BE834247A - Nouveaux composes chimiques utiles en therapeutique humaine - Google Patents
Nouveaux composes chimiques utiles en therapeutique humaineInfo
- Publication number
- BE834247A BE834247A BE160739A BE160739A BE834247A BE 834247 A BE834247 A BE 834247A BE 160739 A BE160739 A BE 160739A BE 160739 A BE160739 A BE 160739A BE 834247 A BE834247 A BE 834247A
- Authority
- BE
- Belgium
- Prior art keywords
- chemical compounds
- compounds useful
- new chemical
- human therapeutics
- therapeutics
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/56—Nitrogen atoms
- C07D211/58—Nitrogen atoms attached in position 4
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP49117503A JPS5152176A (fr) | 1974-10-12 | 1974-10-12 |
Publications (1)
Publication Number | Publication Date |
---|---|
BE834247A true BE834247A (fr) | 1976-02-02 |
Family
ID=14713345
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE160739A BE834247A (fr) | 1974-10-12 | 1975-10-06 | Nouveaux composes chimiques utiles en therapeutique humaine |
Country Status (7)
Country | Link |
---|---|
JP (1) | JPS5152176A (fr) |
AU (1) | AU8564375A (fr) |
BE (1) | BE834247A (fr) |
DE (1) | DE2545501A1 (fr) |
FR (1) | FR2287228A1 (fr) |
NL (1) | NL7511857A (fr) |
SE (1) | SE7511408L (fr) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4203988A (en) | 1975-11-12 | 1980-05-20 | Merck & Co., Inc. | Pyridinyl ureas and pharmaceutical use |
Families Citing this family (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1561023A (en) * | 1977-04-22 | 1980-02-13 | Beecham Group Ltd | 2-methoxy - 5 - chloro aniline derivatives |
US4806552A (en) * | 1980-03-01 | 1989-02-21 | John Wyeth & Brother, Limited | Pyridyl- and/or pyridoyl-(piperid-4-yl) ureas and analogues thereof |
US4722930A (en) * | 1980-03-01 | 1988-02-02 | John Wyeth And Brother Limited | 3-benzoyl-1-[(oxo or thioheteroaryl-ylalkyl)-piperid-4-yl]ureas and derivatives |
CA1173037A (fr) * | 1980-03-01 | 1984-08-21 | John L. Archibald | Piperidine-urees utiles comme anti-depresseurs |
FI95572C (fi) * | 1987-06-22 | 1996-02-26 | Eisai Co Ltd | Menetelmä lääkeaineena käyttökelpoisen piperidiinijohdannaisten tai sen farmaseuttisen suolan valmistamiseksi |
AUPP818099A0 (en) * | 1999-01-14 | 1999-02-11 | Fujisawa Pharmaceutical Co., Ltd. | New n-containing heterocyclic compounds |
FR2802206B1 (fr) * | 1999-12-14 | 2005-04-22 | Sod Conseils Rech Applic | Derives de 4-aminopiperidine et leur utilisation en tant que medicament |
WO2001068604A2 (fr) * | 2000-03-14 | 2001-09-20 | Sepracor, Inc. | Piperidines 3-substituees comprenant un groupement uree et procedes d'utilisation de ces dernieres |
KR101095939B1 (ko) | 2003-01-16 | 2011-12-19 | 아카디아 파마슈티칼스 인코포레이티드 | 신경퇴행성 질환에 대한 치료제로서 선택적 세로토닌2a/2c 리셉터 역작용제 |
US20050261278A1 (en) | 2004-05-21 | 2005-11-24 | Weiner David M | Selective serotonin receptor inverse agonists as therapeutics for disease |
US7820695B2 (en) | 2004-05-21 | 2010-10-26 | Acadia Pharmaceuticals, Inc. | Selective serotonin receptor inverse agonists as therapeutics for disease |
DK2134330T3 (da) | 2007-03-19 | 2013-08-05 | Acadia Pharm Inc | Kominationer af 5-ht2a-inverse agonister og antagonister med antipsykotika |
PT3325444T (pt) | 2015-07-20 | 2021-09-22 | Acadia Pharm Inc | Métodos para preparar n-(4-fluorobenzil)-n-(1-metilpiperidina-4-il)-n'-(4-(2-metilpropiloxi)fenilmetil)carbamida e o seu sal de tartarato e forma polimórfica c |
US10953000B2 (en) | 2016-03-25 | 2021-03-23 | Acadia Pharmaceuticals Inc. | Combination of pimavanserin and cytochrome P450 modulators |
