BE834247A - Nouveaux composes chimiques utiles en therapeutique humaine - Google Patents

Nouveaux composes chimiques utiles en therapeutique humaine

Info

Publication number
BE834247A
BE834247A BE160739A BE160739A BE834247A BE 834247 A BE834247 A BE 834247A BE 160739 A BE160739 A BE 160739A BE 160739 A BE160739 A BE 160739A BE 834247 A BE834247 A BE 834247A
Authority
BE
Belgium
Prior art keywords
chemical compounds
compounds useful
new chemical
human therapeutics
therapeutics
Prior art date
Application number
BE160739A
Other languages
English (en)
Inventor
Katsuu Arimura
Mitsuhiru Konishi
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of BE834247A publication Critical patent/BE834247A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56Nitrogen atoms
    • C07D211/58Nitrogen atoms attached in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)
BE160739A 1974-10-12 1975-10-06 Nouveaux composes chimiques utiles en therapeutique humaine BE834247A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP49117503A JPS5152176A (fr) 1974-10-12 1974-10-12

Publications (1)

Publication Number Publication Date
BE834247A true BE834247A (fr) 1976-02-02

Family

ID=14713345

Family Applications (1)

Application Number Title Priority Date Filing Date
BE160739A BE834247A (fr) 1974-10-12 1975-10-06 Nouveaux composes chimiques utiles en therapeutique humaine

Country Status (7)

Country Link
JP (1) JPS5152176A (fr)
AU (1) AU8564375A (fr)
BE (1) BE834247A (fr)
DE (1) DE2545501A1 (fr)
FR (1) FR2287228A1 (fr)
NL (1) NL7511857A (fr)
SE (1) SE7511408L (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4203988A (en) 1975-11-12 1980-05-20 Merck & Co., Inc. Pyridinyl ureas and pharmaceutical use

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1561023A (en) * 1977-04-22 1980-02-13 Beecham Group Ltd 2-methoxy - 5 - chloro aniline derivatives
US4806552A (en) * 1980-03-01 1989-02-21 John Wyeth & Brother, Limited Pyridyl- and/or pyridoyl-(piperid-4-yl) ureas and analogues thereof
US4722930A (en) * 1980-03-01 1988-02-02 John Wyeth And Brother Limited 3-benzoyl-1-[(oxo or thioheteroaryl-ylalkyl)-piperid-4-yl]ureas and derivatives
CA1173037A (fr) * 1980-03-01 1984-08-21 John L. Archibald Piperidine-urees utiles comme anti-depresseurs
FI95572C (fi) * 1987-06-22 1996-02-26 Eisai Co Ltd Menetelmä lääkeaineena käyttökelpoisen piperidiinijohdannaisten tai sen farmaseuttisen suolan valmistamiseksi
AUPP818099A0 (en) * 1999-01-14 1999-02-11 Fujisawa Pharmaceutical Co., Ltd. New n-containing heterocyclic compounds
FR2802206B1 (fr) * 1999-12-14 2005-04-22 Sod Conseils Rech Applic Derives de 4-aminopiperidine et leur utilisation en tant que medicament
WO2001068604A2 (fr) * 2000-03-14 2001-09-20 Sepracor, Inc. Piperidines 3-substituees comprenant un groupement uree et procedes d'utilisation de ces dernieres
KR101095939B1 (ko) 2003-01-16 2011-12-19 아카디아 파마슈티칼스 인코포레이티드 신경퇴행성 질환에 대한 치료제로서 선택적 세로토닌2a/2c 리셉터 역작용제
US20050261278A1 (en) 2004-05-21 2005-11-24 Weiner David M Selective serotonin receptor inverse agonists as therapeutics for disease
US7820695B2 (en) 2004-05-21 2010-10-26 Acadia Pharmaceuticals, Inc. Selective serotonin receptor inverse agonists as therapeutics for disease
DK2134330T3 (da) 2007-03-19 2013-08-05 Acadia Pharm Inc Kominationer af 5-ht2a-inverse agonister og antagonister med antipsykotika
PT3325444T (pt) 2015-07-20 2021-09-22 Acadia Pharm Inc Métodos para preparar n-(4-fluorobenzil)-n-(1-metilpiperidina-4-il)-n'-(4-(2-metilpropiloxi)fenilmetil)carbamida e o seu sal de tartarato e forma polimórfica c
US10953000B2 (en) 2016-03-25 2021-03-23 Acadia Pharmaceuticals Inc. Combination of pimavanserin and cytochrome P450 modulators
WO2017165635A1 (fr) 2016-03-25 2017-09-28 Acadia Pharmaceuticals Inc. Association de pimavansérine et de modulateurs du cytochrome p450
EP3558311A1 (fr) 2016-12-20 2019-10-30 Acadia Pharmaceuticals Inc. Pimavansérine seule ou en association pour une utilisation dans le traitement de la psychose liée à la maladie d'alzheimer
US11135211B2 (en) 2017-04-28 2021-10-05 Acadia Pharmaceuticals Inc. Pimavanserin for treating impulse control disorder
EP3675827A1 (fr) 2017-08-30 2020-07-08 Acadia Pharmaceuticals Inc. Formulations de pimavansérine
WO2024067304A1 (fr) * 2022-09-28 2024-04-04 瀚远医药有限公司 Composé à activité inhibitrice contre sigma2 et 5ht2a et utilisation

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4203988A (en) 1975-11-12 1980-05-20 Merck & Co., Inc. Pyridinyl ureas and pharmaceutical use

Also Published As

Publication number Publication date
FR2287228A1 (fr) 1976-05-07
NL7511857A (nl) 1976-04-14
JPS5152176A (fr) 1976-05-08
DE2545501A1 (de) 1976-04-22
SE7511408L (sv) 1976-04-13
AU8564375A (en) 1977-04-21

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