrli
FR2291185A1 (fr) Preparation de polyols
BE826488A (fr) Nouveaux epoxydes utiles notamment en therapeutique
IT1028764B (it) Disposizione in apparecchi per la respirazione per comandare leafasi di respirazione
JPS5128345A (ja) In*rainhoshikihedoroshoriho