WO2017165635A1 (fr) | 2016-03-25 | 2017-09-28 | Acadia Pharmaceuticals Inc. | Association de pimavansérine et de modulateurs du cytochrome p450 |
EP3558311A1 (fr) | 2016-12-20 | 2019-10-30 | Acadia Pharmaceuticals Inc. | Pimavansérine seule ou en association pour une utilisation dans le traitement de la psychose liée à la maladie d'alzheimer |
US11135211B2 (en) | 2017-04-28 | 2021-10-05 | Acadia Pharmaceuticals Inc. | Pimavanserin for treating impulse control disorder |
EP3675827A1 (fr) | 2017-08-30 | 2020-07-08 | Acadia Pharmaceuticals Inc. | Formulations de pimavansérine |
WO2024067304A1 (fr) * | 2022-09-28 | 2024-04-04 | 瀚远医药有限公司 | Composé à activité inhibitrice contre sigma2 et 5ht2a et utilisation |
-
1974
- 1974-10-12 JP JP49117503A patent/JPS5152176A/ja active Pending
-
1975
- 1975-10-06 BE BE160739A patent/BE834247A/fr unknown
- 1975-10-09 NL NL7511857A patent/NL7511857A/xx unknown
- 1975-10-10 DE DE19752545501 patent/DE2545501A1/de active Pending
- 1975-10-10 SE SE7511408A patent/SE7511408L/xx unknown
- 1975-10-10 AU AU85643/75A patent/AU8564375A/en not_active Expired
- 1975-10-13 FR FR7531221A patent/FR2287228A1/fr not_active Withdrawn
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4203988A (en) | 1975-11-12 | 1980-05-20 | Merck & Co., Inc. | Pyridinyl ureas and pharmaceutical use |
Also Published As
Publication number | Publication date |
---|---|
FR2287228A1 (fr) | 1976-05-07 |
NL7511857A (nl) | 1976-04-14 |
JPS5152176A (fr) | 1976-05-08 |
DE2545501A1 (de) | 1976-04-22 |
SE7511408L (sv) | 1976-04-13 |
AU8564375A (en) | 1977-04-21 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
BE834247A (fr) | Nouveaux composes chimiques utiles en therapeutique humaine | |
HK74778A (en) | Improvements in or relating to the processing of radiation-sensitive members | |
IT1047093B (it) | Uretandossazolidine e procedimento per produrle | |
BR7500044A (pt) | Aperfeicoamentos em oxigenador de sangue | |
IT977396B (it) | Pila di misura per determinare la concentrazione dell ossigeno in miscugli gassosi | |
SE405447B (sv) | Bubbelblodsyrsettare | |
IT1049058B (it) | Composizione catalitica e procedimento per ottenerla | |
BE856636A (fr) | Nouvelles 7-b-oxyiminoacylcephalosporines, leurs procedes de preparation et leurs applications en therapeutique | |
IT1051791B (it) | Dispositivo per la codificazione in facsilile | |
IT1035815B (it) | Perfezionamenti in scale o relativi ad esse | |
HK61978A (en) | Improvements in or relating to radiograph | |
IT1051792B (it) | Dispositivo per la codificazione in facsilile | |
AT339492B (de) | Hautfeuchthaltemittel | |
NL7514448A (nl) | 1-alkyl-2-(fenoxymethyl)-5-nitro-imidazolen en hun bereiding. | |
BE843931A (fr) | Nouveaux composes chimiques et leurs applications en therapeutique cardio-vasculaire | |
FR2281746A1 (fr) | Nouveaux composes chimiques et leur application en therapeutique humaine | |
AT336802B (de) | Hautfeuchthaltemittel | |
TR18322A (tr) | N-n-diallildikloroasetamid'in | |
IT1044466B (it) | Procedimento e impianto per produrre polivimilcloruro in emulsione | |
NL7514580A (nl) | In water onoplosbare disazomethineverbindingen en hun bereiding en toepassing. | |
IT1041179B (it) | Composti alluminorganici e metodo per produrli | |
FR2291185A1 (fr) | Preparation de polyols | |
BE826488A (fr) | Nouveaux epoxydes utiles notamment en therapeutique | |
IT1028764B (it) | Disposizione in apparecchi per la respirazione per comandare leafasi di respirazione | |
JPS5128345A (ja) | In*rainhoshikihedoroshoriho |